IP Library Granted Patent US 12691124
Granted Patent B2
US 12691124 · App. 17/608,085 · Granted Jul 28, 2026

Methods of controlling and improving brain health

Inventors: Anne Schaefer (New York, NY); Josefa Sullivan (New York, NY); Alexander Tarakhovsky (Amagansett, NY); Uwe Schaefer (New York, NY); Tuo Zhang (New York, NY)
Assignees: Icahn School of Medicine at Mount Sinai; The Rockefeller University
A61K31/5517A61K31/437A61K31/444A61K31/4709A61K31/472A61K31/519A61K31/538A61K31/55A61K31/551A61P25/28
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Quick Facts
Patent No.
US 12691124
App. No.
17/608,085
Granted
Jul 28, 2026
Kind
B2
Abstract

The present disclosure relates to a method of inducing a neuroprotective state comprising administering a Bromodomain and Extra-Terminal motif (BET) inhibitor under conditions effective to induce a neuroprotective state. Also disclosed are methods of preventing and/or treating neurodegenerative disease, methods of reducing microglial inflammation, and methods of restoring microglial homeostasis, where the methods include administering a Bromodomain and Extra-Terminal motif (BET) inhibitor.

Claims (5)

1 . A method of treating Huntington's disease, the method comprising:

administering IBET858 to a subject in need thereof.

2 . The method of claim 1 , wherein IBET858 is administered in an amount between about 10 mg/kg and about 100 mg/kg.

3 . The method of claim 1 , wherein IBET858 is administered once daily for about 1 week.

4 . The method of claim 1 , wherein said administering is carried out intraperitoneally, orally, parenterally, nasally, subcutaneously, intravenously, intramuscularly, intracerebroventricularly, intraparenchymally, by inhalation, intranasal instillation, by implantation, by intracavitary or intravesical instillation, intraocularly, intraarterially, intralesionally, transdermally, topically, intradermally, intrapleurally, intrathecally, or by application to mucous membranes.