IP Library Granted Patent US 8,138,213
Granted Patent B2
US 8,138,213 · App. 13/166,294 · Granted Mar 20, 2012

Isoxazoline-substituted benzamide compound and pesticide

Assignee: Nissan Chemical Industries, Ltd.
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Quick Facts
Patent No.
US 8,138,213
App. No.
13/166,294
Granted
Mar 20, 2012
Kind
B2
Abstract

A 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula (2) or a salt thereof: wherein A1 is a carbon atom or nitrogen atom; X1 is selected from the group consisting of a halogen atom, —SF5, C1-C6haloalkyl, hydroxy C1-C6haloalkyl, C1-C6alkoxy C1-C6haloalkyl, C1-C6haloalkoxy C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6haloalkoxy, C1-C3haloalkoxy C1-C3haloalkoxy, C1-C6haloalkylthio, C1-C6haloalkylsulfinyl and C1-C6haloalkylsulfonyl; X2 is selected from the group consisting of a halogen atom, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, —OR5, —OSO2R5 and —S(O)rR5; Y is selected from the group consisting of a halogen atom, cyano, nitro, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkylsulfonyl, C1-C6haloalkylsulfonyl, —NHR7 and —N(R7)R6; R is selected from the group consisting of a halogen atom, cyano, nitro, —NH2, halosulfonyloxy, C1-C6alkylsulfonyloxy, C1-C6haloalkylsulfonyloxy, phenylsulfonyloxy, phenylsulfonyloxy substituted with (Z)p1 and —C(O)Ra; m1 is an integer of 0 to 2; n is an integer of 0 or 1; p1 is an integer of 1 to 5; and r is an integer of 0 to 2.

Claims (23)

1. A 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula (2) or a salt thereof:

wherein

A 1 is a carbon atom or nitrogen atom;

X 1 is selected from the group consisting of a halogen atom, —SF 5 , C 1 -C 6 haloalkyl, hydroxy C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy C 1 -C 6 haloalkyl, C 1 -C 6 haloalkoxy C 1 -C 6 haloalkyl, C 3 -C 8 halocycloalkyl, C 1 -C 6 haloalkoxy, C 1 -C 3 haloalkoxy C 1 -C 3 haloalkoxy, C 1 -C 6 haloalkylthio, C 1 -C 6 haloalkylsulfinyl and C 1 -C 6 haloalkylsulfonyl;

X 2 is selected from the group consisting of a halogen atom, cyano, nitro, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, —OR 5 , —OSO 2 R 5 and —S(O) r R 5 ,

wherein, when m1 is 2, each X 2 may be identical with or different from each other;

Y is selected from the group consisting of a halogen atom, cyano, nitro, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy, C 1 -C 4 haloalkoxy, C 1 -C 6 alkylthio, C 1 -C 6 haloalkylthio, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylsulfonyl, —NHR 7 and —N(R 7 )R 6 ;

R 3 is C 1 -C 6 haloalkyl or C 3 -C 8 halocycloalkyl;

R 5 is C 1 -C 6 alkyl or C 1 -C 6 haloalkyl;

R 6 is selected from the group consisting of C 1 -C 6 alkyl, —CHO, C 1 -C 6 alkylcarbonyl, C 1 -C 6 haloalkylcarbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 alkylthiocarbonyl, C 1 -C 6 alkoxythiocarbonyl, C 1 -C 6 alkyldithiocarbonyl, C 1 -C 6 alkylsulfonyl or C 1 -C 6 haloalkylsulfonyl,

R7 is hydrogen atom and C1-C6alkyl;

R is selected from the group consisting of a halogen atom, cyano, nitro, —NH2, halosulfonyloxy, C1-C6alkylsulfonyloxy, C1-C6haloalkylsulfonyloxy, phenylsulfonyloxy, phenylsulfonyloxy substituted with (Z) p1 and —C(O)R a ;

R a is selected from the group consisting of a halogen atom, —OH, C 1 -C 6 alkoxy, 1-pyrazolyl, 1-imidazolyl and 1-triazolyl;

Z is selected from the group consisting of a halogen atom, C 1 -C 6 alkyl and C 1 -C 6 haloalkyl,

wherein when p1 is an integer of 2 or more, each Z may be identical with or different from each other;

m1 is an integer of 0 to 2;

n is an integer of 0 or 1;

p1 is an integer of 1 to 5; and

r is an integer of 0 to 2.

2. A pesticide comprising the 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula 2 or a salt thereof according to claim 1 .

3. An agrochemical comprising the 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula 2 or a salt thereof according to claim 1 .

4. An endo- or ecto-parasiticide for mammals or birds comprising the 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula 2 or a salt thereof according to claim 1 .

5. An insecticide or acaricide comprising the 3,5-Bis (substituted aryl) substituted isoxazoline compound of formula 2 or a salt thereof according to claim 1 .

Assignments (1)
CHANGE OF NAME Recorded Sep 21, 2018
From: NISSAN CHEMICAL INDUSTRIES, LTD.
To: NISSAN CHEMICAL CORPORATION
Reel/Frame 047128/0788 →
Priority Claims (2)
JP 2004-061749 · Mar 5, 2004 · national
JP 2004-200119 · Jul 7, 2004 · national
Continuity (4)
Division 12509859 · Jul 27, 2009
Division 11514921 · Sep 5, 2006
Continuation In Part PCTJP2005004268 · Mar 4, 2005
Related Publication 20110251398A1 · Oct 13, 2011