IP Library Granted Patent US 12681018
Granted Patent B2
US 12681018 · App. 17/873,828 · Granted Jul 14, 2026

Photoactive fluorescent compounds and use thereof for labeling of proteins

Inventors: Hilary Plake Beck (Emerald Hills, CA); David Trombley Mcswiggen (Berkeley, CA); Leah Brigit Cleary (Oakland, CA); Daniel James Anderson (Redwood City, CA); Yihong Li (San Bruno, CA); Anne Ruth Sizemore (Scranton, PA)
Assignee: EIKON THERAPEUTICS, INC.
G01N33/582C09B11/24C09B11/28C09K11/06C09K2211/1007C09K2211/1018
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Quick Facts
Patent No.
US 12681018
App. No.
17/873,828
Granted
Jul 14, 2026
Kind
B2
Abstract

Provided herein are novel photoactive fluorescent compounds of Formula (A) or a salt, a single stereoisomer, a mixture of stereoisomers or an isotopic form thereof, wherein G, R, X, Z, and L A are as defined herein, and their use in labeling proteins, for example, tagged proteins, comprising their use for visualizing the location and dynamics of proteins in living cells:

Claims (11)

1 . A compound, having a structure of Formula (IV):

wherein R 1 is —OH, —C(═O)OH, —C(═O)O(C 1-3 alkyl), —C(═O)N(C 1-3 alkyl) 2 , —N(C 1-3 alkyl) 2 , —(CH 2 ) n O(C 1-3 alkyl),

2 . The compound of claim 1 , wherein R 1 is —N(CH 3 ) 2 , —OH,

3 . The compound of claim 1 , having a structure of Formula (V):

4 . The compound of claim 2 , wherein R 1 is —N(CH 3 ) 2 , —OH,

5 . The compound of claim 1 , wherein the compound is:

6 . The compound of claim 1 , wherein the compound is:

7 . A compound having the following structure:

8 . A compound having the following structure:

9 . A compound having the following structure:

10 . A compound having the following structure: