IP Library Granted Patent US 12668793
Granted Patent B2
US 12668793 · App. 17/432,475 · Granted Jun 30, 2026

Sequential encoding methods and related kits

Inventor: Mark S. Chee (San Diego, CA)
Assignee: 2026 DF Peptide Acquisition LLC
C12N15/1065
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Quick Facts
Patent No.
US 12668793
App. No.
17/432,475
Granted
Jun 30, 2026
Kind
B2
Abstract

The present disclosure relates to methods and kits for analyzing a macromolecule. In some embodiments, the present disclosure relates to macromolecule analysis methods which employ barcoding and nucleic acid encoding of molecular recognition events. Also provided herein is a method and related kits for transferring information using a plurality of enzymes, including for performing a ligation, extension, and cleavage reaction with nucleic acid molecules associated with the macromolecule for analysis. In some embodiments, the macromolecule for analysis comprises a peptide, a polypeptide, or a protein.

Claims (21)

1 . A method for analyzing a macromolecule, comprising the steps of:

(a) providing a macromolecule and an associated recording tag joined to a support, wherein the recording tag comprises a double stranded region;

(b) contacting the macromolecule with a binding agent, wherein the binding agent comprises a coding tag with identifying information regarding the binding agent, wherein the binding agent binds to the macromolecule;

(c) covalently joining the 5′ end of the recording tag to the 3′end of the coding tag by a nucleic acid joining reagent;

(d) following (c), extending the recording tag using the coding tag as a template for a polymerase, thereby generating a double stranded extended recording tag; and

(e) cleaving both strands of the double stranded extended recording tag with a double strand nucleic acid cleaving reagent to generate a 3′ overhang in the extended recording tag, wherein a length of the 3′ overhang in the extended recording tag is less than 6 base pairs;

whereby information is transferred from the coding tag to the recording tag to generate the extended recording tag.

2 . The method of claim 1 , wherein in step (d), the double strand nucleic acid cleaving reagent recognizes a recognition sequence of the double stranded extended recording tag.

3 . The method of claim 1 , wherein the cleavage in step (e) releases the binding agent from the macromolecule.

4 . The method of claim 1 , wherein steps (b), (c), (d) and (e) are repeated sequentially one or more times in a cyclic manner.

5 . The method of claim 1 , wherein the macromolecule is a polypeptide.

6 . The method of claim 5 , wherein the polypeptide is obtained by fragmenting a protein from a biological sample.

7 . The method of claim 4 , further comprising removing a portion of the macromolecule prior to repeating step (b).

8 . The method of claim 5 , further comprising removing an N-terminal amino acid (NTAA) of the polypeptide to expose a new NTAA of the polypeptide prior to repeating step (b).

9 . The method of claim 4 , wherein the 3′ overhang of the extended recording tag generated by the double strand nucleic acid cleaving reagent in step (e) is available to hybridize with a second coding tag when step (b) is repeated.

10 . The method of claim 1 , wherein in step (b), the macromolecule is contacted with a plurality of binding agents, wherein the plurality of binding agents comprises the binding agent, and each binding agent of the plurality of binding agents comprises a coding tag with identifying information regarding the corresponding binding agent.

11 . The method of claim 5 , further comprising treating the polypeptide with a reagent for modifying a terminal amino acid of the polypeptide prior to step (b).

12 . The method of claim 1 , wherein the recording tag associated with the macromolecule comprises a nucleic acid hairpin.

13 . The method of claim 1 , wherein the nucleic acid joining reagent of step (c), the polymerase of step (d) and the double strand nucleic acid cleaving reagent of step (e) are provided simultaneously.

14 . The method of claim 1 , wherein the double strand nucleic acid cleaving reagent is a type IIS restriction enzyme.

15 . The method of claim 1 , further comprising analyzing one or more of the extended recording tags, wherein analyzing the extended recording tag(s) comprises a nucleic acid sequencing method.