IP Library Granted Patent US 6,943,171
Granted Patent B2
US 6,943,171 · App. 10/290,011 · Granted Sep 13, 2005

Polycyclic guanine derivative phosphodiesterase V inhibitors

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Quick Facts
Patent No.
US 6,943,171
App. No.
10/290,011
Granted
Sep 13, 2005
Kind
B2
Abstract

A compound having the formula (Ia) or (b), salt or solvate thereof, with the variables as defined herein, which can inhibit selectively phosphodiesterase V and can be useful for treating sexual dysfunction and other physiological disorders, symptoms and diseases:

Claims (17)

1. A compound selected from the group consisting of:

or a pharmaceutically acceptable salt or solvate thereof.

2. The compound according to claim 1 which is:

3. The compound according to claim 1 which is:

4. The compound according to claim 1 which is:

5. The compound according to claim 1 which is:

6. The compound according to claim 1 which is:

7. The compound according to claim 1 which is:

8. A pharmaceutical composition comprising the compound of claim 1 or a salt or solvate thereof and a pharmaceutically acceptable carrier.

9. The composition according to claim 8 , wherein the compound of claim 1 , salt or solvate thereof is administered to a patient in an amount ranging from about 1 to about 1000 milligrams per day.

10. The compound according to claim 1 which is:

11. The compound according to claim 1 which is:

12. The compound according to claim 1 which is:

13. A compound selected from the group consisting of:

or a pharmaceutically acceptable salt or solvate thereof.

14. A compound selected from the group consisting of:

or a pharmaceutically acceptable salt or solvate thereof.

Assignments (3)
CHANGE OF NAME Recorded Aug 30, 2012
From: SCHERING CORPORATION
To: MERCK SHARP & DOHME CORP.
Reel/Frame 028884/0151 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 26, 2003
From: ASBEROM, THEODROS; CLADER, JOHN W.; PISSARNITSKI, DIMITRI A.; STAMFORD, ANDREW W.; XU, RUO
To: SCHERING CORPORATION
Reel/Frame 014208/0213 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 26, 2003
From: HU, YUEQING
To: SCHERING CORPORATION
Reel/Frame 014208/0242 →