IP Library Granted Patent US 9,346,806
Granted Patent B2
US 9,346,806 · App. 13/272,956 · Granted May 24, 2016

6-amino-purin-8-one compounds

Inventors: Keith Biggadike (Stevenage, GB); Diane Mary Coe (Stevenage, GB); Xiao Qing Lewell (Stevenage, GB); Charlotte Jane Mitchell (Stevenage, GB); Stephen Allan Smith (Stevenage, GB); Naimisha Trivedi (Stevenage, GB)
Assignee: GlaxoSmithKline LLC
C07D473/18A61K31/522C07D473/16
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Quick Facts
Patent No.
US 9,346,806
App. No.
13/272,956
Granted
May 24, 2016
Kind
B2
Abstract

Compounds of formula (I): wherein R 1 is C 1-6 alkylamino, C 1-6 alkoxy, or C 3-7 cycloalkyloxy; m is an integer having a value of 3 to 6; n is an integer having a value of 0 to 4; and salts thereof are inducers of human interferon. Compounds which induce human interferon may be useful in the treatment of various disorders, for example the treatment of allergic diseases and other inflammatory conditions for example allergic rhinitis and asthma, the treatment of infectious diseases and cancer, and may also be useful as vaccine adjuvants.

Claims (2)

1. A method of treatment of asthma, which method comprises administering to a human subject in need thereof the compound 6-amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one, or a pharmaceutically acceptable salt thereof.

2. A method of treatment of asthma, which method comprises administering to a human subject in need thereof the compound 6-amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 28, 2013
From: BIGGADIKE, KEITH; COE, DIANE MARY; LEWELL, XIAO QING; MITCHELL, CHARLOTTE JANE; SMITH, STEPHEN ALLAN; TRIVEDI, NAIMISHA
To: SMITHKLINE BEECHAM CORPORATION
Reel/Frame 030104/0001 →
CHANGE OF NAME Recorded Mar 28, 2013
From: SMITHKLINE BEECHAM CORPORATION
To: GLAXOSMITHKLINE LLC
Reel/Frame 030105/0331 →
Continuity (3)
Continuation 12537392 · Aug 7, 2009
Provisional Application 61087777 · Aug 11, 2008
Related Publication 20120035193A1 · Feb 9, 2012