IP Library Granted Patent US 7,632,862
Granted Patent B2
US 7,632,862 · App. 11/787,535 · Granted Dec 15, 2009

Pharmaceutical compositions that modulate HPTPbeta activity

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Quick Facts
Patent No.
US 7,632,862
App. No.
11/787,535
Granted
Dec 15, 2009
Kind
B2
Abstract

HPTPbeta is useful as a target in screening agents effective for the treatment of angiogenesis mediated disorders.

Claims (8)

1. A pharmaceutical composition, comprising:

a) an effective amount of (R)-[1-methylcarbamoyl-2-(4-sulfoaminophenyl)ethyl]-carbamic acid tert-butyl ester; and

b) a pharmaceutically-acceptable carrier.

2. A pharmaceutical composition for modulating an angiogenesis mediated disorder, comprising:

a) about 500 μM of (R)-[1-methylcarbamoyl-2-(4-sulfoaminophenyl)ethyl]-carbamic acid tert-butyl ester; and

b) a pharmaceutically-acceptable liquid carrier.

3. The composition according to claim 2 , wherein the angiogenesis mediated disorder is selected from disorders, diseases, and/or unwanted conditions characterized by a wanted increase in angiogenesis or characterized by reduced angiogenesis selected from the group consisting of skeletal muscle ischemia, myocardial ischemia, stroke, coronary artery disease, peripheral vascular disease, and tissue repair where tissue has been damaged by trauma, surgical procedures, irradiation, laceration, toxic chemicals, viral infection, bacterial infection, non-healing wounds, or burns, or where tissue has been damaged by arthritis or osteoporosis.

4. The composition according to claim 2 , wherein the angiogenesis mediated disorder is tissue ischemia.

Assignments (11)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 17, 2020
From: AERPIO THERAPEUTICS LLC
To: AERPIO PHARMACEUTICALS, INC.
Reel/Frame 052432/0789 →
CHANGE OF NAME Recorded Jul 31, 2019
From: AERPIO THERAPEUTICS, INC.
To: AERPIO THERAPEUTICS LLC
Reel/Frame 049920/0084 →
RELEASE OF SECURITY INTEREST Recorded Oct 31, 2013
From: BANK OF AMERICA, N.A., AS COLLATERAL AGENT
To: WARNER CHILCOTT COMPANY, LLC
Reel/Frame 031531/0538 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 2, 2012
From: AKEBIA THERAPEUTICS, INC.
To: AERPIO THERAPEUTICS, INC.
Reel/Frame 027801/0358 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 27, 2011
From: WARNER CHILCOTT COMPANY, LLC
To: AKEBIA THERAPEUTICS INC.
Reel/Frame 027445/0100 →
PATENT RELEASE Recorded Dec 23, 2011
From: BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT
To: WARNER CHILCOTT COMPANY, LLC
Reel/Frame 027443/0164 →
SECURITY AGREEMENT Recorded Mar 30, 2011
From: WARNER CHILCOTT COMPANY LLC
To: BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 026064/0607 →
RELEASE - REEL 023456, FRAME 0052 Recorded Mar 29, 2011
From: CREDIT SUISSSE AG, CAYMAN ISLANDS BRANCH, AS ADMINISTRATIVE AGENT
To: WARNER CHILCOTT COMPANY LLC
Reel/Frame 026042/0046 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 8, 2010
From: PROCTER & GAMBLE COMPANY, THE
To: WARNER CHILCOTT COMPANY, LLC
Reel/Frame 023796/0417 →
SECURITY AGREEMENT Recorded Nov 2, 2009
From: WARNER CHILCOTT COMPANY, LLC
To: CREDIT SUISSE, CAYMAN ISLANDS BRANCH, AS ADMINISTRATIVE AGENT
Reel/Frame 023456/0052 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 11, 2008
From: PETERS, KEVIN GENE; DAVIS, MICHAEL GLENN
To: PROCTER & GAMBLE COMPANY, THE
Reel/Frame 020357/0522 →