IP Library Granted Patent US 7,977,345
Granted Patent B2
US 7,977,345 · App. 11/571,140 · Granted Jul 12, 2011

c-MET modulators and method of use

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Quick Facts
Patent No.
US 7,977,345
App. No.
11/571,140
Granted
Jul 12, 2011
Kind
B2
Abstract

A compound for modulating kinase activity according to Formula I, or a pharmaceutically acceptable salt thereof, Wherein J 1 , J 2 , J 3 , R 2 , J 4 , Z, Ar and R 3 are as defined in the specification, compositions thereof, and methods of use thereof.

Claims (22)

1. A compound of formula IVc:

wherein:

J 1 is ═CH—;

J 2 is ═C(R 1 )—;

J 3 is ═N—;

J 4 is ═N—;

J 5 is C—H or C—F;

Z is O;

R 1 is independently selected from halogen, trihalomethyl, —CN, —NO 2 , —OR 20 , —N(R 20 )R 20 , —S(O) 0-2 R 20 , —SO 2 N(R 20 )R 20 , —CO 2 R 20 , —C(O)N(R 20 )R 20 , —N(R 20 )SO 2 R 20 , —N(R 20 )C(O)R 20 , —NHCO 2 R 20 , —C(O)R 20 , optionally substituted C 1-6 alkyl, optionally substituted aryl, optionally substituted aryl C 1-6 alkyl optionally substituted heterocyclyl, and optionally substituted heterocyclyl C 1-6 alkyl;

R 2 is H;

each R 3a is independently selected from —H, halogen, trihalomethyl, —CN, —NO 2 , —OR 20 , —N(R 20 )R 20 , —S(O) 0-2 R 20 , —SO 2 N(R 20 )R 20 , —CO 2 R 20 , —C(O)N(R 20 )R 20 , —N(R 20 )SO 2 R 20 , —N(R 20 )C(O)R 20 , —NHCO 2 R 20 , —C(O)R 20 , optionally substituted C 1-6 alkyl, and optionally substituted heterocyclyl;

each R 20 is independently —H, optionally substituted C 1-6 alkyl, optionally substituted aryl, optionally substituted aryl C 1-6 alkyl, optionally substituted heterocyclyl, and optionally substituted heterocyclyl C 1-6 alkyl; or two of R 20 , when taken together with a common nitrogen to which they are attached, can form an optionally substituted five- to seven-membered heterocyclyl, said optionally substituted five- to seven-membered heterocyclyl optionally containing at least one additional annular heteroatom selected from N, O, S, and P; and

each R 70 is independently selected from —H, halogen, trihalomethyl, —CN, —NO 2 , —OR 20 , —N(R 20 )R 20 , —S(O) 0-2 R 20 , —SO 2 N(R 20 )R 20 , —CO 2 R 20 , —C(O)N(R 20 )R 20 , —N(R 20 )SO 2 R 20 , —N(R 20 )C(O)R 20 , —NHCO 2 R 20 , —C(O)R 20 , optionally substituted C 1-6 alkyl, optionally substituted aryl, optionally substituted aryl C 1-6 alkyl, optionally substituted heterocyclyl, and optionally substituted heterocyclyl C 1-6 alkyl.

2. A compound selected from:

Entry

Name

Structure

2

N-(4-fluorophenyl)-N′-[3-fluoro-4-(7H- pyrrolo[2,3-d]pyrimidin-4- yloxy)phenyl]cyclopropane-1,1- dicarboxamide

12

N-{3-fluoro-4-[(6-{[(2-morpholin-4- ylethyl)amino]carbonyl}-7H-pyrrolo[2,3- d]pyrimidin-4-yl)oxy]phenyl}-N′-(4- fluorophenyl)cyclopropane-1,1- dicarboxamide

3. A pharmaceutical composition comprising a compound according to claim 1 or 2 and a pharmaceutically acceptable carrier.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 16, 2007
From: BANNEN, LYNNE CANNE; CHAN, DIVA SZE-MING; DALRYMPLE, LISA ESTHER; JAMMALAMADAKA, VASU; KHOURY, RICHARD GEORGE; LEAHY, JAMES WILLIAM; MAC, MORRISON B; MANN, GRACE; MANN, LARRY W; NUSS, JOHN M; PARKS, JASON JEVIOUS; WANG, YONG; XU, WEI
To: EXELIXIS, INC.
Reel/Frame 018759/0933 →