IP Library Granted Patent US 7,199,124
Granted Patent B2
US 7,199,124 · App. 10/470,751 · Granted Apr 3, 2007

JNK inhibitor

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Quick Facts
Patent No.
US 7,199,124
App. No.
10/470,751
Granted
Apr 3, 2007
Kind
B2
Abstract

The present invention relates to a c-Jun N-terminal kinase inhibitor containing an azole compound (I) substituted by a nitrogen-containing aromatic group having substituent(s)(except a compound represented by the formula: ) or a salt thereof or a prodrug thereof.

Claims (17)

1. An optionally N-oxidized compound represented by the formula:

wherein

Z n is a bond,

W n is a bond,

R 1n in is a hydrogen atom, a hydrocarbon group optionally having substituent(s), a heterocyclic group optionally having substituent(s), an amino group optionally having substituent(s) or an acyl group,

R 2n is an aromatic group optionally having substituent (s), and

R 3n is a hydrogen atom, a hydrocarbon group optionally having substituent(s) or a heterocyclic group optionally having substituent (s) or a prodrug thereof.

2. An optionally N-oxidized compound represented by the formula:

wherein

R 1g is a hydrogen atom, a hydrocarbon group optionally having substituent(s), a heterocyclic group optionally having substituent(s), an amino group optionally having substituent(s) or an acyl group,

R 2g is an aromatic group optionally having substituent (s),

R 3g is a hydrocarbon group optionally having substituent(s) or a heterocyclic group optionally having substituent(s), and

R 4g is a hydrogen atom or a hydrocarbon group optionally having substituent (s) or a prodrug thereof.

3. A prodrug of the compound of claim 1 .

4. A pharmaceutical agent containing a compound of claim 1 or a prodrug thereof.

5. A prodrug of the compound of claim 2 .

6. A pharmaceutical agent containing a compound of claim 2 or a prodrug thereof.

Assignments (2)
CHANGE OF NAME Recorded Jun 2, 2005
From: TAKEDA CHEMICAL INDUSTRIES, LTD.
To: TAKEDA PHARMACEUTICAL COMPANY LIMITED
Reel/Frame 018917/0406 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 30, 2003
From: OHKAWA, SHIGENORI; NARUO, KENICHI; MIWATASHI, SEIJI; KIMURA, HIROYUKI; KAWAMOTO, TOMOHIRO
To: TAKEDA CHEMICAL INDUSTRIES LTD.
Reel/Frame 014529/0909 →