IP Library Granted Patent US 7,939,076
Granted Patent B2
US 7,939,076 · App. 10/831,432 · Granted May 10, 2011

Methods for the therapy of Inflammatory Bowel Disease using a type-1 interferon antagonist

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Quick Facts
Patent No.
US 7,939,076
App. No.
10/831,432
Granted
May 10, 2011
Kind
B2
Abstract

Compositions and methods for the therapy of Inflammatory Bowel Disease (IBD), including Celiac Disease, Crohn's Disease, and Ulcerative Colitis, are disclosed. Illustrative compositions comprise one or more anti-type 1 interferon antagonists, such as anti-type 1 interferon receptor antibody antagonists and fragments thereof, as well as polypeptides and small molecules that inhibit the interaction of type 1 interferon with its receptor (IFNAR).

Claims (16)

1. A method for the treatment of a patient afflicted with ulcerative colitis comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω to the type 1 interferon receptor.

2. A method for the treatment of a patient afflicted with ulcerative colitis or Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β and IFN-ω to the type 1 interferon receptor, and is not administered in combination with another antibody, and wherein administration of the anti-type 1 interferon receptor antibody results in decreased neutrophil infiltration as compared to a control, following administration of the anti-type 1 interferon receptor antibody.

3. A method for the treatment of a patient afflicted with ulcerative colitis or Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω to the type 1 interferon receptor, and is not administered in combination with another antibody, and wherein administration of the anti-type 1 interferon receptor antibody results in improved colon morphology as compared to a control, following administration of the anti-type 1 interferon receptor antibody.

4. A method for the treatment of a patient afflicted with ulcerative colitis or Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω to the type 1 interferon receptor, and is not administered in combination with another antibody, and wherein administration of the anti-type 1 interferon receptor antibody results in decreased mucosal tissue thickness as compared to a control, following administration of the anti-type 1 interferon receptor antibody.

5. A method increasing body weight in a patient afflicted with ulcerative colitis or Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω the type 1 interferon receptor, and is not administered in combination with another antibody, and wherein administration of the anti-type 1 interferon receptor antibody results in measurable body weight increase as compared to a control, following administration of the anti-type 1 interferon receptor antibody.

6. A method for the treatment of a patient afflicted with ulcerative colitis or Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω to the type 1 interferon receptor, and is not administered in combination with another antibody.

7. A method for the treatment of a patient afflicted with Crohn's disease comprising the step of administering to said patient a therapeutically effective amount of a humanized or fully human anti-type 1 interferon receptor monoclonal antibody, wherein the antibody inhibits the binding of IFN-α, IFN-β, and IFN-ω to the type 1 receptor, and is not administered in combination with another antibody.

8. The method of any one of claims 1 , 6 , and 7 , wherein said anti-type 1 interferon receptor antibody is administered by a route selected from the group consisting of intravenous bolus, intravenous slow bolus, and infusion.

9. The method of any one of claims 1 , 6 , and 7 , wherein said anti-type 1 interferon receptor antibody is administered by a route selected from the group consisting of subcutaneously, intramuscularly, transdermally, intradermally, and intravenously.

10. The method of any one of claims 1 , 6 , and 7 , wherein said anti-type 1 interferon receptor antibody is administered in a dosage range of between 0.1 mg/kg body weight and 50 mg/kg body weight, inclusive.

11. The method of claim 10 wherein said anti-type 1 interferon receptor antibody is administered in a dosage range of between 0.5 mg/kg body weight and 10 mg/kg body weight, inclusive.

12. The method of claim 11 wherein said anti-type 1 interferon receptor antibody is administered in a dosage range of between 2 mg/kg body weight and 5 mg/kg body weight, inclusive.

13. The method of any one of claims 1 , 6 , and 7 , wherein said anti-type 1 interferon receptor antibody is administered at a frequency between once per day and once per month, inclusive.

14. The method of claim 13 wherein said anti-type 1 interferon receptor antibody is administered at a frequency between twice per week and every two weeks, inclusive.

15. The method of claim 13 wherein said anti-type 1 interferon receptor antibody is administered at a frequency of approximately once per week.

16. The method of any one of claims 1 , 6 , and 7 , further comprising administration of a second therapeutic selected from the group consisting of an immunosuppressive, an anti-inflammatory, a steroid, an immunomodulatory agent, a cytokine, and a TNF antagonist.

Assignments (3)
MERGER Recorded Mar 19, 2015
From: MEDAREX, L.L.C.
To: E. R. SQUIBB & SONS, L.L.C.
Reel/Frame 035226/0690 →
MERGER Recorded Jun 13, 2013
From: MEDAREX, INC.
To: MEDAREX, L.L.C.
Reel/Frame 030603/0924 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 5, 2005
From: PICKFORD, LESLEY B.; BEBBINGTON, CHRISTOPHER R.; YARRANTON, GEOFFREY T.; KING, DAVID
To: MEDAREX, INC.
Reel/Frame 015533/0571 →