IP Library Granted Patent US 8,247,579
Granted Patent B2
US 8,247,579 · App. 12/522,563 · Granted Aug 21, 2012

Spirocyclic tetronic acid derivatives

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Quick Facts
Patent No.
US 8,247,579
App. No.
12/522,563
Granted
Aug 21, 2012
Kind
B2
Abstract

The present invention relates to novel spirocyclic tetronic acid derivatives of the formula (I) in which R 1 , R 2 and R 3 have the meanings given in the description, to a plurality of processes for their preparation and to their use as pesticides.

Claims (21)

1. A compound of formula (I-3)

2. A process for preparing a compound of the formula (I-3) according to claim 1 , comprising reacting a compound of formula (II)

α) with a compound of formula (III)

in which

R 1 is C 2 H 5 , R 2 and R 3 are CH 3 , and

Hal represents halogen

or

β) with a carboxylic anhydride of formula (IV)

in which

R 1 is C 2 H 5 , R 2 and R 3 are CH 3 ,

optionally in the presence of a diluent and optionally in the presence of an acid binder;

or

γ) with an activated carboxylic acid derivative of formula (V)

in which

R 1 is C 2 H 5 , R 2 and R 3 are CH 3 ,

and

U represents a leaving group introduced by a carboxylic acid-activating reagent,

optionally in the presence of a diluent and optionally in the presence of an acid binder.

3. A pesticide, comprising the compound of formula (I-3) according to claim 1 .

4. A method for controlling animal pests, comprising allowing the compound of formula (I-3) according to claim 1 to act on pests, their habitat, or combinations thereof.

5. A process for preparing a pesticide, comprising mixing the compound of formula (I-3) according to claim 1 with an extender, a surfactant, or a combination thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 23, 2015
From: BAYER CROPSCIENCE AG
To: BAYER INTELLECTUAL PROPERTY GMBH
Reel/Frame 035005/0367 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 11, 2010
From: FISCHER, REINER, DR.; BRETSCHNEIDER, THOMAS, DR.; SCHULTE, HUBERTUS, DR.; KRAUTSTRUNK, GERHARD, DR.; ARNOLD, CHRISTIAN, DR.; SANWALD, ERICH, DR.
To: BAYER CROPSCIENCE AG
Reel/Frame 024068/0485 →