Process for preparing aryl-iminomethyl-carbamino acid esters
View Patent ↗The invention relates to a process suitable for large-scale industrial use for preparing compounds of general formula (I) wherein: R 1 denotes a group selected from among methyl, ethyl, propyl, cyclopentyl, cyclohexyl, phenyl, benzyl and —C(Me 2 )phenyl, each of which is optionally mono-, di- or trisubstituted by hydroxy; and, R 2 denotes a group selected from among methyl, ethyl, propyl and benzyl.
1. A compound of the formula (IVA) or the tautomeric form thereof
wherein
R 1 denotes a group selected from among methyl, ethyl, propyl, cyclopentyl, cyclohexyl, phenyl, benzyl and —C(Me 2 )phenyl, each of which may be mono-, di- or trisubstituted by hydroxy; and
R 2 denotes a group selected from among methyl, ethyl, propyl and benzyl.