IP Library Granted Patent US 12708655
Granted Patent B2
US 12708655 · App. 18/260,195 · Granted Aug 18, 2026

Botanicals as WNT/beta-catenin activators, molecular pathway regulators, tissue regenerators and health biomarker regulators

Inventors: Peter R. Feldman (Thornhill, CA); Luciano E. Marra (Toronto, CA); Dennis M. Brown (Menlo Park, CA); Deborah J. Cahan (Thornhill, CA)
Assignee: Arbor Life Holdings, Ltd.
A61K36/28A61K31/10A61K31/355A61K31/4188A61K31/522A61K36/03A61K36/074A61K36/21A61K36/232A61K36/31A61K36/42A61K36/48A61K36/537A61K36/539A61K36/704A61K36/73A61K45/06A61K47/46A61P17/00A61P17/14
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Quick Facts
Patent No.
US 12708655
App. No.
18/260,195
Granted
Aug 18, 2026
Kind
B2
Abstract

The present disclosure provides botanicals and/or biotin or analogs thereof, that proliferate or reduce stem cell populations and activate or attenuate Wat/β-Catenin signaling and thus treat or prevent diseases related to signal transduction. In particular, the disclosure provides Botanicals and Biotin or analogs thereof, that proliferate or reduce stem cell populations and activate or attenuate Wnt/β-Catenin signaling in tissues expressing WntlOB including, adipose, adrenal, artery, blood, bone marrow, brain, breast, cervix, colon, esophagus, heart, intestine, kidney, liver, lung, muscle, ovary, pituitary, prostate, skin, spleen, testis, thyroid, uterus and vagina. The present compositions and methods are particularly suited to growing and melanizing hair.

Claims (125)

1 . A method for maintaining or increasing proliferation of dermal papilla stem cells, follicular unit density, total hairs per follicular unit, terminal hairs per follicular unit, anagen hairs per follicular unit, hair diameter, hair growth rate, follicle productivity, or scalp coverage comprising administering a composition comprising:

biotin

0.005% to 1.00%; 

caffeine

0.0001% to 1.00%;  

Chenopodium quinoa

 0.1% to 2.00%;

Eclipta prostrata

0.01% to 4.00%;

Lupinus

0.01% to 6.00%;

Malus domestica

0.01% to 4.00%;

methylsulfonylmethane

0.005% to 2.00%; 

Momordica charantia

0.01% to 6.00%;

Moringa olifiera

0.01% to 6.00%;

Ocimum basilicum

0.01% to 6.00%;

Pisum sativum

0.01% to 6.00%;

Rosmarinus officinalis

0.01% to 4.00%;

Scutellaria baicalensis

0.01% to 4.00%;

Vitamin E (α tocopherol)

   0.005% to 2.00%; and

proanthocyanidin

0.01% to 4.00%.

2 . The method according to claim 1 , wherein the composition is a topical composition and further comprises a fragrance ingredient comprising one or more of Cedrus deodora, Juniperus virginiana, Matricaria chamomilla, Anthemis nobilis, Helichrysium angustifolia, Jasmine grandiflorum, Lavandula angustifolia, Mentha piperita, Citrus sinensis, Achillea millefolium, Citrus bergamia, Calendula , or Tea Tree.

3 . The method according to claim 1 , wherein the composition is a shampoo and comprises:

biotin

0.025%; 

caffeine

0.0010%;  

Chenopodium quinoa

0.50%;

Eclipta prostrata

0.03%;

Lupinus

1.00%;

Malus domestica

0.06%;

methylsulfonylmethane

0.8%;

Momordica charantia

0.05%;

Moringa olifiera

1.00%;

Rosmarinus officinalis

0.03%;

Scutellaria baicalensis

0.10%;

Vitamin E (α tocopherol)

     0.2%; and

Ocimum basilicum

  0.00%, and

Pisum sativum

0.00%

proanthocyanidin

0.19%.

4 . The method according to claim 1 , wherein the composition is a conditioner and comprises:

biotin

0.025%; 

caffeine

0.0010%;  

Chenopodium quinoa

0.50%;

Eclipta prostrata

0.15%;

Lupinus

2.50%;

Malus domestica

0.19%;

methylsulfonylmethane

0.8%;

Momordica charantia

0.10%;

Moringa olifiera

2.00%;

Rosmarinus officinalis

0.03%;

Scutellaria baicalensis

0.10%;

Vitamin E (α tocopherol)

     0.4%; and

Ocimum basilicum

  0.00%, and

Pisum sativum

0.00%

proanthocyanidin

0.56%.

5 . The method according to claim 1 , wherein the composition is a scalp or a skin cream and comprises:

biotin

0.025%; 

caffeine

0.0010%;  

Chenopodium quinoa

1.50%;

Eclipta prostrata

0.30%;

Lupinus

2.50%;

Malus domestica

0.25%;

methylsulfonylmethane

0.8%;

Momordica charantia

0.20%;

Moringa olifiera

2.00%;

Ocimum basilicum

2.00%;

Pisum sativum

4.00%;

Rosmarinus officinalis

0.30%;

Scutellaria baicalensis

0.17%;

Vitamin E (α tocopherol)

    0.50%; and

proanthocyanidin

0.75%.