IP Library › Granted Patent US 7,632,854

Granted Patent B2

US 7,632,854 · App. 10/990,866 · Granted Dec 15, 2009

Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them

Assignee: Pfizer Italia S.r.l.

View Patent ↗

Loading inventors, assignments & file history…

Monitor This Case

Get email alerts when status or documents change.

Order Certified Copies

Most orders are placed with the USPTO same day — all within 24 business hours.

Order via The Patent Place →

Pre-filled with this patent's details

Quick Facts

Patent No.: US 7,632,854
App. No.: 10/990,866
Granted: Dec 15, 2009
Kind: B2

External Links

USPTO Patent Center↗ Full Patent PDF↗

Abstract

Compounds which are indazole derivatives and pharmaceutically acceptable salts thereof, together with pharmaceutical compositions comprising them, as well as combinatorial libraries of indazole derivatives, as set forth in the specification, are disclosed; these compounds or compositions may be useful in the treatment of diseases caused by and/or associated with an altered protein kinase activity such as cancer, cell proliferative disorders, Alzheimer's disease, viral infections, auto-immune diseases and neurodegenerative disorders.

Claims (1064)

1. A compound of formula (I)

wherein

R is, in position 5 or 6 of the indazole ring, a halogen atom or an optionally substituted group selected from straight or branched C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, or aryl which is selected from phenyl, indanyl, biphenyl, α-or β-naphthyl, fluorenyl, 9,10-dihydroanthracenyl, pyridyl, pyrazinyl, pyrimidinyl, pyridazinyl, indolyl, imidazolyl, imidazopyridyl, 1,2-methylenedioxyphenyl, thiazolyl, isothiazolyl, pyrrolyl, pyrrolyl-phenyl, furyl, phenyl-furyl, benzotetrahydrofuranyl, oxazolyl, isoxazolyl, pyrazolyl, chromenyl, thienyl, benzothienyl, isoindolinyl, benzoimidazolyl, isoindolinyl-phenyl, quinolinyl, isoquinolinyl, 2,6-diphenyl-pyridyl, quinoxalinyl, pyrazinyl, phenyl-quinolinyl, benzofurazanyl, 1,2,3-triazolyl, 1-phenyl-1,2,3-triazolyl, pyran, pyrroline, or pyrazoline;

R 1 is an optionally substituted group selected from —NHCOR′;

R a and R b are, each independently, hydrogen or a straight or branched C 1 -C 6 alkyl group;

R′ and R″ are, each independently, hydrogen or an optionally substituted group selected from straight or branched C 1 -C 6 alkyl, C 2 -C 6 alkenyl or alkynyl, C 3 -C 6 cycloalkyl or cycloalkyl C 1 -C 6 alkyl, aryl or aryl C 1 -C 6 alkyl wherein aryl is as above defined, or a 5or 6 membered heterocyclyl or heterocyclyl C 1 -C 6 alkyl; or, when taken together with the nitrogen atom to which they are attached, R′ and R″ may form an optionally substituted 4 to 7 membered heterocycle, optionally containing an additional heteroatom selected from S, O or N; or isomers, tautomers, and pharmaceutically acceptable salts thereof.

2. A compound of formula (I) according to claim 1 wherein R is an optionally substituted aryl group and R 1 is a group —NHCOR′, wherein R″ is as defined in claim 1 .

3. A library of two or more compounds of formula (I)

wherein

R is, in position 5 or 6 of the indazole ring, a halogen atom or an optionally substituted group selected from straight or branched C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, or aryl which is selected from phenyl, indanyl, biphenyl, α- or β-naphthyl, fluorenyl, 9,10-dihydroanthracenyl, pyridyl, pyrazinyl, pyrimidinyl, pyridazinyl, indolyl, imidazolyl, imidazopyridyl, 1,2-methylenedioxyphenyl, thiazolyl, isothiazolyl, pyrrolyl, pyrrolyl-phenyl, furyl, phenyl-furyl, benzotetrahydrofuranyl, oxazolyl, isoxazolyl, pyrazolyl, chromenyl, thienyl, benzothienyl, isoindolinyl, benzoimidazolyl, isoindolinyl-phenyl, quinolinyl, isoquinolinyl, 2,6-diphenyl-pyridyl, quinoxalinyl, pyrazinyl, phenyl-quinolinyl, benzofurazanyl, 1,2,3-triazolyl, 1-phenyl-1,2,3-triazolyl, pyran, pyrroline, or pyrazoline;

R 1 is an optionally substituted group selected from —NHCOR′;

R a and R b are, each independently, hydrogen or a straight or branched C 1 -C 6 alkyl group;

R′ and R″ are, each independently, hydrogen or an optionally substituted group selected from straight or branched C 1 -C 6 alkyl, C 2 -C 6 alkenyl or alkynyl, C 3 -C 6 cycloalkyl or cycloalkyl C 1 -C 6 alkyl, aryl or aryl C 1 -C 6 alkyl wherein aryl is as above defined, or a 5 or 6 membered heterocyclyl or heterocyclyl C 1 -C 6 alkyl; or, when taken together with the nitrogen atom to which they are attached, R′ and R″ may form an optionally substituted 4 to 7 membered heterocycle, optionally containing an additional heteroatom selected from S, O or N;

or isomers, tautomers, and pharmaceutically acceptable salts thereof.

4. A pharmaceutical composition comprising an effective amount of a compound of formula (I) according to claim 1 and, at least, one pharmaceutically acceptable excipient, carrier or diluent.

5. A pharmaceutical composition according to claim 4 further comprising one or more chemotherapeutic agents.

6. A compound of formula (I) according to claim 1 , optionally in the form of a pharmaceutically acceptable salt, is selected from the group consisting of:

N-[6-(3-methylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

2-methyl-N-[6-(3-methylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]cyclobutanecarboxarnide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-3-cyclopentylpropanarnide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}butanamide;

N-{6-[3-(acetyhtmino)phenyl]-1H-indazol-3-yl}-2-phenoxypropanamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-3-cyclopentylpropanainide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-(4-methoxyphenyl)acetamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxarnide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-chiorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

3-cyclopentyl-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

3-cyclopentyl-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}butanamide;

N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}cyclopropanecarboxamide;

2-methyl-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}propanamide;

2-phenoxy-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

2-(3-methoxyphenyl)-N-[6-(3-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(3-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(3-methylphenyl)-1H-indazol-3-yl]acetamide;

2-methoxy-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

3-fluoro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

3-chloro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

3,4,5-trimethoxy-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

3,5-dichloro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2,4-dimethoxy-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2,3,6-trifluoro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-2-(3-methoxyphenyl)acetamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-2,2-diphenylacetamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-3,4,5-trimethoxybenzamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2,2diphenylacetamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-(benzyloxy)acetamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-3-chlorobenzamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

2-(benzyloxy)-N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]acetamide;

2-(benzyloxy)-N-[6-(3-chlorophenyl)-1H-indazol -3-yl]acetamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(3-chiorophenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(3-chiorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

3,5-dichloro-N-[6-(3-chlorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]acetamide;

2-cyclopentyl-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]acetamide

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

3,5-dichloro-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

2,3,6-trifluoro-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-(benzyloxy)-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

2-methoxy-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

3,4,5-trimethoxy-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2,3,6-trifluoro-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

3cyclopentyl-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]butanamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]butanamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}cyclopentanecarboxamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]cyclopentanecarboxamide

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

3-cyclopentyl-N-[6-(2-methylphenyl)-1-indazol-3-yl]propanamide;

N-[6-(2-methylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

2-methoxy-N-[6-(2-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-methylphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3-cyclopentylpropanamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-3-cyclopentylpropanamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

3-cyclopentyl-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(2,4-dimethoxyphenyl) 1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

3-fluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

3-chloro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

2,3,6-trifluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2-methylphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(2-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-methylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2-methylphenyl)-1H-indazol-3-yl]acetamide;

2-methoxy-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

3-fluoro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

3-chloro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

3,4,5-trimethoxy-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

3,5-dichloro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

2,4-dimethoxy-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

2,3,6-trifluoro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-(benzyloxy)acetamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-cyclopentylacetamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-methoxybenzamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3-chlorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3,5-dichlorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide

2-(benzyloxy)-N-[6-(4-cyanophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]furan-2-carboxamide

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(4-cyanophenyl) 1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

2-(benzyloxy)-N-[6-(2,4-difluorophenyl) 1H-indazol-3-yl]acetamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2-methoxybenzamide

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide

2-(benzyloxy)-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(3-cyanophenyl)-1H-indazol-3-y1]acetamide;

N-[6(3-cyanophenyl)-1H-indazol-3-yl]-2methoxybenzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3,5-dimethylphenyl)-1H -indazol-3-yl]cyclobutanecarboxamide;

3-cyclopentyl-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(2-ethoxyphenyl) 1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6(2-ethoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide ;

3-cyclopentyl-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]propanamide

N-[6-(2,6-dimethylphenyl) 1H-indazol-3-yl]-2-(4-methoxyphenyl)acetamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2-phenylacetamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}cyclopropanecarboxamide;

2-methyl-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}propanamide;

2-phenoxy-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}propanamide;

2-methoxy-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-1-3-yl}acetamide;

N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-phenylacetamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}acetamide;

3-cyclopentyl-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}butanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}cyclopropanecarboxamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-methylpropanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-phenoxypropanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3 -yl}cyclopentanecarboxamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

N-[6-(2,5-(dimethoxyphenyl)-1H-indazol-3-yl]-2-(3-methoxypheny)acetamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2(benzyloxy)-N-[6-(2,5-dimethoxyphenyl)1H-indazol-3-yl]acetamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,5-dimethoxyphenyl) 1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6(2,5-dimethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

2-(benzyloxy)-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3 ,5-dimethylphenyl)-1H-indazol-3-yl]-furan-2-carboxamide;

2-cyclopentyl-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6-(3-ethoxyphenyl-1H-indazol-3-yl]benzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]-2-(3-methoxypheny)acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

3-chloro-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

3,5-dichloro-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

3,5-dichloro-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2,3,6-trifluorobenzamide;

N-{6-[4-(ethylsulfanyl)phenyl]1H-indazol-3-yl}acetamide;

3-cyclopentyl-N-{6-[4-(ethylsulfanyl)phenyl]1H-indazol-3-yl}propanamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}butanamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2-methylpropanamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2-phenoxypropanamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

3-cyclopentyl-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3 -yl}propanamide;

N-{6-[2-methoxy-5-(propan-2-yl) phenyl]-1H-indazol-3-yl}cyclopropanecarboxamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}-2-methylpropanamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}-2-phenoxypropanamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}cyclopentanecarboxamide;

2-methoxy-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

3-cyclopentyl-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}propanamide;

2-(4-methoxyphenyl)-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}butanamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}cyclopropanecarboxamide;

2-methyl-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}-2-phenoxypropanamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}cyclopentanecarboxamide;

2-methoxy-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}cyclobutanecarboxamide;

3-cyclopentyl-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}butanamide;

2-methyl-N-{6-[3(trifluoromethoxy)phenyl]1H-indazol-3-yl}propanamide;

2-phenoxy-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}propanamide;

N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}cyclopentanecarboxamide;

N-[6-(2,5-dimethylphenyl) 1H-indazol-3-yl]-2-phenylacetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]cyclopropanecarboxarnide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-1-yl]cyclobutanecarboxamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2-(4-methoxyphenyl)acetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]butanamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,5-difluorophenyl(-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]2-methoxyacetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(3,4-difluorophenyl)-1-H-indazol-3-yl]propanamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3,4-difluorophenyl)-1H -indazol-3-yl]cyclobutanecarboxamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}furan-2-carboxamide;

2-cyclopentyl-N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-3,4,5-trimethoxybenzamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2,4-dimethoxybenzamide;

2-(3-methoxyphenyl)-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]1H-indazol-3-yl}acetamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}-2,2-diphenylacetamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}furan-2-carboxamide;

2-cyclopentyl-N-{6-[2-methoxy-5(propan-2-yl)phenyl]-1H-indazol-3-yl}acetamide;

2-methoxy-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3-chloro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3,4,5-trimethoxy-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3,5-dichloro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,4-dimethoxy-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,3,6-trifluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-(3-methoxyphenyl)-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}-2,2-diphenylacetamide;

2-(benzyloxy)-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

2-cyclopentyl-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

2-methoxy-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

3-chloro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

3,4,5-trimethoxy-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

3,5-dichloro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,4-dimethoxy-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,3,6-triiluoro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,2-diphenyl-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

2-(benzyloxy)-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

2-(benzyloxy)-N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

3-chloro-N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

3-chloro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

2,3,6-trifluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

2-methoxy-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]-2-phenylacetamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]-2-(4-methoxyphenyl)acetamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]butanamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-fluorophenyl) 1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(4-fluorophenyl) 1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]-2-methoxyacetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2-phenylacetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(3-methoxyphenyl) 1H-indazol-3-yl]propanamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

2-methoxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]propanamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]butanamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]propanamide;

2-methyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]propanamide;

2-phenoxy-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]propanamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-(6-phenyl-1H-indazol-3-yl)acetamide;

3-cyclopentyl-N-(6-phenyl-1H-indazol-3-yl)propanamide;

N-(6-phenyl-1H-indazol-3-yl)butanamide;

N-(6-phenyl-1H-indazol-3-yl)cyclopropanecarboxamide;

N-(6-phenyl-1H-indazol-3-yl)propanamide;

2-methyl-N-(6-phenyl-1H-indazol-3-yl)propanamide;

2-phenoxy-N-(6-phenyl-1H-indazol-3-yl)propanamide;

N-(6-phenyl-1H-indazol-3-yl)cyclopentanecarboxamide;

2-methoxy-N-(6-phenyl-1H-indazol-3-yl)acetamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]-2-phenylacetamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(4-methylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]propanamide;

2-methyl-N-[6-(4-methylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]butanamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

2-methoxy-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(thiophen-2-yl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]propanamide;

N-[6-(thiophen-2-yl)-1H-indazol-3-yl]butanamide;

N-[6-(thiophen-2-yl)-1H-indazol-3-yl]cyclopropanecarboxamide;

2-methyl-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]propanamide;

N-[6-(thiophen-2-yl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2-phenylbutanamide;

2-(benzyloxy)-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2-methylbutanamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]cyclobutanecarboxamide

2-(3-methoxyphenyl)-N-[6-(thiophen-3-y1)-1H-indazol-3-yl]acetamide;

2,2-diphenyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]acetamide;

2-(benzyloxy)-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]acetamide;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]furan-2-carboxamide;

N-(6-phenyl-1H-indazol-3-yl)cyclobutanecarboxamide;

2,2-diphenyl-N-(6-phenyl-1H-indazol-3-yl)acetamide;

2(benzyloxy)-N-(6-phenyl-1H-indazol-3-yl)acetamide;

2-methyl-N-(6-phenyl1H-indazol-3-yl)butanamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(4-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(4-methylphenyl-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(4-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

2-(3-methoxyphenyl)-N-[6-(2-methoxyphenyl) 1H-indazol-3-yl]acetamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(thiophen-2-yl)-1H-indazol-3-yl]cyclobutanecarboxamide;

2-(3-methoxyphenyl)-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]acetamide;

2,2-diphenyl-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]acetamide;

2-(benzyloxy)-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]acetamide;

N-[6-(thiophen-2-yl) 1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(thiophen-3-yl)1H-indazol-3-yl]acetamide;

N-(6-phenyl-1H-indazol-3-yl)furan-2-carboxamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

3-cyclopentyl-N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2-phenoxypropanamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

3-cyclopentyl-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]propanamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]cyclopropanecarboxamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-methylpropanamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide

2-(benzyloxy)-N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-{6[4(propan-2-yl)phenyl]-1H-indazol-3-yl}furan-2carboxamide;

2-methoxy-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3,4,5-trimethoxy-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,3,6-trifluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-(3-methoxypheny)acetamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2,2-diphenylacetamide;

2-(benzyloxy)-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[4(dimethylamino)phenyl]-1H-indazol-3-yl}furan-2-carboxamide;

2-cyclopentyl-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}acetamide;

N-{6[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-methoxybenzamide;

3-chloro-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-3,4,5-trimethoxybenzamide;

N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}furan-2carboxamide;

2-cyclopentyl-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

3,4,5-trimethoxy-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2,4-dimethoxy-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2,3,6-trifluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

3-chloro-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

3,5-dichloro-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2-(3-methoxyphenyl)acetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]furan-2-carboxamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

2-(benzyloxy)-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(4-fluorophenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-cyclopentyl-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]cyclobutanecarboxamide;

2-(3-methoxyphenyl)-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-2,2-diphenylacetamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-cyclopentylacetamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-3-fluorobenzamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2,4-dimethoxybenzamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]2-methoxybenzamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-3,4,5-trimethoxybenzamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2,3,6-trifluorobenzamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]furan-2-carboxamide;

2-(benzyloxy)-N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]acetamide;

N-{6-[4-(trifluorornethoxy)phenyl]-1H-indazol-3-yl}furan-2-carboxamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2-cyclopentylacetamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2-methoxybenzamide;

3,5-dichloro-N-[6-(4-cyanophenyl)-1H-indazol-3-yl]benzamide;

2-cyclopentyl-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,6-dimethylphenyl) 1H-indazol-3-yl]-2,2-diphenylacetamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2-methoxyacetamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2,3,6-trifluorobenzamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]cyclopentanecarboxamide;

2-methoxy-N-[6-(4-methylphenyl)-1H-indazol-3-yl]acetamide;

2-phenoxy-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]propanamide;

2-methoxy-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]acetamide;

2-(3-methoxyphenyl)-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]acetamide;

2-cyclopentyl-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

2,3,4,5-tetrafluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,4-(4-chlorophenoxy)-N-{6-[4(propan-2-yl)phenyl]-1H-indazol-3-yl}acetamide;

2,4-difluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2,3,4,5-tetrafluorobenzamide;

2-(4-chlorophenoxy)-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2,4-difluorobenzamide;

2-{[6-(4-cyanophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(2,4-difluorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,4-difluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

3-cyano-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

2-{[6-(3-cyanophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2,3,4,5-tetrafluoro-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

2,4-difluoro-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]acetamide;

2,4-difluoro-N-[6-(4-fluorophenyl)-1H-indazol-3-yl]benzamide;

2,4-difluoro-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

3,4-difluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

3-cyano-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2-fluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2,6-difluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

2-{[6-(3-cyanophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

2-(4-chlorophenoxy)-N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-Nalpha-[(4-methylphenyl)sulfonyl]-L-phenylalaninamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-Nalpha-[4-methylphenyl)sulfonyl]-L-phenylalaninamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,3,4,5-tetrafluoro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(3-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]-Nalpha-[(4-methylphenyl)sulfonyl]-L-phenylalaninamide;

2,4-difluoro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-2-(4-chlorophenoxy)acetamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-Nalpha-[(4-methylphenyl)sulfonyl]-L-phenylalaninamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2-(4-chlorophenoxy)acetamide;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

2-chloro-N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3-chlorophenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]acetamide;

2,4-difluoro-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3 -yl}benzamide;

2-(4-chlorophenoxy)-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

2,4-difluoro-N-{6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

3-cyano-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2-fluoro-N-[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2,6-difluoro-N[6-(3-methylphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(3-methylphenyl) 1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-methylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(4-acetylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(4-acetylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(4-acetylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]pentanamide;

2-{[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-chloro-4-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

2-{[6-(3-chlorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-chiorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]-4-phenoxybutanamide;

2-{[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3,4-dichlorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(3-fluorophenyl)-1H-indazol-3-yl]pentanamide;

2-fluoro-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]benzamide;

2,6-difluoro-N-[6-(3-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(3-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

2-oxo-2-({6-[4-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}amino)ethyl acetate;

2-oxo-1-phenyl-2-({6-[4-(trifluoromethoxy)pheny]-1H-indazol-3-yl}amino)ethyl acetate;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

2-chloro-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

3-cyano-N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,5-dimethoxyphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

3-cyano-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3,5-dimethylphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

3-cyano-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(3-ethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-ethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

3-cyano-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(2-ethoxyphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(2-ethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2-ethoxyphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

3-cyano-N-[6-(2,6-dimethylphenyl)1H-indazol-3-yl]benzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,6-dimethylphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(3,4-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

4-phenoxy-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}butanamide;

3,4-difluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3-cyano-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-fluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,6-difluoro-N-{6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-oxo-2-({6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}amino)ethyl acetate;

2-oxo-1-phenyl-2-({6-[4-(propan-2-yl)phenyl]-1H-indazol-3-yl}amino)ethyl acetate;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}pentanamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-3,4-difluorobenzamide;

3-cyano-N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}benzamide;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-fluorobenzamide;

2-({6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}amino)-2-oxoethyl acetate;

2-({6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}amino)-2-oxo-1-phenylethyl acetate;

N-{6-[4-(dimethylamino)phenyl]-1H-indazol-3-yl}-2-(thiophen-2-yl)acetamide;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

3,4-difluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

3-cyano-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-fluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

2,4-dichloro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(2-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2-fluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

3,4-difluoro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

3-cyano-N-[6-(2-methylphenyl) 1H-indazol-3-yl]benzamide;

2-fluoro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(2-methylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2-methylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-3-cyanobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]2,4-dichlorobenzamide;

2-{[6-(3-acetylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(3-acetylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-3,4-difluorobenzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(4-cyanophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2,3,4,5-tetrafluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]acetamide;

2,4-difluoro-N-[6-(2-fluorophenyl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-[6-(2-methylphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(2-methylphenyl) 1H-indazol-3-yl]acetamide;

2,4-difluoro-N-[6-(2-methylphenyl)-1H-indazol-3-y1]benzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2-(4-chlorophenoxy)acetamide;

N-[6-(3-acetylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

N-[6-(4-cyanophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

N-[6-(2,4-difluorophenyl)-1H-indazol-3-yl]-Nalpha-[(4-methylphenyl))sulfonyl]-L-phenylalaninamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-ylZ]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

N-[6-(2,4-dimethoxyphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

N-[6-(3-cyanophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2,3,4,5-tetrafluorobenzamide;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2,4-difluorobenzamide;

2,3,4,5-tetrafluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-(4-chlorophenoxy)-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-H-indazol-3-yl}cyclohexanecarboxamide;

2,4-difluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,3,4,5-tetrafluoro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2-(4-chlorophenoxy)-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}acetamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}cyclohexanecarboxamide;

2,4-difluoro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,3,4,5-tetrafluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2-(4-chlorophenoxy)-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}acetamide;

2,4-difluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(2,5-dimethylphenyl)-1I-1-indazol-3-yl]acetamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-chloro-N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-6-fluorobenzamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2,3,4,5-tetrafluorobenzamide;

2-(4-chlorophenoxy)-N-[6-(3,4-difluorophenyl)-1H-indazol-3-yl]acetamide;

N[6-(3,4-difluorophenyl)-1H-indazol-3-yl]-2,4-difluorobenzamide;

2,3,4,5-tetrafluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

2,4-difluoro-N-[6-(5-fluoro-2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-[6-(thiophen-2-yl-1H-indazol-3-yl]benzamide;

2,4-difluoro-N-[6-(thiophen-2-yl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

2,4-difluoro-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-[6-(4-methylphenyl)-1H-indazol-3-yl]benzamide;

2-(4-chlorophenoxy)-N-[6-(4-methylphenyl)-1H-indazol-3-yl]acetamide;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]cyclohexanecarboxamide;

2,4-difluoro-N-[6-(4-methylphenyl-1H-indazol-3-yl]benzamide;

2,3,4,5-tetrafluoro-N-(6-phenyl-1H-indazol-3-yl)benzamide;

2-(4-chlorophenoxy)-N-(6-phenyl-1H-indazol-3-yl)acetamide;

N-(6-phenyl-1H-indazol-3-yl)cyclohexanecarboxamide;

2,4-difluoro-N-(6-phenyl-1H-indazol-3-yl)benzamide;

2,4-difluoro-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]benzamide;

2-{[6-(3,4-difluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-{6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}-2,6-difluorobenzamide;

2-({6-[4-ethylsulfanyl)phenyl]-1H-indazol-3-yl}amino)-2-oxoethyl acetate;

2-({6-[4-(ethylsulfanyl)phenyl]-1H-indazol-3-yl}amino)-2-oxo-1-phenylethyl acetate;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}-3-phenylpropanamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}pentanamide;

b 3 , 4 -difluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

3-cyano-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl }benzamide;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-fluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,6-difluoro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2,4-dichloro-N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}benzamide;

2-({6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}amino) -2-oxoethyl acetate;

2-({6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}amino)-2-oxo-1-phenylethyl acetate;

N-{6-[2-methoxy-5-(propan-2-yl)phenyl]-1H-indazol-3-yl}-2-(thiophen-2-yl)acetamide;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}-3-phenylpropanamide;

3,4-difluoro-N-{6-[2-(methylsulfanyl)phenyl]1H-indazol-3-yl}benzamide;

3-cyano-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2-fluoro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,6-difluoro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2,4-dichloro-N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}benzamide;

2-({6-[2-(methylsulfanyl)phenyl]1H-indazol-3yl}amino)-2-oxoethyl acetate;

2-({6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}amino)-2-oxo-1-phenylethyl acetate;

N-{6-[2-(methylsulfanyl)phenyl]-1H-indazol-3-yl}-2-(thiophen-2-yl)acetamide;

3,4-difluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

3-cyano-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2-fluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2,6-difluoro-N-{6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}benzamide;

2-oxo-2-({6-[3-(trifluoromethoxy)phenyl]-1H-indazol-3-yl}amino)ethyl acetate;

2-oxo-1-phenyl-2-({6-[3(trifluoromethoxy)phenyl]-1H-indazol-3-yl}amino)ethyl acetate;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-3 ,4-difluorobenzamide;

3-cyano-N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2-{[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(2,5-dimethylphenyl)-1H-indazol-3-yl]-2-(thiophen-2-yl)acetamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-3-phenylpropanamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]pentanamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]benzamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2-fluorobenzamide;

N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]-2,6-difluorobenzamide;

2,4-dichloro-N-[6-(2,5-difluorophenyl)-1H-indazol-3-yl]benzamide;

2-{[6-(2,5-difluorophenyl)-1H-indazol-3-yl]amino}-2-oxoethyl acetate;

2-{[6-(2,5-difluorophenyl)-1H-indazol-3-yl]amino}-2-oxo-1-phenylethyl acetate;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

N-butyl-N′-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-butyl-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(morpholin-4-yl)ethyl]urea;

1-[3-(1H-imidazol-1-yl)propyl]-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-(tetrahydrofuran-2-ylmethyl)urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-(2-phenylethyl)urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-(3-phenylpropyl)urea;

1-[6-(4-methoxyphenyl)-1H-indazoi-3-yl]-3-propylurea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-(2-methylpropyl)urea;

1-(cyclopropylmethyl)-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(1-methylpyrrolidin-2- yl)ethyl]urea;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(morpholin-4-yl)ethyl]urea;

1-[3-(1H-imidazol-1-yl)propyl]-3-[6-(3-methoxyphenyl)-1H-indazol-3-yl]urea;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(tetrahydrofuran-2-ylmethyl)urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(2-phenylethyl)urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(3-phenylpropyl)urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(2-methylpropyl)urea;

1-(cyclopropylmethyl)-3-[6-(3-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-[2-(morpholin-4-yl)ethyl]-3[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-[3-(1H-imidazol-1-yl)propyl]-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-(tetrahydrofuran-2-ylmethyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-(2-phenylethyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-(3-phenylpropyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-propyl-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-(2-methylpropyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-(cyclopropylmethyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-[2-(methylpyrrolidin-2-yl)ethyl ]-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-butyl-3-[6-(4-methylphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-[2-(morpholin-4-yl)ethyl]urea;

1-[3-(1H-imidazol-1-yl)propyl]-3-[6-(4methylphenyl)-1H-indazol-3-yl]urea;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-(3-phenylpropyl)urea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-propylurea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-(2-methylpropyl)urea;

1-(cyclopropylmethyl)-3-[6-(4-methylphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea;

1-butyl-3-[6-(2-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(morpholin-4-yl)ethyl]urea;

1-[3-(1H-imidazol-1-yl)propyl]-3-[6-(2-methoxyphenyl)-1H-indazol-3 -yl]urea;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(2-rnethoxyphenyl)-1H-indazol-3-yl]-3-(tetrahydroftiran-2-ylmethyl)urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-(2-phenylethyl)urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-(3-phenylpropyl)urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-propylurea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-(2-methylpropyl)urea;

1-(cyclopropylmethyl)-3-[6-(2-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-butyl-3-[6-(3-methylphenyl)-1H-indazol-3-yl]urea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-[2-(morpholin-4-yl)ethyl]urea;

1-[3(1H-imidazol-1-yl)propyl]-3-[6-(3-methylphenyl)-1H-indazol-3-yl]urea;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-(2-phenylethyl)urea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-propylurea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-(2-methylpropyl)urea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}piperidine-1-carboxamide;

N-[3-(3-{[(butylamino)carbonyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-(3-{3-[(butylcarbamoyl)amino]-1H-indazol-6-yl}phenyl)acetamide;

N-{3-[3-({[2-(morpholin-4-yl)ethyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide;

N-{3-[3-({[3-(1H-imidazol-1-yl)propyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide; N-[3-(3-{[(tetrahydrofuran-2-ylmethyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-[3(3-{[(2-phenylethyl)carbamoyl]amino }-1H-indazol-6-yl)phenyl]acetamide;

N-[3-(3-{[(3-phenylpropyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-(3-{3-[(propylcarbamoyl)amino]-1H-indazol-6-yl}phenyl)acetamide;

N-[3-(3-{[(cyclopropylmethyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]aeetamide;

N-{3-[3-({[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperidine-1-carboxamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperazine-1-carboxamide;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea;

1-(3-aminopropyl)-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-(2-aminoethyl)-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

4-hydroxy-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-(3-hydroxypropyl)-3-[6-(4-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(pyridin-2-yl)ethyl]urea;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(piperidin-1-yl)ethyl]urea;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({[6-(4-methoxyphenyl)-1H-indazol-3-yl]carbamoyl}amino)ethyl]acetamide;

4-acetyl-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperidine-1-carboxamide;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperazine-1-carboxamide;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea;

4-hydroxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-(3-hydroxypropyl)-3-[6-(3-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(pyridin-2-yl)ethyl]urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(piperidin-1-yl)ethyl]urea;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({[6-(3-methoxyphenyl)-1H-indazol-3-yl]carbamoyl}amino)ethyl]acetamide; 4-acetyl-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

4-methyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperidine-1-carboxamide;

4-methyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[3-(2-oxopyrrolidin-1-yl)propyl]-3-[6-(thiophen-3-yl)1H-indazol-3-yl]urea;

1-(3-aminopropyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-(2-aminoethyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

4-hydroxy-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-(3-hydroxypropyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1[2-(pyridin-2-yl)ethyl]-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

1-[2-(piperidin-1-yl)ethyl]-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

N-[6-(thiophen-3-yl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({([6-(thiophen-3-yl)-1H-indazol-3-yl]carbamoyl}amino)ethyl]acetamide;

4-acetyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperazine-1-carboxamide;

4-methyl-N-[6(4-methylphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

4-methyl-N-[6-(4-methylphenyl)1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea;

1-(3-aminopropyl)-3-[6-(4-methylphenyl)-1H-indazol-3-yl]urea;

1-(2-aminoethyl)-3-[6-(4-methylphenyl)-1H-indazol-3-yl]urea;

4-hydroxy-N-[6-(4-methylphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-(3-hydroxypropyl)-3-[6-(4-methylphenyl)-1H-indazol-3-yl]urea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-[2-(pyridin-2-yl)ethyl]urea;

1-[6-(4-methylphenyl)-1H-indazol-3-yl]-3-[2-(piperidin-1-yl)ethyl]urea;

N-[6-(4-methylphenyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({[6-(4methylphenyl)-1H-indazol-3-yl]carhamoyl}amino)ethyl]acetamide;

4-acetyl-N-[6-(4-methylphenyl)-1H-indarzol-3-yl]piperazine-1-carboxamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperidine-1-carboxamide;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-4-methylpiperazine-1-carboxarnide;

1-[6-(2-methoxyphenyl) 1H-indazol-3-yl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea;

1-(3-aminopropyl)-3-[6-(2-methoxyphenyl)-1H-indazol-3-yl]urea;

1-(2-aminoethyl)-3-[6-(2-methoxyphenyl)-1H-indazol-3-yl]urea;

4-hydroxy-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

1-(3-hydroxypropyl)-3-[6-(2-methoxyphenyl)-1H-indazol-3-yl]urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(pyridin-2-yl)ethyl]urea;

1-[6-(2-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(piperidin-1-yl)ethyl]urea;

N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({[6-(2-methoxyphenyl)1H-indazol-3-yl]carbamoyl}amino)ethyl]acetamide;

4-acetyl-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-(2-aminoethyl)-3-[6-(thiophen-2-yl)-1H-indazol-3-yl]urea;

4-methyl-N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

4-methyl-N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea;

1-(3-aminopropyl)-3-[6-(3-methylphenyl)-1H-indazol-3-yl]urea;

1-(2-aminoethyl)-3-[6-(3-methylphenyl)-1H-indazol-3-yl]urea;

4-hydroxy-N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperidine-1 -carboxamide;

1-(3-hydroxypropyl)-3-[6-(3-methylphenyl)-1H-indazol-3-yl]urea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-[2-(pyridin-2-yl)ethyl]urea;

1-[6-(3-methylphenyl)-1H-indazol-3-yl]-3-[2-(piperidin-1-yl)ethyl]urea;

N-[6-(3-methylphenyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide;

N-[2-({[6-(3-methylphenyl)-1H-indazol-3-yl]carbamoyl}amino)ethyl]acetamide;

4-acetyl-N-[6-(3-methylphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-4-methylpiperidine-1-carboxamide;

N-{3-[3-({[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}(amino)-1H-indazol-6-yl]phenyl}acetamide;

N-[3-(3-{[(3-aminopropyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-[3-(3-{[(2-aminoethyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-{6-[3-(acetylamino)phenyl]-1H-indazol-3-yl}-4-hydroxypiperidine-1-carboxamide;

N-[3-(3-{[(3-hydroxypropyl)carbamoyl]amino}-1H-indazol-6-yl)phenyl]acetamide;

N-{3-[3-({[2-(pyridin-2-yl)ethyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide;

N-{3-[3-({[2-(piperidin-1-yl)ethyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide;

N-{3-[3-({[2-(acetylamino)ethyl]carbamoyl}amino)-1H-indazol-6-yl]phenyl}acetamide;

1-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-(3-methoxypropyl)urea;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-methylpiperidine-1-carboxamide;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]-4-(pyridin-2-yl)piperazine-1-carboxamide;

4-benzyl-N-[6-(4-methoxyphenyl)1H-indazol-3-yl]piperidine-1-carboxamide;

1-[(1-ethylpyrrolidin-2-yl)methyl]-3-[6-(4-methoxyphenyl )-1H-indazol-3-yl]urea;

4-(furan-2-ylcarbonyl)-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(thiophen-2-yl)ethyl]urea;

1[6-(4-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea;

N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]thiomorpholine-4-carboxamide;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(3-methoxypropyl)urea;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-methylpiperidine-1-carboxamide;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-(2-methylbutyl)urea;

N[6-(3-methoxyphenyl)-1H-indazol-3-yl]-4-(pyridin-2-yl)piperazine-1-carboxamide;

4-benzyl-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperidine-1-carboxamide;

N˜3˜,N˜3˜-diethyl-N˜1˜-[6-(3methoxyphenyl)-1H-indazol-3-yl]piperidine-1,3-dicarboxamide;

N-[6-(3-methoxyphenyl)1H-indazol-3-yl]-3 ,5-dimcthylpiperidine-1-carboxamide;

1[(1-ethylpyrrolidin-2-yl)methyl]-3-[6-(3-methoxyphenyl)-1H-indazol-3-yl]urea;

4-(furan-2-ylcarbonyl)-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]piperazine-1-carboxamide;

1-[6-(3-melhoxyphenyl)-1H-indazol-3-yl]-3-[2-(thiophen-2-yl)ethyl]urea;

1-[6-(3-methoxyphenyl)-1H-indazol-3-yl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea;

N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]thiomorpholine-4-carboxamide;

1-(3-methoxypropyl)-3-[6-(thiophen-3-yl)-1H-indazol-3-yl]urea;

3-methyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperidine-1-carboxamide;

4-benzyl-N-[6-(thiophen-3-yl)-1H-indazol-3-yl]piperidine-1-carboxamide; and

1-butyl-3-[6-(3-methoxyphenyl)-1H-indazol-3-yl]urea.

Assignments (3)

ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 2, 2017

From: PFIZER ITALIA S.R.L.

To: NERVIANO MEDICAL SCIENCES S.R.L

Reel/Frame 041154/0945 →

MERGER Recorded Sep 12, 2006

From: PHARMACIA ITALIA S.P.A.

To: PFIZER ITALIA S.R.L.

Reel/Frame 018248/0222 →

ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 25, 2005

From: MARTINA, KATIA; BRILL, WOLFGANG

To: PHARMACIA ITALIA S.P.A.

Reel/Frame 016304/0560 →

Continuity (1)

Related Publication 20060106083A1 · May 18, 2006