IP Library Granted Patent US 8,377,939
Granted Patent B2
US 8,377,939 · App. 12/134,553 · Granted Feb 19, 2013

Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators 842

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Quick Facts
Patent No.
US 8,377,939
App. No.
12/134,553
Granted
Feb 19, 2013
Kind
B2
Abstract

Compounds of Formula I: wherein R 1 and Q are as described in the specification, pharmaceutically-acceptable salts, methods of making, pharmaceutical compositions containing and methods for using the same.

Claims (5)

1. A compound that is: 7-methyl-5-(3-piperazin-1-ylmethyl-[1,2,4]oxadiazol-5-yl)-2-(4-trifluoromethoxybenzyl)-2,3-dihydroisoindol-1-one having the following structure;

or a pharmaceutically acceptable salt thereof, a hydrate thereof, or a combination of said compound, salt or hydrate.

2. A pharmaceutical composition comprising a compound or a pharmaceutically acceptable salt or a hydrate or a combination according to claim 1 and a pharmaceutically acceptable carrier or excipient.

3. A method for the treatment schizophrenia, anxiety, or generalized anxiety disorder in an animal in need of such treatment, comprising the step of administering to said animal a therapeutically effective amount of a compound or a pharmaceutically acceptable salt or a hydrate or a combination according to claim 1 .

4. A method for the treatment schizophrenia, anxiety, or generalized anxiety disorder in an animal in need of such treatment, comprising the step of administering to said animal a therapeutically effective amount of a pharmaceutical composition according to claim 2 .

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 19, 2008
From: CLAYTON, JOSHUA; EGLE, IAN; EMPFIELD, JAMES; ISAAC, METHVIN; SLASSI, ABDELMALIK; FOLMER, JAMES; MA, FUPENG
To: ASTRAZENECA AB
Reel/Frame 021562/0768 →