IP Library Granted Patent US 12692526
Granted Patent B2
US 12692526 · App. 17/769,998 · Granted Jul 28, 2026

Enzymatic synthesis of oligonucleotides

Inventors: Benjamin Allred (San Jose, CA); Handong Li (San Jose, CA)
Assignee: MGI Holdings Co., Limited
C12P19/34C12N9/1241C12Q1/6853
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Quick Facts
Patent No.
US 12692526
App. No.
17/769,998
Granted
Jul 28, 2026
Kind
B2
Abstract

Provided are compositions and methods directed to using a short template and a polymerase or ligase to synthesize an oligonucleotide. The template is designed such that only one nucleotide is added to the primer in each round of synthesis.

Claims (35)

1 . A method for synthesizing an oligonucleotide, comprising:

(a) providing a plurality of immobilized primers, wherein the 5′ terminus of each primer is attached to a solid support;

(b) combining the plurality of immobilized primers and

(i) a plurality of templates comprising between 2 and 100 nucleotides, wherein each template hybridizes to a primer generating a single overhang nucleotide at the 5′ terminus of the template;

(ii) a plurality of unincorporated nucleotides; and

(iii) a polymerase;

wherein the plurality of the immobilized primers are extended at the 3′ terminus by the polymerase-mediated incorporation of a single unincorporated nucleotide, wherein the single incorporated nucleotide is complementary to the single overhang nucleotide of the template hybridized to the primer; and then

(c) removing the hybridized templates and excess unincorporated nucleotides; and

(d) repeating steps (b) and (c) multiple times until the synthesis of the oligonucleotide is complete.

2 . The method of claim 1 , wherein the nucleotides in the plurality of nucleotides are 3′ protected nucleotides.

3 . The method of claim 2 , wherein the protective group of the 3′ protected nucleotides is selected from the group consisting of 3′-O-azidomethyl, 3′-O-allyl, 3′-O-methoxymethyl, 3′-O-nitrobenzyl, 3′-O-azidomethylene, and 3′-O-aminoalkoxyl.

4 . The method of claim 1 , wherein a solution comprising Ca 2+ is added prior to step (c) to prevent further elongation.

5 . The method of claim 4 , wherein the solution comprising Ca 2+ is removed in step (c) together with the plurality of templates and the excess nucleotides.

6 . The method of claim 5 , wherein a solution comprising Mg 2+ is added prior to step (d) to promote incorporation of the nucleotide to the 3′ terminus of the primer.

7 . The method of claim 1 , wherein the templates in the plurality of templates comprise between 5 and 50 nucleotides.

8 . The method of claim 1 , wherein the templates in the plurality of templates comprise between 5 and 20 nucleotides.

9 . The method of claim 1 , wherein the primers in the plurality of primers have the same sequence.

10 . The method of claim 9 , wherein the templates in the plurality of templates have the same sequence.

11 . The method of claim 1 , wherein at least two primers in the plurality of primers have different sequences.

12 . The method of claim 11 , wherein at least two templates in the plurality of templates have different sequences.

13 . A method for synthesizing an oligonucleotide, comprising:

(a) providing a plurality of immobilized primers, wherein the 5′ terminus of each primer is attached to a solid support;

(b) combining the plurality of immobilized primers and

(i) a plurality of hairpin templates comprising between 10 and 100 nucleotides, wherein each hairpin template comprises a phosphorothioate linkage between the two nucleotides at the 5′ terminus of each hairpin template, each hairpin template hybridizes to a primer, and the nucleotide at the 5′ terminus of the hairpin template is placed adjacent to the nucleotide at the 3′ terminus of the primer;

(ii) a ligase;

wherein the plurality of the immobilized primers are extended at the 3′ terminus by the ligase-mediated incorporation of the nucleotide at the 5′ terminus of the hairpin template; and then

(c) cleaving the phosphorothioate linkage;

(d) removing the plurality of hairpin templates;

(e) repeating steps (b) to (d) until the synthesis of the oligonucleotide is complete.

14 . The method of claim 13 , wherein cleaving the phosphorothioate linkage is performed by adding a solution of Ag + or Hg + .

15 . The method of claim 13 , wherein each hairpin template comprises at least one non-natural nucleotides.

16 . The method of claim 13 , wherein the primers in the plurality of primers have the same sequence.

17 . The method of claim 16 , wherein the hairpin templates in the plurality of hairpin templates have the same sequence.

18 . The method of claim 13 , wherein at least two primers in the plurality of primers have different sequences.

19 . The method of claim 18 , wherein at least two hairpin templates in the plurality of hairpin templates have different sequences.