IP Library Granted Patent US 8,486,961
Granted Patent B2
US 8,486,961 · App. 12/539,869 · Granted Jul 16, 2013

Pyrrolo[4,3,2-de]quinolin-8-amine compounds and methods of their preparation and use

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Quick Facts
Patent No.
US 8,486,961
App. No.
12/539,869
Granted
Jul 16, 2013
Kind
B2
Abstract

The present invention relates to compounds of formula I: methods of their use, processes for their preparation and isolated actinomycetes strains capable of preparing pyrrolo[4,3,2-de]quinolin-8-amine compounds.

Claims (3)

1. The compound (E)-N-(8-amino-4-(3-methoxyacryloyl)pyrrolo[4,3,2-de]quinolin-6-yl)isobutyramide, or a tautomer, stereoisomer or pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising the compound of claim 1 or a tautomer, stereoisomer or pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier.

3. The pharmaceutical composition of claim 2 , wherein said compound, tautomer, stereoisomer or pharmaceutically acceptable salt thereof is present in sufficient amount to treat prostate cancer or breast cancer in an patient.

Assignments (2)
CHANGE OF NAME Recorded Jun 16, 2010
From: WYETH
To: WYETH LLC
Reel/Frame 024541/0922 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 23, 2009
From: HE, MIN; JANSO, JEFFREY EDWIN; YU, KER; MCDONALD, LEONARD ALEXANDER; BARBIERI, LAUREL RITA; GOPALSAMY, ARIAMALA
To: WYETH
Reel/Frame 023270/0213 →