IP Library › Patent Application 12743560
Patent Application
App. No. 12/743,560

Peripheral Phenolic Opioid Antagonist

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Quick Facts
Patent No.
US None
App. No.
12/743,560
Abstract

N-Methyldiprenorphine, useful as an opioid antagonist.

Claims (6)

1 . N-methyldiprenorphine.

2 . A process for the preparation of N-methyldiprenorphine, which comprises methylating diprenorphine.

3 . A pharmaceutical composition, which comprises N-methyldiprenorphine and a pharmaceutically acceptable carrier.

4 . N-methyldiprenorphine, for use in therapy.

5 . N-methyldiprenorphine, for use as an opioid antagonist.

6 . A method of antagonising the action of an opioid in a patient undergoing opioid treatment, which comprises administering to said patient an effective amount of N-methyldiprenorphine.

Assignments (2)
CHANGE OF NAME Recorded May 9, 2012
From: PHARMACOFORE, INC.
To: SIGNATURE THERAPEUTICS, INC.
Reel/Frame 028185/0192 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 28, 2010
From: JENKINS, THOMAS E.; WRAY, JONATHAN W.
To: PHARMACOFORE, INC.
Reel/Frame 024459/0573 →