Soil treating agent or seed treating agent comprising quinoline compounds or salts thereof as active ingredient, or method for preventing plant diseases by using the same
View Patent ↗A soil treating agent or a seed treating agent having excellent prevention effects against various plant pathogens (particularly against rice blast) is provided. A soil treating agent or seed treating agent, comprising one or more compounds of the general formula (Ia), (Ib) or (Ic): (wherein R 1 , R 2 : C 1 -C 6 alkyl (may be substituted), aryl (may be substituted), heteroaryl (may be substituted), aralkyl (may be substituted) and the like; R 3 , R 4 : H, C 1 -C 6 alkyl (may be substituted), halogen, C 1 -C 6 alkoxy and the like; X: halogen, C 1 -C 6 alkyl (may be substituted), C 2 -C 6 alkenyl (may be substituted), C 2 -C 6 alkynyl (may be substituted), aryl (may be substituted), heteroaryl (may be substituted), C 1 -C 6 alkoxy and the like; Y: halogen, C 1 -C 6 alkyl, C 1 -C 6 alkoxy, OH; n: 0 to 4; m: 0 to 6) or salts thereof as an active ingredient.
1. A method for treating or controlling a plant disease selected from the group consisting of rice blast, Bakanae disease of rice, Fusarium blight of wheat, seedling blight of wheat, Rhizoctonia seedling blight of cucumber, Pythium damping-off of cucumber, Fusarium wilt of cucumber, damping off of tomato and Fusarium wilt of tomato comprising treating plant seeds with a seed treating composition comprising one or more compounds selected from the group consisting of
3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoguinolin-1-yl)quinoline,
8-fluoro-3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoquinolin-1-yl)guinoline,
3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoquinolin-1-yl)-8-methylquinoline,
3-(4,4-difluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline,
3-(4,4,5-trifluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline,
5-fluoro-3,3,4,4-tetramethyl-8b-quinolin-3-yl-4,8b-dihydro-3H-oxazireno[3,2-a]isoquinoline,
4,4,5-trifluoro-3,3-dimethyl-8b-quinolin-3-yl-4,8b-dihydro-3H-oxazireno[3,2-a]isoquinoline,
3-(5-fluoro-3,3,4,4-tetramethyl-2-oxido-3,4-dihydroisoquinolin-1-yl)quinoline, and
3-(4,4,5-trifluoro-3,3-dimethyl-2-oxido-3,4-dihydroisoquinolin-1-yl)quinoline, as an active ingredient,
wherein the treatment of the plant seeds is carried out by spraying the composition on the plant seeds, coating the plant seeds with the composition, dipping the plant seeds into the composition or dust-coating the plant seeds with the composition, to control pathogens which adhere to the surface of plant seeds and to control pathogens which infect the inside of the plant seeds, or to control an onset of said disease caused by a pathogen or an onset of said disease which is observed after the sowing of the plant seeds.
2. The method according to claim 1 , wherein the compounds are applied in an amount of 0.001 to 50 g per kg of the plant seeds in a case where the plant seeds are disinfected.
3. The method according to claim 1 , wherein the compounds are applied in an amount of 0.01 to 10 g per kg of the plant seeds in a case where the plant seeds are disinfected.
4. The method according to claim 1 , wherein the compound is selected from the group consisting of
3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoquinolin-1-yl)quinoline,
3-(4,4-difluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline,
3-(4,4,5-trifluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline,
3-(5-fluoro-3,3,4,4-tetramethyl-2-oxido-3,4-dihydroisoquinolin-1-yl)quinoline,
5-fluoro-3,3,4,4-tetramethyl-8b-quinolin-3-yl-4,8b-dihydro-3H-oxazireno[3,2-a]isoquinoline and
3-(4,4,5-trifluoro-3,3-dimethyl-2-oxido-3,4-dihydroisoquinolin-1-yl)quinoline.
5. The method according to claim 1 , wherein the compound is 3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoquinolin-1-yl)quinoline.
6. The method according to claim 1 , wherein the compound is 5-fluoro-3,3,4,4-tetramethyl-8b-quinolin-3-yl-4,8b-dihydro-3H-oxazireno[3,2-a]isoquinoline.
7. The method according to claim 1 , wherein the compound is 3-(5-fluoro-3,3,4,4-tetramethyl-2-oxido-3,4-dihydroisoquinolin-1-yl)quinoline.