IP Library Granted Patent US 8,138,347
Granted Patent B2
US 8,138,347 · App. 12/121,891 · Granted Mar 20, 2012

Quinoline derivatives as PI3 kinase inhibitors

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Quick Facts
Patent No.
US 8,138,347
App. No.
12/121,891
Granted
Mar 20, 2012
Kind
B2
Abstract

Invented is a method of inhibiting the activity/function of PI3 kinases using quinoline derivatives. Also invented is a method of treating one or more disease states selected from: autoimmune disorders, inflammatory diseases, cardiovascular diseases, neurodegenerative diseases, allergy, asthma, pancreatitis, multiorgan failure, kidney diseases, platelet aggregation, cancer, sperm motility, transplantation rejection, graft rejection and lung injuries by the administration of quinoline derivatives.

Claims (4)

1. A compound, which is 2,4-difluoro-N-{2-(methyloxy)-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl}benzenesulfonamide, or a pharmaceutically acceptable salt thereof.

2. A compound, which is represented by the following structure

3. A pharmaceutically acceptable salt of a compound of claim 1 .

4. A pharmaceutical composition comprising a compound or a pharmaceutically acceptable salt of claim 1 and a pharmaceutically acceptable carrier.

Assignments (3)
CHANGE OF NAME Recorded Sep 15, 2013
From: SMITHKLINE BEECHAM CORPORATION
To: GLAXOSMITHKLINE LLC
Reel/Frame 031217/0381 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 28, 2008
From: ADAMS, NICHOLAS D.; BURGESS, JOELLE LORRAINE; DARCY, MICHAEL GERARD; DONATELLI, CARLA A.; KNIGHT, STEVEN DAVID; NEWLANDER, KENNETH ALLEN; RIDGERS, LANCE; SARPONG, MARTHA A.; SCHMIDT, STANLEY J.
To: SMITHKLINE BEECHAM CORPORATION
Reel/Frame 021454/0110 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 4, 2008
From: ADAMS, NICHOLAS D.; BURGESS, JOELLE LORRAINE; DARCY, MICHAEL GERARD; DONATELLI, CARLA A.; KNIGHT, STEVEN DAVID; NEWLANDER, KENNETH ALLEN; RIDGERS, LANCE; SARPONG, MARTHA A.; SCHMIDT, STANLEY J.
To: SMITHKLINE BEECHAM CORPORATION
Reel/Frame 021333/0246 →