IP Library Granted Patent US 6,987,100
Granted Patent B2
US 6,987,100 · App. 10/652,242 · Granted Jan 17, 2006

Pharmaceutical compositions for treating bone lesions in multiple myeloma

Assignee: Astellas Pharm Inc.
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Quick Facts
Patent No.
US 6,987,100
App. No.
10/652,242
Granted
Jan 17, 2006
Kind
B2
Abstract

Pharmaceutical compositions for treating bone lesions in multiple myeloma or pharmaceutical compositions for treating multiple myeloma which contain as an active ingredient a compound having both of an effect of suppressing bone resorption accompanying multiple myeloma and an effect of inhibiting multiple myeloma, more particularly, 1-hydroxy-2-(imidazo[1,2-a]pyridin-3-yl)ethane-1,1-bisphosphonic acid or its salt.

Claims (4)

1. A method for treating bone lesions in a patient suffering from multiple myeloma and bone lesions by both inhibiting proliferation of myeloma cells and suppressing bone resorption, comprising administering to said patient a pharmaceutically effective amount of 1-hydroxy-2-(imidazo[1,2-a]pyridin-3-yl)ethane-1,1-bisphosphonic acid or a salt thereof, and a pharmaceutically acceptable carrier or diluent.

2. The method of treating bone lesions according to claim 1 , wherein 1-hydroxy-2-(imidazo[1,2-a]pyridin-3-yl)ethane-1,1-bisphosphonic acid or a salt thereof is administered orally in a dose of 1 to 20 mg per day.

3. The method of treating bone lesions according to claim 1 , wherein 1-hydroxy-2-(imidazo[1,2-a]pyridin-3-yl)ethane-1,1-bisphosphonic acid or a salt thereof is administered orally in a dose of 3 to 10 mg per day.

4. A method of both inhibiting myeloma cell proliferation and suppressing bone resorption, comprising administering orally 1-hydroxy-2-(imidazo[1,2-a]pyridin-3-yl)ethane-1,1-bisphosphonic acid or a salt thereof in a dose of 1 to 20 mg per day to a patient suffering from multiple myeloma and bone lesions.

Assignments (1)
MERGER Recorded Sep 22, 2005
From: YAMANOUCHI PHARMACEUTICAL CO., LTD.
To: ASTELLAS PHARMA INC.
Reel/Frame 016570/0324 →
Priority Claims (1)
JP P.10-368399 · Dec 25, 1998 · national
Continuity (2)
Continuation 0986912200
Related Publication 20040043966A1 · Mar 4, 2004