IP Library Granted Patent US 12691134
Granted Patent B2
US 12691134 · App. 17/829,801 · Granted Jul 28, 2026

Treatment of cerebrovascular disease with neurogenic locus notch homolog protein 3 (NOTCH3) agents

Inventors: Juan Rodriguez-Flores (Tarrytown, NY); Alan Shuldiner (Tarrytown, NY); Aris Baras (Tarrytown, NY); Danish Saleheen (Scarsdale, NY); Shareef Khalid (White Plains, NY)
Assignees: Regeneron Pharmaceuticals, Inc.; Center for Non-Communicable Diseases SMC Private Limited
A61K31/7105A61K38/465C12Q1/6883C12N15/1138C12Q2600/156
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Quick Facts
Patent No.
US 12691134
App. No.
17/829,801
Granted
Jul 28, 2026
Kind
B2
Abstract

The present disclosure provides methods of treating subjects having a cerebrovascular disease by administering Neurogenic Locus Notch Homolog Protein 3 (NOTCH3) agents, and methods of identifying subjects having an increased risk of developing a cerebrovascular disease.

Claims (5)

1 . A method of treating a subject having a subcortical stroke, an ischemic stroke, a hemorrhagic stroke, or a parenchymal stroke, the method comprising administering a Neurogenic Locus Notch Homolog Protein 3 (NOTCH3) agent to the subject, wherein the NOTCH3 agent comprises an inhibitory nucleic acid molecule, a small interfering RNA (siRNA), or a short hairpin RNA (shRNA) that hybridizes to a NOTCH3 nucleic acid molecule, and wherein the subject is heterozygous or homozygous for a NOTCH3 missense variant nucleic acid molecule encoding NOTCH3 Arg1231Cys, and wherein the subject has no family history of stroke.

2 . A method of treating a subject having a subcortical stroke, an ischemic stroke, a hemorrhagic stroke, or a parenchymal stroke, the method comprising:

detecting the presence or absence of a NOTCH3 missense variant nucleic acid molecule encoding a NOTCH3 predicted gain-of-function polypeptide in a biological sample obtained from the subject; and

administering a Neurogenic Locus Notch Homolog Protein 3 (NOTCH3) agent to the subject, wherein the NOTCH3 agent comprises an inhibitory nucleic acid molecule, a small interfering RNA (siRNA), or a short hairpin RNA (shRNA) that hybridizes to a NOTCH3 nucleic acid molecule,

wherein the subject is heterozygous or homozygous for a NOTCH3 missense variant nucleic acid molecule encoding NOTCH3 Arg1231Cys, and wherein the subject has no family history of stroke.