Patent Assignment
Reel/Frame 017636/0297
Merger
Recorded: 2006-05-18
Pages: 16
Assignor
MERRELL PHARMACEUTICALS INC.
Executed: 2005-10-27
Assignee
AVENTIS INC.
300 SOMERSET CORPORATE BLVD., BRIDGEWATER, NEW JERSEY, 08807
Covered Properties
(241)
Process for Preparing 2,6-Di-Tertiarybutyl-4-Mercaptophenol
Patent:
4,734,527 →
Application:
06/920,813 →
4-Hydroxy-4-(Substituted Alkenyl)Cyclohexanecarboxylic Acids
Patent:
4,748,274 →
Application:
06/928,759 →
2-Chloro-4-((Cyanomethyl)Thio)Phenyl N-Methyl Carbamate for Treating Carcinomas
Patent:
4,804,682 →
Application:
06/930,838 →
Medroxalol Intermediates
Patent:
4,697,024 →
Application:
06/933,821 →
Medroxalol Intermediates
Patent:
4,701,541 →
Application:
06/933,825 →
Process for Preparing 2,6-Di-Tertiarybutyl-4-Mercaptophenol and 4,4' -Isopropylidenedithio-Bis-(2,6-Di-Tertiarybutylphenol) by Electrocatalysis
Patent:
4,772,363 →
Application:
07/003,115 →
Cycloalkane(1,2-C:4,3-C')Dipyrazoles and Their Use as Bronchodilators
Patent:
4,734,429 →
Application:
07/007,304 →
Dipyrazoles and Their Use as Bronchodilators
Patent:
4,734,430 →
Application:
07/007,305 →
Thiopyranodipyrazoles and Their Use as Bronchodilators
Patent:
4,734,431 →
Application:
07/007,308 →
Beta-(Fluoromethylene)-5-Hydroxytryptophan and Derivatives and Their Use as Prodrugs for Mao Inhibition
Patent:
4,822,812 →
Application:
07/053,212 →
Castanospermine for Inhibiting Tumor Metastasis
Patent:
4,792,558 →
Application:
07/055,589 →
Cardiotonic Tricyclic Imidazolones
Patent:
4,743,607 →
Application:
07/055,666 →
(Arylor Heteroaromatic Methyl)-2,2'-Bi-1H-Imidazoles and Their Use as Anti-Hypertensive Agents
Patent:
4,839,375 →
Application:
07/078,352 →
Heterocyclyl-2-Propyn-1-Amines
Patent:
4,743,617 →
Application:
07/091,338 →
Anti-Retroviral Castanospermine Esters
Patent:
5,004,746 →
Application:
07/102,070 →
3-Aryl-5-Alkylthio-4H-1,2,4-Triazoles
Patent:
4,900,743 →
Application:
07/126,191 →
Sulfhydryl Containing Tricyclic Lactams and Their Pharmacological Methods of Use
Patent:
4,824,832 →
Application:
07/139,485 →
Condtinuous Large-Scale Production of Ethyl 2,2,-Difluoro-4- Pentenoate and 2-Fluorinated Methyl Aninoacetonitriles by Use of a Flow Reactor
Patent:
4,847,401 →
Application:
07/145,694 →
Allenyl Amines
Patent:
4,847,288 →
Application:
07/153,106 →
Enhancement of Prazosin
Patent:
4,868,182 →
Application:
07/153,542 →
Cardiotonic Alkanoyl and Aroyl Oxazolones
Patent:
4,866,182 →
Application:
07/157,430 →
Novel Alkoxyimino Ether Derivatives of 5-Acyl-2(1H)-Pyridinones
Patent:
4,849,522 →
Application:
07/166,147 →
Adenosine Derivatives with Unsaturated Substitutions for the 5'- Hydroxymethyl Group
Patent:
4,996,308 →
Application:
07/173,782 →
Cardiotonic Tricyclic Oxazolones
Patent:
4,803,210 →
Application:
07/183,537 →
Process for Preparing 4,4'- Isopropylidenedithio-Bis- (2,6-Di-Tertiarybutylphenol) by Electrocatalysis
Patent:
4,861,443 →
Application:
07/209,763 →
19-Substituted Progesterone Derivatives Useful as 19-Hydroxylase Inhibitors
Patent:
4,910,191 →
Application:
07/212,409 →
19-Fluoro-Or Cyano- 21-Hydroxyprogesterone Derivatives Useful as 19-Hydroxylase Inhibitors
Patent:
4,920,114 →
Application:
07/212,410 →
Novel Chemical Compounds
Patent:
4,912,117 →
Application:
07/219,415 →
Aromatic 2-Aminoalkyl-1,2-Benzoisothiazol-3(2H)-One-1,1-Dioxide Derivatives
Patent:
4,857,526 →
Application:
07/244,894 →
Synthesis of Intermediate Useful in the Preparation of Nojirimycin and Related Compounds
Patent:
4,908,439 →
Application:
07/245,848 →
Substituted Imidazo(2,1-B)Quinazolin-5(3H)-Ones and Related Tricyclic Compounds and Use as Bronchodilators
Patent:
4,871,732 →
Application:
07/247,797 →
Imidazole Antiarrhythmics
Patent:
4,868,194 →
Application:
07/248,768 →
1,4-Disubstituted-Piperidinyl Compounds Useful as Analgesis and Muscle Relaxants
Patent:
4,870,083 →
Application:
07/254,208 →
Antihistaminic Piperidinyl Benzimidazoles
Patent:
4,908,372 →
Application:
07/256,959 →
Treatment of Fibromyalgia
Patent:
4,877,798 →
Application:
07/262,168 →
Use of Beta-(Fluoromethylene)-5-Hydroxytryptophan and Derivatives as Prodrugs for Mao Inhibition
Patent:
4,879,305 →
Application:
07/278,904 →
Hypocholesterolemic and Antiatherosclerotic Uses of Bis(3,5-Di-Tertiary-Butyl-4-Hydroxyphenylthio)Methane
Patent:
4,900,757 →
Application:
07/281,433 →
Use of 1,4-Disubstituted-Piperidinyl Compounds in the Manufacture of a Medicament for the Treatment of Insomnia
Patent:
4,908,369 →
Application:
07/299,913 →
5-Substituted Ornithine Derivatives
Patent:
4,902,719 →
Application:
07/305,247 →
Novel Alkoxyimino Ether Derivatives of 5-Acyl-2(1H)-Pyridinones
Patent:
4,920,229 →
Application:
07/321,704 →
Pharmaceutical Composition for Piperidinoalkanol Derivatives
Patent:
4,929,605 →
Application:
07/325,254 →
Pharmaceutical Compositions for Piperidinoalkanol-Ibuprofen Combination
Patent:
4,999,226 →
Application:
07/344,183 →
Aromatic 2-Aminoalkyl-1,2-Benzoisothiazol-3-(2H)One-1,1-Dioxide and Their Use as Anxiolytic and Anti-Hypertensive Agents
Patent:
4,920,118 →
Application:
07/366,824 →
Esters of Hexahydro-8-Hydroxy-2,6-Methano-2H-Quinolizin-3(4H)-One and Related Compounds
Patent:
4,906,755 →
Application:
07/376,172 →
5'-Deoxy-5',5'-Dihalo-Adenosines and Purine Analogues
Patent:
4,997,925 →
Application:
07/380,068 →
Pharmaceutically Active 3-Heteroaryl-2-Fluoro-1-Olefins
Patent:
4,981,868 →
Application:
07/384,944 →
Process for the Preparation of Castanospermine Esters
Patent:
4,970,317 →
Application:
07/390,794 →
Novel Chemical Compounds for the Prophylactic Treatment of Migraine
Patent:
5,021,428 →
Application:
07/428,256 →
Hypocholesterolemic Use of Bis(3,5-Di-Tertiary-Butyl-4- Hydroxyphenylthio)Methane
Patent:
4,954,528 →
Application:
07/433,985 →
Antiretroviral Aryloxy Substituted Furan Ketones
Patent:
4,977,185 →
Application:
07/438,541 →
Pharmaceutical Composition for Piperidinoalkanol-Decongestant Combination
Patent:
4,996,061 →
Application:
07/438,966 →
5'DEOXY-4',5'-Unsaturated-5'-Substituted Adenosines
Patent:
4,997,924 →
Application:
07/445,892 →
Treatment of Tumors with Autologous Lak Cells, Interleukin-2 and an Ornithine Decarboxylase Inhibitor
Patent:
5,002,879 →
Application:
07/449,288 →
Process for the Preparation of Sulfhydryl Containing Tricyclic Lactams
Patent:
5,095,110 →
Application:
07/483,955 →
Process for the Preparation of Castanospermine
Patent:
5,066,807 →
Application:
07/492,507 →
Method of Inhibiting Interleukin-1 Release and Alleviating Interleukin-1 Mediated Conditions
Patent:
4,975,467 →
Application:
07/499,567 →
Hydroxymethyl-Indolizidines and Quinolizidines and Their Use as Alpha-Glucosidade I Inhibitors
Patent:
5,028,614 →
Application:
07/502,602 →
Anticoagulant Peptide Alcohols
Patent:
4,971,953 →
Application:
07/504,719 →
Medicament Compositions Derived from Quinolizine and Quinolizinone and Use Thereof
Patent:
5,011,846 →
Application:
07/527,676 →
Derivatives of 6-Aminooctahydroindolizinetriol
Patent:
5,079,254 →
Application:
07/532,522 →
Novel 2,6-Di-Alkyl-4-Silyl-Phenols as Antiatherosclerotic Agents
Patent:
5,155,250 →
Application:
07/548,052 →
Novel Antidepressants
Patent:
5,149,714 →
Application:
07/569,259 →
Isolation of Castanospermine and Its Use as an Antidiabetic Agent
Patent:
6,136,820 →
Application:
07/622,305 →
N-Aralkyl-Piperidine-Methanol Derivatives
Patent:
5,169,096 →
Application:
07/637,089 →
Polyamine Derivatives as Antineoplastic Agents
Patent:
5,109,024 →
Application:
07/652,953 →
Phenoxy-Heterocyclic Compounds
Patent:
5,134,154 →
Application:
07/665,108 →
8-Substituted Purines as Selective Adenosine Receptor Agents
Patent:
5,208,240 →
Application:
07/667,943 →
Phenoxy and Phenylthio, Amino Substituted Benzocycloalkane Derivatives in the Treatment and Prevention of Drug-Resistant Protozoal Infections
Patent:
5,134,168 →
Application:
07/668,390 →
2,19-Methyleneoxy and 2,19-Methylenethio Bridged Steroids as Aromatase and 19-Hydroxylase Inhibitors
Patent:
5,099,037 →
Application:
07/674,640 →
Intermediates in a Process for the Preparation of Castanospermine
Patent:
5,093,501 →
Application:
07/712,780 →
Method for the Production of (-) 2-Difluormethyl-Ornithine
Patent:
5,217,886 →
Application:
07/722,042 →
(+)-Alpha-(2,3-Dimethoxyphenyl)-1-(2-(4-Fluorophenyl)Ethyl)-4- Piperidinemethanol
Patent:
5,134,149 →
Application:
07/736,194 →
Certain Pharmaceutically Active 6H-Imidazo(1,2-A)Pyridine-5-Ones
Patent:
5,109,006 →
Application:
07/750,758 →
Novel Azadecalin Amides and Thioamides as Inhibitors of Cholesterol Biosynthesis
Patent:
5,278,171 →
Application:
07/776,143 →
3-Amidoindolyl Derivatives and Pharmaceutical Compositions Thereof
Patent:
5,189,054 →
Application:
07/795,572 →
Pharmaceutical Lozenges
Patent:
5,322,694 →
Application:
07/847,856 →
Superior Tasting Composition Having Porous Particles and the Process of Preparing Such Pharmaceutical Composition
Patent:
5,302,396 →
Application:
07/884,299 →
Calcium Uptake Inhibitors
Patent:
5,248,825 →
Application:
07/892,440 →
S-Adenosyl Methionine Decarboxylase Inhibitors
Patent:
5,416,076 →
Application:
07/896,733 →
Novel Amino and Nitro Containing Tricyclic Compounds Useful as Inhibitors of Ace
Patent:
5,208,230 →
Application:
07/905,494 →
Cyclic Nitrones, Pharmaceutical Compositons Thereof and Their Use in Treating Shock.
Patent:
5,292,746 →
Application:
07/926,109 →
Novel Bis[4-(2,6-Di-Alkylypheno]Silane Derivatives as Antiatherosclerotic Agents
Patent:
5,281,738 →
Application:
07/939,561 →
1,4 Benzodioxin Derivatives and Their Use as Serotinin 5TH1A Agonists
Patent:
5,387,604 →
Application:
07/962,434 →
Anticoagulant Peptides
Patent:
5,232,912 →
Application:
07/970,596 →
Piperidyl Sulfonamides and Sulfoxamides as Inhibitors of Cholesterol Biosynthesis
Patent:
5,350,758 →
Application:
07/993,497 →
Controlled Release Formulation for Pharmaceutical Compounds
Patent:
5,320,853 →
Application:
07/995,309 →
Calcuim Uptake Inhibitors
Patent:
5,409,942 →
Application:
08/027,305 →
Neuropeptide Y Agonists and Partial Agonists
Patent:
5,395,823 →
Application:
08/032,526 →
Process for the Production of 2-Imidazolones
Patent:
5,338,862 →
Application:
08/039,539 →
Novel Amino and Nitro Containing Tricyclic Compounds Useful as Inhibitors of Ace
Patent:
5,308,841 →
Application:
08/046,326 →
Alpha-Mannosidase and Fucosidase Inhibitors
Patent:
5,382,709 →
Application:
08/075,984 →
Novel Bis[4-(2,6-Di-Alkyl)Phenol]Silane Derivatives as Antiatherosclerotic Agents
Patent:
5,304,668 →
Application:
08/077,619 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Tricyclic Derivatives Useful as Inhibitors of Enkephalinase
Patent:
5,420,271 →
Application:
08/078,787 →
Novel Difluoro Statone Analogs
Patent:
5,559,140 →
Application:
08/081,368 →
Process for Preparing 2,6-Di-Tertiarybutyl-4-Mercaptophenol and 4,4'-Isopropylidenedithio-Bis-(2,6-Di-Tertiarybutylphenol)
Patent:
5,401,883 →
Application:
08/088,462 →
Method for Producing an Orexigenic Effect
Patent:
5,352,686 →
Application:
08/097,097 →
5-Aryl-4-Alkyl-3H-1,2,4-Triazole-3-Thiones Useful as Memory Enhancers
Patent:
5,331,002 →
Application:
08/105,693 →
Sulfonic Acid Derivatives in the Treatment of Viral Diseases
Patent:
5,359,131 →
Application:
08/106,311 →
Antiallergic Compounds
Patent:
5,380,731 →
Application:
08/108,786 →
2'-Halomethylidene Cytidine, Uridine and Guanosine Compounds and Their Pharmaceutical Compositions
Patent:
5,378,693 →
Application:
08/113,505 →
Serotonin Receptor Agents
Patent:
5,436,246 →
Application:
08/119,791 →
Novel Aminoacetylmercapto Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,424,425 →
Application:
08/119,924 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,428,158 →
Application:
08/146,646 →
Mercaptoacetylamido Pyridazo [1,2]Tyridazo[1,2]Pyridazine, Pyrazolo[1,2]Pyridazine, Pyridazol[1,2-a][1,2] Diazepine and Pyrazolol[1,2-a][1,2] Diazepine
Patent:
5,366,973 →
Application:
08/146,857 →
Novel Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,430,145 →
Application:
08/149,572 →
Calcium Uptake Inhibitors
Patent:
5,500,429 →
Application:
08/154,146 →
Heterocyclic-Nmda Antagonists
Patent:
5,470,844 →
Application:
08/159,913 →
Novel 2-Substituted Indane-2-Carboxyalkyl Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,457,196 →
Application:
08/163,235 →
Amino and Nitro Containing Tricycle Compounds Useful as Inhibitors of Ace
Patent:
5,389,628 →
Application:
08/164,047 →
Nmda Antagonists
Patent:
5,484,814 →
Application:
08/165,144 →
Cyclic Nitrones
Patent:
5,397,789 →
Application:
08/170,543 →
Nmda Antagonists
Patent:
5,360,814 →
Application:
08/187,353 →
Arylalkoxyphenoxy-Imidazoline Compounds
Patent:
5,407,954 →
Application:
08/194,137 →
Polyfluorinated Tripeptide Thrombin Inhibitors
Patent:
5,391,705 →
Application:
08/199,039 →
Piperidinyl Thiacyclic Derivatives
Patent:
5,371,093 →
Application:
08/201,149 →
Method of Using 4-Amino- Steroids in the Treatment of Benign Prostatic Hyperplasia
Patent:
5,436,237 →
Application:
08/201,878 →
Selective Adenosine Receptor Agents
Patent:
5,391,739 →
Application:
08/207,338 →
Treatment of Obsessive-Compulsive Disorders with 5-HT2 Antagonists
Patent:
5,618,824 →
Application:
08/209,084 →
Novel Polyamine Derivatives
Patent:
5,753,714 →
Application:
08/213,386 →
Carbocyclic Adenosine Analogs Useful as Immunosuppressants
Patent:
5,514,688 →
Application:
08/241,814 →
Novel Peptidase Inhibitors
Patent:
5,496,927 →
Application:
08/248,847 →
Novel Triaryl-Ethylene Derivatives
Patent:
5,525,633 →
Application:
08/259,797 →
5'-Vinylhalo-Aristeromycin/Adenosine Analogs as Immunosuppressants
Patent:
5,470,837 →
Application:
08/260,617 →
Nmda Antagonists
Patent:
5,470,870 →
Application:
08/261,609 →
Novel Substituted Alkyldiamine Derivatives
Patent:
5,597,845 →
Application:
08/262,209 →
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Patent:
6,242,606 →
Application:
08/275,685 →
1-Piperidinyl Alkanoylanyl Sulfonamides for Treatment of Cardiac Arrhythmia.
Patent:
5,478,846 →
Application:
08/279,623 →
2,6-Methano-2H-Quinolizin Derivative as 5-HT3-Receptor Antagonist
Patent:
5,508,287 →
Application:
08/290,792 →
Novel Amino and Nitro Containing Tricyclic Compounds Useful as Inhibitors of Ace
Patent:
5,468,745 →
Application:
08/292,638 →
1-Phenyl-3-Phenyl-2-Propyne-1-Ones as Calcium Uptake Inhibitors
Patent:
5,446,068 →
Application:
08/307,538 →
Cardioprotective Tocopherol Analogs
Patent:
5,500,444 →
Application:
08/313,657 →
Hydrazide Derivatives of 3,4-Dihydro-2H-1-Benzopyrans
Patent:
5,545,660 →
Application:
08/318,670 →
Cardioprotective Agents
Patent:
5,510,373 →
Application:
08/318,784 →
Novel Orally-Active Elastase Inhibitors
Patent:
5,478,811 →
Application:
08/323,418 →
Substituted Pyrrolidin-3-Yl-Alkyl-Piperidines
Patent:
5,635,510 →
Application:
08/332,027 →
9-Purinyl Phosphonic Acid Derivatives
Patent:
5,538,978 →
Application:
08/336,703 →
Novel Antidepressants
Patent:
5,561,152 →
Application:
08/350,236 →
Cyclic Nitrone Compounds Useful in Treating Stroke
Patent:
5,498,778 →
Application:
08/352,470 →
Novel 2,6-Di-Alkyl-4-SILY1-Phenols as Antiatherosclerotic Agents
Patent:
5,532,400 →
Application:
08/353,736 →
2'-Ethenylidene Cytidene, Uridine and Guanosine Derivatives
Patent:
5,616,702 →
Application:
08/362,366 →
Novel Process for Piperidine Derivatives
Patent:
5,631,375 →
Application:
08/369,234 →
(+)-Alpha-(2,3-Dimethoxyphenyl)-1-[2-(4-Fluorophenyl)Ethyl]-4- Piperidinemethanol
Patent:
5,561,144 →
Application:
08/372,694 →
3-Amidoindolyl Derivative
Patent:
5,491,153 →
Application:
08/372,710 →
Novel 9-N-Bicyclic Nuceoside Agents Useful as Selective Inhibitors of Proinflammatory Cytokines
Patent:
6,420,373 →
Application:
08/372,712 →
5H-Dibenzo (a,D) Cycloheptenes as Muscarinic Receptor Anyagonists
Patent:
5,508,280 →
Application:
08/380,472 →
Novel Acetylcholinesterase Inhibitors
Patent:
5,693,668 →
Application:
08/382,941 →
Novel Carbocyclic Nucleoside Agents Useful as Selective Inhibitors of Proinflammatory Cytokines
Novel 2-Substituted Indane-2-Mercaptoacetylamide Tricyclic Derivatives Useful as Inhibitors of Enkephalinase
Patent:
5,491,141 →
Application:
08/396,833 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Tricyclic Derivatives Useful as Inhibitors of Enkephalinase
Patent:
5,491,142 →
Application:
08/396,945 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,486,513 →
Application:
08/396,947 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,529,996 →
Application:
08/397,298 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Disulfide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,567,814 →
Application:
08/397,304 →
Novel Processes for Preparing (S)-4-Amino-Hepta-5,6-Dienoic Acid and Intermediates Thereof
Patent:
5,654,477 →
Application:
08/400,314 →
Novel Mercaptoacetylamide Bicyclic Lactam Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,635,502 →
Application:
08/406,979 →
Anticoagulant Peptides
Patent:
5,789,540 →
Application:
08/412,356 →
Novel Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,527,795 →
Application:
08/417,179 →
Novel Mercaptoacetylamide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,491,143 →
Application:
08/417,424 →
Process for the Preparation of Ribonucleotide Reductase Inhibitors
Patent:
5,589,587 →
Application:
08/419,315 →
Novel 2-Substituted Indane-2-Carboxyalkyl Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,591,739 →
Application:
08/423,675 →
Method of Effecting Immunosuppression by Administering Carbocyclic Adenosine Analogs
Patent:
5,631,258 →
Application:
08/427,937 →
Novel Process for Piperidine Derivatives
Patent:
5,675,009 →
Application:
08/431,587 →
Novel Process for Piperidine Derivatives
Patent:
5,644,061 →
Application:
08/432,487 →
Anticoagulant Peptides
Patent:
5,495,000 →
Application:
08/432,617 →
Novel Process for Piperidine Derivatives
Patent:
5,618,940 →
Application:
08/432,660 →
Novel Process for Piperidine Derivatives
Patent:
5,652,370 →
Application:
08/432,731 →
Novel Process for Piperidine Derivatives
Patent:
5,654,433 →
Application:
08/433,299 →
Novel Process for Piperidine Derivatives
Patent:
5,650,516 →
Application:
08/433,777 →
Novel Process for Piperidine Derivatives
Patent:
5,663,353 →
Application:
08/434,134 →
Process for the Preparation of Ribonucleotide Reductase Inhibitors
Patent:
5,508,393 →
Application:
08/439,536 →
3-(Indol-3-Yl)-Propenoic Acid Derivatives and Pharmaceutical Compositions Thereof
Patent:
5,519,048 →
Application:
08/441,911 →
Piperidinyl Thiacyclic Derivatives
Patent:
5,739,150 →
Application:
08/457,199 →
Cyclic Nitrones
Patent:
5,677,315 →
Application:
08/458,310 →
Cyclic Nitrones
Patent:
5,532,252 →
Application:
08/458,311 →
Cyclic Nitrones
Patent:
5,525,615 →
Application:
08/458,314 →
Cyclic Nitrones
Patent:
5,527,812 →
Application:
08/458,318 →
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Patent:
6,147,216 →
Application:
08/458,747 →
Antiarrhythmic Piperidin-1-Yl-2,2-Dialkylpropanone Arylsulfonamide Derivatives
Patent:
5,541,201 →
Application:
08/460,029 →
Nmda Antagonists
Patent:
5,606,063 →
Application:
08/462,406 →
(+)-Alpha-(2,3-Dimethoxyphenyl)-1-[2-(4-Flurophenyl)Ethyl]-4- Piperidinemethanol
Patent:
5,721,249 →
Application:
08/476,538 →
Substituted Pyrrolidin-3-Yl-Alkyl-Piperidines
Patent:
5,648,366 →
Application:
08/477,167 →
Novel Peptidase Inhibitors
Patent:
5,849,866 →
Application:
08/481,666 →
(+)-Alpha_(2,3-Dimethoxyphenyl)-1-[2-(4-Fluorophenyl)Ethyl]-4- Piperidinemethanol
Patent:
5,700,813 →
Application:
08/485,700 →
(+)-A-(2,3-Dimethoxyphenyl)-1-[2-(4-Fluorophenyl)Ethyl]-4- Piperidinemethanol
Patent:
5,700,812 →
Application:
08/485,701 →
Substituted Pyrrolidin-3-Yl-Alkyl-Piperidines
Patent:
5,661,160 →
Application:
08/487,375 →
Method of Treating a Neoplastic Disease State by Conjunctive Therapy with 2'-Fluoromethylidene Derivatives and Radiation or Chemotherapy
Patent:
5,595,979 →
Application:
08/495,720 →
Xanthine Derivatives as Adenosine A1 Receptor Antagonists
Patent:
5,840,729 →
Application:
08/500,991 →
Nmda Antagonism Method
Patent:
5,547,991 →
Application:
08/502,980 →
Trifunctional Antithrombin and Antiplatelet Peptides
Patent:
5,681,925 →
Application:
08/502,989 →
Unsaturated Acetylene Phosphonate Derivatives of Purines
Patent:
5,817,647 →
Application:
08/505,168 →
3-Aminoindolyl Derivatives
Patent:
5,703,107 →
Application:
08/554,212 →
3-Amidoindolyl Derivatives
Patent:
5,675,018 →
Application:
08/554,621 →
Aromatic Acetylcholinesterase Inhibitors
Patent:
5,663,448 →
Application:
08/557,120 →
Novel Indane-2-Mercaptoacetylamide Disulfide Derivatives Useful as Inhibitors of Enkephalinase
Patent:
5,604,221 →
Application:
08/571,022 →
Novel 2-Substituted Indane-2-Mercaptoacetylamide Disulfide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,629,309 →
Application:
08/572,326 →
Difluoro Statone Analogs
Patent:
5,717,093 →
Application:
08/578,698 →
Novel Indole Derivatives Useful to Treat Estrogen-Related Neoplasms and Disorders
Patent:
5,877,202 →
Application:
08/594,505 →
Difluoro Statone Antiviral Analogs
Patent:
5,831,094 →
Application:
08/596,336 →
Stable Pharmaceutical Composition of Terfenadine and Ibuprofen
Patent:
5,691,352 →
Application:
08/624,362 →
Inhibitors of Beta-Amyloid Protein Production
Patent:
5,977,074 →
Application:
08/624,407 →
Heterocyclic Benzenesulfonylimine Derivatives as Inhibitors of Il-1 Action
Patent:
5,668,143 →
Application:
08/648,150 →
Acylated Enol Derivatives as Prodrugs of Elastase Inhibitors
Patent:
5,698,523 →
Application:
08/670,136 →
Novel Mercaptoacetylamido 1,3,4,5-Tetrahydro-Benzo[C]Azepin-3-One Disulfide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,731,306 →
Application:
08/673,250 →
Macrocyclic Difluorostatone Derivatives Useful as Antiviral Agents
Patent:
5,969,132 →
Application:
08/676,208 →
Neurokinin Receptor Cell Lines
Patent:
5,807,742 →
Application:
08/692,287 →
Perfluoroalkyl Ketone Inhibitors of Elastase and Processes for Making the Same
Patent:
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Application:
08/737,905 →
Novel 2'-Halomethylidene, 2'-Ethenylidene and 2'-Ethynl Cytidine, Uridine and Guanosine Derivatives
Patent:
5,792,841 →
Application:
08/744,652 →
Prolyl Endopeptidase Inhibitors
Patent:
5,661,167 →
Application:
08/759,323 →
(S)-4-Amino-Hepta-5,6-Dienoic Acid and Intermediates Therof
Patent:
5,756,762 →
Application:
08/781,566 →
Anti-Viral Compounds
Patent:
5,716,973 →
Application:
08/788,098 →
Substituted Pyrrolidin-3-Yl-Alkyl-Piperidines
Patent:
5,861,416 →
Application:
08/795,576 →
Substituted Pyrrolidin-3-Yl-Alkyl-Piperidines
Patent:
5,824,690 →
Application:
08/798,664 →
Cyclic Neurokinin a Antagonists
Patent:
5,731,286 →
Application:
08/811,913 →
Cyclic Antiplatelet Peptides with Pseudo-Bond
Patent:
6,107,275 →
Application:
08/835,274 →
Peptide Lung Surfactants and Therapeutic Combinations
Patent:
5,861,481 →
Application:
08/855,740 →
Acylated Enol Derivatives as Prodrugs of Elastase Inhibitors
Patent:
5,972,897 →
Application:
08/882,764 →
Novel Mercaptoacetylamino 1,3,4,5-Tetrahydro-Benzo(C)Azepin-2-One Disulefide Derivatives Useful as Inhibitors of Enkephalinase and Ace
Patent:
5,880,119 →
Application:
08/910,053 →
Process for the Production of Vinyl-Gaba
Patent:
6,090,979 →
Application:
08/912,770 →
Use of Certain Esters of Hexahydro-8-Hydroxy-2,6-METHAN0-2H- Quinolozin-3(4H)-One and Related Compounds for Treating Cognitive Disorders
Patent:
5,910,501 →
Application:
08/921,956 →
Difluoro Statone Analogs
Patent:
6,114,380 →
Application:
08/925,943 →
Treating Depression by Administering an Antidepressant
Patent:
5,880,120 →
Application:
08/937,224 →
(+) -@- (2,3-Dimethoxyphenyl)-1-(2-(4-Fluorephenyl) Ethyl)-4- Piepridinemethanol
Patent:
5,874,445 →
Application:
08/942,629 →
Compounds and Pharmaceutical Uses of Peptides of Bombesin and Grp
Patent:
5,834,433 →
Application:
08/960,130 →
Anticoagulant Peptides
Patent:
6,005,071 →
Application:
09/022,738 →
16 Unsaturated C17 Heterocyclic Steroids Useful as Steroid C17-20 Lyase Inhibitors
Patent:
5,965,548 →
Application:
09/072,778 →
Methods and Compositions Using Delta 16 Unsaturated C 17 Heterocyclic Steroids Useful as Steroid C 17-20 Lyase Inhibitors
Patent:
5,977,094 →
Application:
09/072,779 →
Difluoro Statone Antiviral Analogs
Patent:
5,948,778 →
Application:
09/081,307 →
Novel 2'-Halomethylidene, 2'-Ethenylidene and 2'-Ethynyl Cytidine, Uridine and Guanosine Derivatives
Patent:
5,977,325 →
Application:
09/089,839 →
Ethylenil and Allenic Phosphonate Derivatives of Purines
Patent:
5,922,696 →
Application:
09/131,761 →
Novel Peptidase Inhibitors
Patent:
6,130,315 →
Application:
09/139,009 →
Derivatives of Amide Analogs of Certain Methano Bridged Quinolizines
Patent:
5,955,470 →
Application:
09/181,888 →
(+)-A-(2,3-Dimethoxyphenyl)-1-[2-(4-Fluorophenyl) Ethyl}-4-Piperidinemethanol
Patent:
6,004,980 →
Application:
09/191,898 →
Novel Antid
Patent:
6,136,803 →
Application:
09/209,200 →
Novel Orally-Active Elastase Inhibitors
Patent:
6,265,381 →
Application:
09/491,814 →
Method of Providing an Antihistaminic Effect in a Hepatically Impaired Patient
Patent:
6,399,632 →
Application:
09/663,343 →
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
Patent:
6,340,761 →
Application:
09/725,298 →
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
Novel Intermediates Useful for the Preparation of Antihistaminic Piperidine Derivatives
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