IP Library Granted Patent US 7,745,436
Granted Patent B2
US 7,745,436 · App. 11/105,818 · Granted Jun 29, 2010

Disalt inhibitors of IL-12 production

View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 7,745,436
App. No.
11/105,818
Granted
Jun 29, 2010
Kind
B2
Abstract

This invention relates to disalt nitrogen-heteroaryl inhibitors of IL-12 production, and related methods and pharmaceutical compositions.

Claims (7)

1. A disalt represented by the formula:

wherein each M − is a conjugate base of a Bronsted acid.

2. The disalt of claim 1 , wherein M − is the conjugate base of a Bronsted acid selected from the group consisting of hydrochloric acid, nitric acid, sulfuric acid, hydrobromic acid, hydroiodic acid, perchloric acid, phosphoric acid, alkylsulfonic acids, arylsulfonic acids, halogenated alkylsulfonic acids, halogenated acetic acids, picric acid, oxalic acid, citric acid, formic acid, ascorbic acid and benzoic acid.

3. The disalt of claim 2 , wherein M − is methanesulfonate.

4. The disalt of claim 2 , wherein M − is bromide.

5. The disalt of claim 2 , wherein M − is chloride.

6. A pharmaceutical composition comprising a pharmaceutically acceptable carrier and a disalt according to claim 1 .

Assignments (5)
SECURITY INTEREST Recorded Feb 18, 2026
From: ORPHAI THERAPEUTICS INC.
To: ACADIA WOODS PARTNERS, LLC, AS AGENT
Reel/Frame 074910/0274 →
SECURITY INTEREST Recorded Jul 17, 2025
From: MADRIGAL PHARMACEUTICALS, INC.
To: LSI FINANCING LLC, AS ADMINISTRATIVE AGENT
Reel/Frame 072038/0693 →
SECURITY INTEREST Recorded Jun 23, 2025
From: ORPHAI THERAPEUTICS INC.
To: ACADIA WOODS PARTNERS, LLC
Reel/Frame 071697/0788 →
CHANGE OF NAME Recorded May 3, 2021
From: SYNTA PHARMACEUTICALS CORP.
To: MADRIGAL PHARMACEUTICALS, INC.
Reel/Frame 056121/0785 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 21, 2005
From: KOSTIK, ELENA; SUN, LIJUN
To: SYNTA PHARMACEUTICALS CORP.
Reel/Frame 016923/0719 →