IP Library Granted Patent US 7,812,049
Granted Patent B2
US 7,812,049 · App. 10/763,807 · Granted Oct 12, 2010

Method and therapeutic/cosmetic topical compositions for the treatment of rosacea and skin erythema using α

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Quick Facts
Patent No.
US 7,812,049
App. No.
10/763,807
Granted
Oct 12, 2010
Kind
B2
Abstract

The present invention is directed to the treatment of skin erythema as exhibited in rosacea and other conditions characterized by increased erythema (redness) of the skin. These conditions exhibit dilation of blood vessels due to a cutaneous vascular hyper-reactivity. In particular, the present invention is directed to a novel composition and method for the treatment of skin erythema using α 1 -adrenergic receptor (α 1 -adrenoceptor) agonists incorporated into cosmetic, pharmacological or dermatological compositions for topical application to the skin.

Claims (10)

1. A method of treating erythema resulting from rosacea in a subject comprising administering topically to the skin of said subject a composition comprising about 0.05% to about 30% of oxymetazoline as the sole active agent for treating the erythema resulting from rosacea, wherein said oxymetazoline is effective to decrease the erythema resulting from rosacea.

2. The method of claim 1 , wherein said composition is selected from solutions, gels, lotions, creams, ointments, foams, emulsions, microemulsions, milks, serums, aerosols, sprays, dispersions, microcapsules, vesicles and microparticles thereof.

3. The method of claim 1 , wherein said composition is selected from soaps and cleansing bars.

4. The method of claim 1 , wherein said composition is a cream.

5. The method of claim 1 , wherein said composition is a gel.

6. The method of claim 1 , wherein said composition is a lotion.

7. The method of claim 1 , wherein said erythema resulting from rosacea is elicited by at least one factor selected from the group consisting of intake of food, of hot or alcoholic drinks, temperature variations, heat, exposure to ultraviolet or infrared radiation, exposure to low relative humidity, exposure of the skin to strong winds or currents of air, exposure of the skin to surfactants, irritants, irritant dermatological topical agents, and cosmetics.

8. The method of claim 1 , wherein said composition comprises about 0.1% to about 10% of said oxymetazoline.

9. The method of claim 1 , wherein said composition further comprises about 50% to about 99.999% of a carrier.

10. The method of claim 1 , wherein said composition further comprises about 70% to about 99.99% of a carrier.

Assignments (5)
RELEASE OF SECURITY INTEREST Recorded Jan 11, 2023
From: EVENING POST GROUP, LLC
To: EPI HEALTH, LLC
Reel/Frame 062347/0129 →
SECURITY INTEREST Recorded Mar 14, 2022
From: EPI HEALTH, LLC
To: EVENING POST GROUP, LLC
Reel/Frame 059364/0509 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 30, 2011
From: VICEPT THERAPEUTICS, INC.
To: ALLERGAN, INC.
Reel/Frame 027302/0782 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 22, 2009
From: ASPECT PHARMACEUTICALS, LLC
To: VICEPT THERAPEUTICS, INC.
Reel/Frame 023408/0935 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 17, 2007
From: SHANLER, STUART D.; ONDO, ANDREW
To: ASPECT PHARMACEUTICALS LLC
Reel/Frame 019566/0023 →