IP Library Granted Patent US 9,334,281
Granted Patent B2
US 9,334,281 · App. 12/231,988 · Granted May 10, 2016

Fluorochromes for organelle tracing and multi-color imaging

Inventors: Wayne Forrest Patton (Dix Hills, NY); Praveen Pande (Holbrook, NY); Yuejun Xiang (Bayside, NY); Zaiguo Li (Fresh Meadows, NY); James J. Donegan (Long Beach, NY); Elazar Rabbani (New York, NY)
Assignee: ENZO LIFE SCIENCES, INC.
C07D487/06C07C225/34C07C225/36C07C229/18C07C335/20C07D213/74C07D295/135C07F9/5304C07F9/65038C09B1/005C09B1/51C09B1/512C09B1/5155C40B40/04G01N33/5005G01N33/5011C07C2103/24
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Quick Facts
Patent No.
US 9,334,281
App. No.
12/231,988
Granted
May 10, 2016
Kind
B2
Abstract

Provided are compounds, methods and kits for identifying in cells of interest organelles including nuclei and a wide variety of organelles other than nuclei (non-nuclear organelles), as well as cell regions or cell domains. These compounds and methods can be used with other conventional detection reagents for identifying the location or position or quantity of organelles and even for distinguishing between organelles in cells of interest.

Claims (21)

1. A compound selected from:

2. The compound having the structure

3. A multimeric compound comprising two or more of the compounds of claim 1 or 2 joined together through a linkage group comprising a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkenyl group, a substituted or unsubstituted heteroalkyl group, a substituted or unsubstituted heteroalkenyl group comprising an amide, or one or more substituted or unsubstituted aromatic rings.

4. A compound comprising two organelle-targeting fluorochrome compounds having the structure:

wherein R 1 -R 4 and R 5 -R 8 are independently selected from

H,

OH,

a halide,

a nitro group,

a substituted amine,

a CN group,

a charged group comprising a salt of an organic acid, an onium group or a protonated amine, wherein

said salt of an organic acid comprises a sulfate, a sulfonate, a phosphate, a phosphonate, a carboxylate, a borate, or a combination thereof, and

said onium group comprises a quaternary ammonium, a sulfonium, a phosphonium, or a combination thereof,

a substituted or unsubstituted alkyl or alkenyl group,

a substituted or unsubstituted amine, and

a thiourea group;

wherein only one member of R 1 -R 8 comprises the structure NH-A-R a R b , wherein A is a C 2-8 alkylene group and R a and R b are independently selected from H, a C 1-4 alkyl, a C 2-4 hydroxyalkyl and a C 2-4 aminoalkyl; and

wherein said two or more compounds are joined together through a linkage group comprising a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkenyl group, a substituted or unsubstituted heteroalkyl group, a substituted or unsubstituted heteroalkenyl group comprising an amide, or one or more substituted or unsubstituted aromatic rings.

5. The compound of claim 4 selected from

6. A compound selected from the group consisting of

Assignments (3)
RELEASE OF SECURITY INTEREST Recorded Jul 24, 2023
From: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
To: ENZO BIOCHEM, INC.; ENZO CLINICAL LABS, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP; ENZO LIFE SCIENCES, INC.
Reel/Frame 064369/0031 →
SECURITY INTEREST Recorded Apr 3, 2023
From: ENZO LIFE SCIENCES, INC.; ENZO CLINICAL LABS, INC.; ENZO BIOCHEM, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP
To: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
Reel/Frame 063239/0103 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 19, 2009
From: PATTON, WAYNE FORREST; PANDE, PRAVEEN; XIANG, YUEJUN; LI, ZAIGUO; DONEGAN, JAMES J.; RABBANI, ELAZAR
To: ENZO LIFE SCIENCES, INC. C/O ENZO BIOCHEM, INC.
Reel/Frame 022178/0769 →
Continuity (1)
Related Publication 20100062429A1 · Mar 11, 2010