IP Library Granted Patent US 12668822
Granted Patent B2
US 12668822 · App. 18/674,484 · Granted Jun 30, 2026

Multi-mechanistic channeling within a biocatalytic cascade for the production of 1,3-diaminopropane

Inventors: Shelby L. Hooe (Washington, DC); Igor L. Medintz (Washington, DC); Gregory A. Ellis (Washington, DC); Kimihiro Susumu (Hanover, MD); Tanya Tschirhart (Washington, DC)
Assignee: The Government of the United States of America, as represented by the Secretary of the Navy
C12P13/001B01J31/003B01J35/45C12N9/0008C12N9/1096C12N9/1217C12N9/88C12N11/18C12P5/02C12Y102/01011C12Y206/01076C12Y207/02004C12Y401/01086C12Y403/01001B82Y30/00B82Y40/00
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 12668822
App. No.
18/674,484
Granted
Jun 30, 2026
Kind
B2
Abstract

Described herein is a one-pot, four-enzyme cascade of enzymes, three bound to quantum dots with one enzyme free in solution, for the conversion in vitro of fumarate to 1,3-diaminopropane. The cascade operates via two distinctly different enzymatic channeling mechanisms which simultaneously function to increase the overall rate. The first three enzymes of the pathway (AspB->LysC->Asd) were able to engage in channeling in a nanoparticle displayed format, but addition of the last two enzymes to this pathway in this format (AspB->LysC->Asd->Dat->Ddc) did not result in complete channeling through the entire pathway to the final diaminopropane product. Surprisingly, replacement of the last two enzymes (Dat->Ddc) with a naturally occurring fused Dat-Ddc hybrid (Daba) provided for full channeling in this system (AspB->LysC->Asd->Daba).

Claims (7)

1 . A method of conducting a cascade reaction, comprising:

providing an enzymatic cascade comprising (1) metallic quantum dots (QDs) having a plurality of enzymes bound thereto, the plurality of enzymes comprising three enzymes comprising the amino acid sequences of SEQ ID NOs: 1, 2, and 3, respectively, and (2) a fourth enzyme comprising the amino acid sequence of SEQ ID NO: 6 not bound to the QDs;

contacting the enzymatic cascade with fumarate; and

allowing a reaction to proceed so that each of the plurality of enzymes acts in succession to produce 1,3-diaminopropane from the fumarate.

2 . The method of claim 1 , wherein the reaction is conducted in the presence of an enzyme comprising the amino acid sequence of SEQ ID NO: 7.

3 . An enzymatic cascade comprising (1) metallic quantum dots (QDs) having a plurality of enzymes bound thereto, the plurality of enzymes comprising three enzymes comprising the amino acid sequences of SEQ ID NOS: 1, 2, and 3, respectively, and (2) a fourth enzyme comprising the amino acid sequence of SEQ ID NO: 6 not bound to the QDs.

4 . The enzymatic cascade of claim 3 further comprising an enzyme comprising the amino acid sequence of SEQ ID NO: 7.