Granted Patent
B2
US 7,897,763 · App. 12/257,558 · Granted Mar 1, 2011
Process for the preparation of substituted phenylalanines
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Abstract
Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
Claims (7)
1. A compound of the formula:
or a salt thereof, wherein:
P 1 is R 1 , aryl-alkyl, heteroaryl-alkyl, or —C(O)R 13 ;
P 2 is aryl-alkyl, heteroaryl-alkyl, or —C(O)R 13 ;
R 1 is hydrogen or optionally substituted alkyl, alkyl-aryl, alkyl-heterocycle, aryl, or heterocycle; and
each R 13 is independently alkyl, aryl-alkyl, aryl, heterocycle, alkoxy, aryloxy, or aryl-alkoxy.
2. The compound of claim 1 , which is of the formula:
Assignments (10)
RELEASE OF INTELLECTUAL PROPERTY SECURITY AGREEMENT RECORDED AT R/F 63227/0852
Recorded Jan 7, 2025
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Recorded Apr 4, 2023
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Recorded Sep 30, 2020
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ASSIGNMENT OF ASSIGNOR'S INTEREST
Recorded Sep 14, 2020
From: LEXICON PHARMACEUTICALS, INC.
To: TERSERA THERAPEUTICS LLC
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RELEASE OF SECURITY INTEREST
Recorded Sep 14, 2020
From: BIOPHARMA CREDIT PLC
To: LEXICON PHARMACEUTICALS, INC.
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SECURITY INTEREST
Recorded Sep 9, 2020
From: TERSERA THERAPEUTICS LLC
To: NEWSTONE CAPITAL PARTNERS, LLC
Reel/Frame 053721/0037 →
SECURITY INTEREST
Recorded Dec 20, 2017
From: LEXICON PHARMACEUTICALS, INC.
To: BIOPHARMA CREDIT PLC
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