IP Library Granted Patent US 7,943,651
Granted Patent B2
US 7,943,651 · App. 11/736,606 · Granted May 17, 2011

Compounds

Assignee: Glaxo Group Limited
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 7,943,651
App. No.
11/736,606
Granted
May 17, 2011
Kind
B2
Abstract

The present invention provides compounds of formula (I): pharmaceutical compositions comprising the compounds and the use of the compounds for the manufacture of a medicament, particularly for the treatment of inflammation and/or allergic conditions.

Claims (8)

1. 1-{[3-(4-{[(2R)-4-[5-Fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)phenyl]carbonyl}-D-prolinamide:

2. A pharmaceutical composition comprising a compound as claimed in claim 1 , optionally in admixture with one or more physiologically acceptable diluents or carriers.

3. A pharmaceutical composition according to claim 2 , wherein said composition is adapted for intranasal delivery.

4. A pharmaceutical composition comprising the compound of claim 1 , in combination with one or more therapeutically active agents.

5. 1-{[3-(4-{[(2R)-4-[5-Fluoro-2-(methyloxy) phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl) phenyl]carbonyl}-D-prolinamide:

or a salt thereof.

6. A pharmaceutical composition comprising 1-{[3-(4-{[(2R)-4-[5-Fluoro-2-(methyloxy) phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)phenyl]carbonyl}-D-prolinamide:

and one or more suspending agents.

Assignments (2)
CHANGE OF ADDRESS Recorded Apr 16, 2025
From: GLAXO GROUP LIMITED
To: GLAXO GROUP LIMITED
Reel/Frame 071044/0904 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 24, 2007
From: BIGGADIKE, KEITH; COOPER, ANTHONY WILLIAM JAMES; HOUSE, DAVID; MCLAY, IAIN MCFARLANE; WOOLLAM, GRAHAME ROBERT
To: GLAXO GROUP LIMITED
Reel/Frame 019742/0318 →
Priority Claims (4)
GB 0607840.6 · Apr 20, 2006 · national
GB 0620382.2 · Oct 13, 2006 · national
GB 0706515.4 · Apr 3, 2007 · national
GB 0706516.2 · Apr 3, 2007 · national
Continuity (1)
Related Publication 20070265326A1 · Nov 15, 2007