IP Library Granted Patent US 9,173,862
Granted Patent B2
US 9,173,862 · App. 12/937,669 · Granted Nov 3, 2015

Methods and compositions for treating and identifying compounds to treat age-related macular degeneration

Inventors: Brian McKay (Marana, AZ); John A. Martens (Tucson, AZ)
Assignee: Arizona Board of Regents, a Body Corporate of the State of Arizona, Acting for and on Behalf of the University of Arizona
A61K31/195A61K31/00A61K31/07A61K31/355A61K31/375A61K33/30A61K33/34
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Quick Facts
Patent No.
US 9,173,862
App. No.
12/937,669
Granted
Nov 3, 2015
Kind
B2
Abstract

The present invention provides methods for treating or limiting development of age-related macular degeneration, as well as methods for identifying compound suitable for such use.

Claims (26)

1. A method for treating age-related macular degeneration (AMD), comprising administering to a subject with AMD an amount of an agonist of the OA1 receptor selected from the group consisting of L-DOPA, an L-DOPA analogue, and pharmaceutically acceptable salts thereof, effective for treating AMD.

2. The method of claim 1 , wherein the agonist comprises L-DOPA, or a pharmaceutically acceptable salt thereof.

3. The method of claim 1 , wherein the L-DOPA analogue comprises an L-DOPA prodrug, or a pharmaceutically acceptable salt thereof.

4. The method of claim 3 , wherein the L-DOPA prodrug comprises an L-DOPA ester, or a pharmaceutically acceptable salt thereof.

5. The method of claim 3 , wherein the L-DOPA prodrug comprises a bile acid conjugate of L-DOPA, or a pharmaceutically acceptable salt thereof.

6. The method of claim 3 wherein the L-DOPA prodrug comprises a di- or tri-peptide L-DOPA analogue, or a pharmaceutically acceptable salt thereof.

7. The method claim 1 , wherein the subject is over the age of 60.

8. The method of claim 1 , wherein the subject has wet AMD.

9. The method of claim 1 , wherein the subject has dry AMD.

10. The method of claim 1 , further comprising administering to the subject a combination of a vitamin C source, a vitamin E source, a beta-carotene source, a zinc source, and a copper source.

11. The method of claim 10 , comprising administering

between 450 mg and 600 mg vitamin C;

between 400 IU and 540 IU vitamin E;

between 17.2 mg and 28 mg beta-carotene;

between 68 mg and 100 mg zinc; and

between 1.6 mg and 2.4 mg copper.

12. The method claim 2 , wherein the subject is over the age of 60.

13. The method of claim 2 , wherein the subject has wet AMD.

14. The method of claim 2 , wherein the subject has dry AMD.

15. The method of claim 2 , further comprising administering to the subject a combination of a vitamin C source, a vitamin E source, a beta-carotene source, a zinc source, and a copper source.

16. The method of claim 15 , comprising administering

between 450 mg and 600 mg vitamin C;

between 400 IU and 540 IU vitamin E;

between 17.2 mg and 28 mg beta-carotene;

between 68 mg and 100 mg zinc; and

between 1.6 mg and 2.4 mg copper.

Assignments (2)
CONFIRMATORY LICENSE Recorded May 23, 2011
From: UNIVERSITY OF ARIZONA
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 026328/0501 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 5, 2010
From: MCKAY, BRIAN
To: ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA, ACTING FOR AND ON BEHALF OF THE UNIVERSITY OF ARIZONA
Reel/Frame 025328/0020 →
Continuity (2)
Provisional Application 61124624 · Apr 18, 2008
Related Publication 20110044908A1 · Feb 24, 2011