IP Library Granted Patent US 8,309,141
Granted Patent B2
US 8,309,141 · App. 12/527,302 · Granted Nov 13, 2012

Herbal composition PHY906 and its use in chemotherapy

Assignee: Yale University
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Quick Facts
Patent No.
US 8,309,141
App. No.
12/527,302
Granted
Nov 13, 2012
Kind
B2
Abstract

This invention provides herbal compositions useful for increasing the therapeutic index of chemotherapeutic compounds. This invention also provides methods useful for improving the quality of life of an individual undergoing chemotherapy. Furthermore, this invention improves the treatment of disease by increasing the therapeutic index of chemotherapy drugs by administering the herbal composition PHY906 to a mammal undergoing such chemotherapy.

Claims (42)

1. A method of treating cancer in a mammal comprising co-administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

2. The method of claim 1 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via oral or parenteral route.

3. The method of claim 2 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via intravenous route.

4. The method of claim 1 , wherein the herbal preparation consists of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora, and one or more pharmaceutically acceptable carrier.

5. The method of claim 1 , wherein the herbal preparation is administered before the administration of the chemotherapeutic formulation.

6. The method of claim 1 , wherein the herbal preparation is administered after the administration of the chemotherapeutic formulation.

7. The method of claim 1 , wherein the herbal preparation is administered concurrently with the administration of the chemotherapeutic formulation.

8. A method of relieving side effects of a chemotherapeutic compound in a mammal comprising co-administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

9. The method of claim 8 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via oral or parenteral route.

10. The method of claim 9 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via intravenous route.

11. The method of claim 8 , wherein the herbal preparation consists of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora, and one or more pharmaceutically acceptable carrier.

12. The method of claim 8 , wherein the herbal preparation is administered before the administration of the chemotherapeutic formulation.

13. The method of claim 8 , wherein the herbal preparation is administered after the administration of the chemotherapeutic formulation.

14. The method of claim 8 , wherein the herbal preparation is administered concurrently with the administration of the chemotherapeutic formulation.

15. A method of enhancing anticancer activity of a chemotherapeutic compound in a mammal comprising administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

16. The method of claim 15 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via oral or parenteral route.

17. The method of claim 16 , wherein the herbal preparation is administered via oral route, and the chemotherapeutic formulation is administered via intravenous route.

18. The method of claim 15 , wherein the herbal preparation consists of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora, and one or more pharmaceutically acceptable carrier.

19. The method of claim 15 , wherein the herbal preparation is administered before the administration of the chemotherapeutic formulation.

20. The method of claim 15 , wherein the herbal preparation is administered after the administration of the chemotherapeutic formulation.

21. The method of claim 15 , wherein the herbal preparation is administered concurrently with the administration of the chemotherapeutic formulation.

22. A method of treating cancer in a mammal comprising separately administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

23. The method of claim 22 wherein the chemotherapeutic formulation comprises 5-fluorouracil (5-FU) and leucovorin (LV).

24. The method of claim 22 wherein the chemotherapeutic formulation comprises irinotecan (CPT-11), 5-fluorouracil (5-FU), and leucovorin (LV).

25. A method of relieving side effects of a chemotherapeutic compound in a mammal comprising separately administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

26. The method of claim 25 wherein the chemotherapeutic formulation comprises 5-fluorouracil (5-FU) and leucovorin (LV).

27. The method of claim 25 wherein the chemotherapeutic formulation comprises irinotecan (CPT-11), 5-fluorouracil (5-FU), and leucovorin (LV).

28. A method of enhancing anticancer activity of a chemotherapeutic compound in a mammal comprising separately administering a therapeutically effective amount of

i) an herbal preparation consisting essentially of Scutellaria baicalensis, Glycyrrhiza uralensis, Ziziphus jujuba and Paeonia lactiflora; and

ii) a chemotherapeutic formulation comprising a chemotherapeutic compound selected from the group consisting of irinotecan (CPT-11), 5-fluorouracil (5-FU), etoposide (VP-16), beta-L-Dioxolane-cytidine (L-OddC), leucovorin (LV) and combinations thereof.

29. The method of claim 28 wherein the chemotherapeutic formulation comprises 5-fluorouracil (5-FU) and leucovorin (LV).

30. The method of claim 28 wherein the chemotherapeutic formulation comprises irinotecan (CPT-11), 5-fluorouracil (5-FU), and leucovorin (LV).

Assignments (11)
RELEASE OF SECURITY INTEREST Recorded Oct 29, 2021
From: MACQUARIE US TRADING LLC
To: KADMON CORPORATION, LLC
Reel/Frame 057973/0751 →
TERMINATION OF PATENT AND TRADEMARK SECURITY AGREEMENT Recorded Nov 25, 2019
From: PERCEPTIVE CREDIT OPPORTUNITIES FUND, LP
To: KADMON CORPORATION, LLC
Reel/Frame 051106/0677 →
SECURITY INTEREST Recorded Sep 8, 2015
From: KADMON CORPORATION, LLC
To: MACQUARIE US TRADING LLC
Reel/Frame 036573/0001 →
RELEASE OF SECURITY INTEREST Recorded Sep 1, 2015
From: MACQUARIE US TRADING LLC
To: KADMON CORPORATION, LLC
Reel/Frame 036518/0862 →
SECURITY INTEREST Recorded Aug 31, 2015
From: KADMON CORPORATION, LLC
To: PERCEPTIVE CREDIT OPPORTUNITIES FUND, LP
Reel/Frame 036515/0084 →
SECURITY AGREEMENT Recorded Jun 25, 2013
From: KADMON CORPORATION LLC
To: MACQUARIE US TRADING LLC
Reel/Frame 030679/0212 →
SECURITY AGREEMENT Recorded Jun 25, 2013
From: KADMON CORPORATION LLC
To: MACQUARIE US TRADING LLC
Reel/Frame 030679/0116 →
SECURITY AGREEMENT Recorded Nov 23, 2011
From: KADMON CORPORATION, LLC
To: CORTLAND CAPITAL MARKET SERVICES LLC, AS ADMINISTRATIVE AGENT
Reel/Frame 027278/0787 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 14, 2011
From: PHYTOCEUTICA, INC.
To: YALE UNIVERSITY
Reel/Frame 027063/0387 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 1, 2010
From: LIU, SHWU-HUEY
To: PHYTOCEUTICA, INC.
Reel/Frame 024624/0740 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 1, 2010
From: JIANG, ZAOLI; CHENG, YUNG-CHI
To: YALE UNIVERSITY
Reel/Frame 024624/0724 →
Continuity (6)
Continuation In Part 11100433 · Apr 7, 2005
Continuation In Part 10220876
Continuation In Part 09522055 · Mar 9, 2000
Provisional Application 60901310 · Feb 15, 2007
Provisional Application 60625943 · Nov 9, 2004
Related Publication 20100255129A9 · Oct 7, 2010