IP Library Granted Patent US 6,861,390
Granted Patent B2
US 6,861,390 · App. 10/493,456 · Granted Mar 1, 2005

Derivatives of UK-2A

View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 6,861,390
App. No.
10/493,456
Granted
Mar 1, 2005
Kind
B2
Abstract

Derivatives of UK-2A are provided.

Claims (17)

1. A compound according to Formula One:

wherein:

Z is selected from the group consisting of H, R 11 , OR 11 , OC(O)R 11 , OC(O)OR 11 , and OC(O)NR 11 R 12 , OC(O)NR 11-12 R 12-11 ;

R 11 is selected from the group consisting of C 1 -C 8 alkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkynyl, C 3 -C 8 cycloalkyl, aryl, and heteroaryl;

R 12 is selected from the group consisting of H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, C 2 -C 5 alkenyl, and C 2 -C 5 alkynyl;

NR 11-12 R 12-11 is a 5 to 8 membered ring, where the members of the ring are selected from the group consisting of C, O, and S

Q is selected from the group consisting of H, CH 3 , CH 2 CH 3 , CF 3 , Ph, CH═CH 2 , and cyclopropyl;

M is selected from the group consisting of H, CH 3 , CH 2 CH 3 , CF 3 , Ph, CH═CH 2 , or cyclopropyl;

T is selected from the group consisting of O, OC(O), OC(O)O, S, SC(O), SC(O)O,

 G is selected from the group consisting of H, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 2 -C6 alkynyl, C 3 -C 6 cycloalkyl, aryl, and heteroaryl;

optionally, G and M may form a 3-8 membered carbocyclic system;

optionally, M and Q may form a 3-8 membered carbocyclic system;

wherein each of the alkyl, alkoxy, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, benzyl, aryl, and heteroaryl may be substituted with one or more substituents.

2. A compound of claim 1 which is {[2-({[(3S,7R,8R,9S)-7-benzyl-8-(isobutyryloxy)-9-methyl-2,6-dioxo-1,5-dioxonan-3-yl]amino}carbonyl)-4-methoxy-3-pyridinyl]oxy}methyl cyclopentanecarboxylate.

3. A compound of claim 1 which is (3S,6S,7R,8R)-8-benzyl-3-{[(3-{[(ethoxyacetyl)oxy]methoxy}-4-methoxy-2-pyridinyl)carbonyl]amino}-6-methyl-4,9-dioxo-1,5-dioxonan-7-yl 2-methylpropanoate.

4. A composition comprising (1) a compound according to claim 1 , 2 , or 3 , and (2) at least one compound selected from other fungicides, insecticides, nematocides, miticides, arthropodicides, or bactericides.

5. A process comprising using a compound according to claims 1 , 2 , or 3 , or a composition according to claim 4 , in a disease inhibiting and phytologically acceptable amount, to prevent, control, or eradicate, fungal disease.

Assignments (2)
CHANGE OF NAME Recorded Nov 8, 2021
From: DOW AGROSCIENCES LLC
To: CORTEVA AGRISCIENCE LLC
Reel/Frame 058044/0184 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 24, 2005
From: MEYER, KEVIN; ROGERS, RICHARD; NIYAZ, NOORMOHAMED; YAO, CHENGLIN; BUTZ, JENIFER; NADER, BASSAM
To: DOW AGROSCIENCES LLC
Reel/Frame 016179/0869 →