IP Library Granted Patent US 7,687,662
Granted Patent B2
US 7,687,662 · App. 12/217,243 · Granted Mar 30, 2010

Proteasome inhibitors

Assignee: Millennium Pharmaceuticals, Inc.
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Quick Facts
Patent No.
US 7,687,662
App. No.
12/217,243
Granted
Mar 30, 2010
Kind
B2
Abstract

The present invention provides novel compounds useful as proteasome inhibitors. The invention also provides pharmaceutical compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various diseases.

Claims (7)

1. A compound of formula (I):

wherein:

Z 1 and Z 2 together form a moiety derived from a boronic acid complexing agent; and

Ring A is selected from the group consisting of

2. The compound of claim 1 , wherein Ring A is selected from the group consisting of

3. A pharmaceutical composition comprising a compound of claim 1 and a pharmaceutically acceptable carrier.

4. A pharmaceutical composition comprising a compound of claim 2 and a pharmaceutically acceptable carrier.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 10, 2022
From: MILLENNIUM PHARMACEUTICALS, INC.
To: TAKEDA PHARMACEUTICAL COMPANY LIMITED
Reel/Frame 061726/0250 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 16, 2013
From: OLHAVA, EDWARD J.; DANCA, MIHAELA DIANA
To: MILLENNIUM PHARMACEUTICALS INC.
Reel/Frame 030221/0518 →
Continuity (2)
Continuation 1189041200 · Aug 6, 2007
Related Publication 20090042836A1 · Feb 12, 2009