IP Library Granted Patent US 8,658,649
Granted Patent B2
US 8,658,649 · App. 12/401,254 · Granted Feb 25, 2014

Kinase inhibitor

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Quick Facts
Patent No.
US 8,658,649
App. No.
12/401,254
Granted
Feb 25, 2014
Kind
B2
Abstract

The invention is directed to a compound of formula (I): and the prodrugs, and pharmaceutically acceptable salts and solvates of such compounds and their prodrugs. Such a compound has valuable pharmaceutical properties, in particular the ability to inhibit protein kinases.

Claims (8)

1. A compound of formula (I):

or a corresponding N-oxide, or a prodrug; or a pharmaceutically acceptable salt of such of compound; or an N-oxide or a prodrug of the salt.

2. A pharmaceutical composition, comprising a compound according to claim 1 , together with at least one pharmaceutically acceptable carrier or excipient.

3. The compound according to claim 1 , wherein the salt is selected from:

hydrochloride, hydrobromide, sulphate, phosphate, nitrate, sulfamate, acetate, citrate, lactate, tartrate, malonate, oxalate, salicylate, propionate, succinate, fumarate, maleate, methylene-bis-b-hydroxynaphthoate, gentisate, isethionate, di-p-toluoyltartrate, methane-sulfonate, ethanesulfonate, benzenesulfonate, p-toluenesulfonate, cyclohexylsulfamate and quinate.

4. The compound according to claim 1 , wherein the salt is hydrochloride.

5. The compound according to claim 1 , wherein the salt is acetate.

6. The compound according to claim 1 , wherein the salt is citrate.

Assignments (2)
CHANGE OF NAME Recorded Aug 2, 2011
From: SANOFI-AVENTIS
To: SANOFI
Reel/Frame 026686/0522 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 16, 2009
From: GILLESPY, TIMOTHY; EYNOTT, PAUL; ALLEN, ELIZABETH; YU, KIN; ZILBERSTEIN, ASHER
To: SANOFI-AVENTIS
Reel/Frame 023241/0253 →