HIV inhibiting 2-(4-cyanophenylamino) pyrimidine oxide derivatives
View Patent ↗HIV replication inhibitors of formula (I) a pharmaceutically acceptable addition salt; or a stereochemically isomeric form thereof, wherein R 1 is halo; R 2 and R 3 each independently are C 1-6 alkyl. Pharmaceutical compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
1. A compound of formula
or a pharmaceutically acceptable addition salt thereof, wherein
R 1 is bromo;
R 2 and R 3 are methyl.
2. A pharmaceutical composition comprising a pharmaceutically acceptable carrier and as active ingredient a therapeutically effective amount of a compound as claimed in claim 1 .
3. A process for preparing a composition according to claim 2 , the process comprising intimately mixing the active ingredient and the carrier.