IP Library Granted Patent US 8,106,058
Granted Patent B2
US 8,106,058 · App. 12/162,395 · Granted Jan 31, 2012

Anti-arenaviral compounds

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Quick Facts
Patent No.
US 8,106,058
App. No.
12/162,395
Granted
Jan 31, 2012
Kind
B2
Abstract

Described herein are 4-methyl-piperazine-1-carbothioic acid amide derivatives and analogs, as well as compositions containing the same, for the treatment or prophylaxis of viral infections and diseases associated therewith, particularly those viral infections and associated diseases caused by hemorrhagic fever viruses, such as Arenaviruses.

Claims (4)

1. A method of treating an arenavirus infection comprising administering to a subject an effective amount of a compound selected from the group consisting of 4-methyl-piperazine-1-carbothioic acid (3,4-dichloro-phenyl)-amide and 4-ethyl-piperazine-1-carbothioic acid (3,4-dichloro-phenyl)-amide.

2. The method according to claim 1 further comprising administering to the subject an additional antiviral agent selected from the group consisting of zidovudine, acyclovir, ganciclovir, vidarabidine, idoxuridine, trifluridine, foscarnet, interferon, amantadine, rimantadine, and ribavirin.

3. A method for the treatment of an arenavirus infection comprising administering to a mammal in need thereof, an effective amount of 4-methyl-piperazine-carbothioic acid (3,4-dichloro-phenyl)-amide.

4. A method for the treatment of an arenavirus infection comprising administering to a mammal in need thereof, an effective amount of 4-ethyl-piperazine-1-carbothioic acid (3,4-dichloro-phenyl)-amide.

Assignments (6)
RELEASE OF SECURITY INTEREST Recorded Apr 2, 2015
From: GENERAL ELECTRIC CAPITAL CORPORATION, AS AGENT
To: SIGA TECHNOLOGIES, INC.
Reel/Frame 035319/0001 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2014
From: SIGA TECHNOLOGIES INC.
To: KINETA FOUR LLC
Reel/Frame 033588/0427 →
RELEASE OF SECURITY INTEREST Recorded Aug 14, 2014
From: GENERAL ELECTRIC CAPITAL CORPORATION
To: SIGA TECHNOLOGIES INC.
Reel/Frame 033544/0324 →
SECURITY AGREEMENT Recorded Dec 31, 2012
From: SIGA TECHNOLOGIES, INC.
To: GE CAPITAL EQUITY INVESTMENTS, INC. C/O GE HEALTHCARE FINANCIAL SERVICES, INC.
Reel/Frame 029557/0771 →
CONFIRMATORY LICENSE Recorded Dec 22, 2011
From: SIGA TECHNOLOGIES, INC.
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 027437/0889 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 4, 2008
From: HRUBY, DENNIS E.; BOLKEN, TOVE C.; DAI, DONGCHENG
To: SIGA TECHNOLOGIES, INC.
Reel/Frame 021780/0824 →