IP Library Granted Patent US 12698499
Granted Patent B2
US 12698499 · App. 16/759,665 · Granted Aug 4, 2026

Identifying epigenetic and transcriptional targets to prevent and reverse T cell exhaustion

Inventors: E. John Wherry (Havertown, PA); Omar Khan (Philadelphia, PA); Martha Jordan (Wynnewood, PA)
Assignee: The Trustees of the University of Pennsylvania
C12N15/113A61K40/11A61K40/42A61K40/46C12N5/0636C12Q1/6883C12N2501/505C12Q2600/106C12Q2600/158
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Quick Facts
Patent No.
US 12698499
App. No.
16/759,665
Granted
Aug 4, 2026
Kind
B2
Abstract

The present invention provides methods of preventing, reversing or increasing T cell exhaustion in a patient having a disease. The present invention also provides methods for treating a disease in a patient having the disease. The present invention also provides an engineered T cell comprising a high priority epigenetic pathway that has been targeted, and uses thereof.

Claims (17)

1 . A method of making an improved cell therapy composition, comprising the steps of:

(a) obtaining a sample comprising lymphocytes from a subject;

(b) reducing or eliminating expression of one or more genes required for the induction and/or maintenance of exhausted CD8+ T lymphocytes (T EX ) in the lymphocytes; and

(c) engineering the lymphocytes to target a therapeutically relevant antigen;

wherein the one or more genes required for the induction and/or maintenance of T EX is a transcription factor or a gene involved in epigenetic modification of DNA; and

wherein the transcription factor is TOX.

2 . The method of claim 1 , wherein the sample comprising T cells from the subject comprises blood, ascites, pleural effusion, lymph, mucus, broncho-alveolar lavage, or tissue.

3 . The method of claim 2 , wherein the sample comprising T cells from the subject comprises CD8+ T cells, tumor-associated lymphocytes, or tumor-infiltrating lymphocytes (TILs).

4 . The method of claim 1 , wherein expression of the one or more genes required for the induction and/or maintenance of T EX in the lymphocytes is reduced.

5 . The method of claim 1 , wherein expression of the one or more genes required for the induction and/or maintenance of T EX in the lymphocytes is eliminated.

6 . The method of claim 4 , wherein expression of the one or more genes required for the induction and/or maintenance of T EX in the lymphocytes is reduced by a method selected from the group consisting of RNA interference, clustered interspersed short palindromic repeat (CRISPR)/CRISPR-associated protein (Cas) system, meganucleases, transcription activator-like effector nucleases (TALENs), Zinc-finger nucleases (ZFNs), antisense, ribozymes and CRISPR inhibition system comprising dead Cas9.

7 . The method of claim 5 , wherein expression of the one or more genes required for the induction and/or maintenance of T EX in the lymphocytes is eliminated by a method selected from the group consisting of RNA interference, clustered interspersed short palindromic repeat (CRISPR)/CRISPR-associated protein (Cas) system, meganucleases, transcription activator-like effector nucleases (TALENs), Zinc-finger nucleases (ZFNs), antisense, ribozymes and CRISPR inhibition system comprising dead Cas9.

8 . The method of claim 1 , wherein the engineering the lymphocytes to target a therapeutically relevant antigen comprises introduction of a recombinant T cell receptor capable of binding a desired antigen/MHC or neo-antigen/MHC combination or introduction of a chimeric antigen receptor capable of binding a desired therapeutically relevant antigen.

9 . A method of reducing or preventing T cell exhaustion in a lymphocyte obtained from a subject, comprising the steps of:

reducing or eliminating expression of one or more genes required for the induction and/or maintenance of exhausted CD8+ T lymphocytes (T EX ) in the lymphocyte;

wherein the gene required for induction and/or maintenance of exhausted CD8+ T lymphocytes is TOX; and

wherein the lymphocyte is a CD8+ T cell.