IP Library Patent Application 12871860
Patent Application
App. No. 12/871,860

COMBINATIONS OF RETIGABINE AND SODIUM CHANNEL INHIBITORS OR SODIUM CHANNEL-INFLUENCING ACTIVE COMPOUNDS FOR TREATING PAINS

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Quick Facts
Patent No.
US None
App. No.
12/871,860
Abstract

The invention relates to pharmaceutical combinations of retigabine and sodium channel inhibitors for treating, pains which are accompanied by an increase in muscle tone.

Claims (11)

1 . The use of retigabine or its pharmaceutically utilizable salts in combination with sodium channel-inhibiting or -influencing substances, or of their therapeutically utilizable salts, for treating pains which are accompanied by an increase in muscle tone.

2 . The use as claimed in claim 1 , wherein the sodium channel-inhibiting or -influencing substances employed are tolperisone or its analogs eperisone or silperisone, or riluzole, propafenone, lidocaine, flecainide or metixen, or their pharmaceutically utilizable salts.

3 . The use as claimed in claim 1 , wherein the sodium channel-inhibiting or -influencing substances employed are tolperisone or its analogs, such as eperisone or silperisone, or their pharmaceutically utilizable salts.

4 . The use of retigabine in combination with tolperisone or its analogs, such as eperisone or silperisone, or their pharmaceutically utilizable salts, for treating pains which are accompanied by an increase in muscle tone.

5 . The use as claimed in claim 1 , for treating pains associated with neuralgias.

6 . The use as claimed in claim 1 , for treating pains associated with arthritis and arthrosis.

7 . The use as claimed in claim 1 , for treating pains associated with chronic or episodic tension headache.

8 . The use as claimed in claim 1 , for treating pains associated with lower spastic paraparesis syndrome (e.g. lower paraspasm, transverse myelitis, multiple sclerosis, heritable inferior spastic paraplegia (Stuempel paraplegia), disturbances of the spinal blood circulation and cerebral paralysis involving lower spastic paresis).

9 . The use as claimed in claim 1 , for treating pains associated with tetraparesis in connection with cervical myelopathy, cervical brachialgia or vertebral dysplasia.

10 . The use as claimed in claim 1 , for treating pains associated with Parkinson's disease.

11 . The use of retigabine or its pharmaceutically utilizable salts in combination with sodium channel-inhibiting or -influencing substances, and of their therapeutically utilizable salts, for producing a medicament for oral, rectal, intravenous, transdermal or subcutaneous or intracutaneous administration for treating pains which are accompanied by an increase in muscle tone.

Assignments (3)
RELEASE OF SECURITY INTEREST Recorded Apr 8, 2025
From: BARCLAYS BANK PLC, AS COLLATERAL AGENT
To: SOLTA MEDICAL, INC.; PRECISION DERMATOLOGY, INC.; BAUSCH HEALTH IRELAND LIMITED (F/K/A/ VALEANT PHARMACEUTICALS IRELAND LIMITED); SALIX PHARMACEUTICALS, INC.; SALIX PHARMACEUTICALS, LTD; SANTARUS, INC.; MEDICIS PHARMACEUTICAL CORPORATION; HUMAX PHARMACEUTICAL S.A.; SOLTA MEDICAL IRELAND LIMITED; BAUSCH & LOMB MEXICO, S.A. DE C.V.; BAUSCH+LOMB OPS B.V.; BAUSCH HEALTH AMERICAS, INC.; BAUSCH HEALTH COMPANIES INC.; BAUSCH HEALTH HOLDCO LIMITED; BAUSCH HEALTH MAGYARORSZAG KFT (A/K/A BAUSCH HEALTH HUNGARY LLC); BAUSCH HEALTH POLAND SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA (F/K/A VALEANT PHARMA POLAND SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA); BAUSCH HEALTH US, LLC; BAUSCH HEALTH, CANADA INC. / SANTE BAUSCH, CANADA INC.; ICN POLFA RZESZOW SPOLKA AKCYJNA (A/K/A ICN POLFA RZESZOW S.A.); ORAPHARMA, INC.; PRZEDSIEBIORSTWO FARMACEUTYCZNE JELFA SPOLKA AKCYJNA (A/K/A PRZEDSIEBIORSTWO FARMACEUTYCZNE JELFA S.A.); SOLTA MEDICAL DUTCH HOLDINGS B.V.; V-BAC HOLDING CORP.; VRX HOLDCO LLC; 1261229 B.C. LTD.; 1530065 B.C. LTD.
Reel/Frame 070778/0199 →
NOTICE OF SUCCESSION OF AGENCY Recorded Jan 9, 2015
From: GOLDMAN SACHS LENDING PARTNERS, LLC
To: BARCLAYS BANK PLC, AS SUCCESSOR AGENT
Reel/Frame 034749/0689 →
SECURITY AGREEMENT Recorded Jul 18, 2011
From: VALEANT PHARMACEUTICALS INTERNATIONAL, A DELAWARE CORPORATION; ATON PHARMA, INC., A DELAWARE CORPORATION; CORIA LABORATORIES, LTD., A DELAWARE CORPORATION; DOW PHARMACEUTICAL SCIENCES, INC., A DELAWARE CORPORATION; VALEANT PHARMACEUTICALS NORTH AMERICA LLC, A DELAWARE LLC; PRESTWICK PHARMACEUTICALS, INC., A DELAWARE CORPORATION; VALEANT BIOMEDICALS, INC., A DELAWARE CORPORATION
To: GOLDMAN SACHS LENDING PARTNERS LLC, AS COLLATERAL AGENT
Reel/Frame 026606/0061 →