IP Library Granted Patent US 8,754,090
Granted Patent B2
US 8,754,090 · App. 13/340,522 · Granted Jun 17, 2014

Use of inhibitors of bruton's tyrosine kinase (Btk)

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Quick Facts
Patent No.
US 8,754,090
App. No.
13/340,522
Granted
Jun 17, 2014
Kind
B2
Abstract

Disclosed herein are methods for treating a cancer comprising: a. administering a Btk inhibitor to a subject sufficient to result in an increase or appearance in the blood of a subpopulation of lymphocytes defined by immunophenotyping; b. determining the expression profile of one or more biomarkers from one or more subpopulation of lymphocytes; and c. administering a second agent based on the determined expression profile.

Claims (2)

1. A method for treating mantle cell lymphoma in an individual who has already received at least one prior therapy for mantle cell lymphoma comprising administering to the individual once per day between about 420 mg to about 840 mg of an oral dose of an inhibitor of Bruton's tyrosine kinase (Btk) having the structure:

2. The method of claim 1 , wherein the once per day oral dose is about 560 mg.

Assignments (5)
CORRECTIVE ASSIGNMENT TO CORRECT THE CONVEYING PARTY DATA PREVIOUSLY RECORDED ON REEL 036058 FRAME 0429. ASSIGNOR(S) HEREBY CONFIRMS THE MERGER. Recorded May 17, 2016
From: OXFORD AMHERST CORPORATION; PARMACYCLICS, INC.
To: PHARMACYCLICS, INC.
Reel/Frame 038722/0001 →
CORRECTIVE ASSIGNMENT TO CORRECT THE CONVEYING PARTY DATA PREVIOUSLY RECORDED ON REEL 036058 FRAME 0755. ASSIGNOR(S) HEREBY CONFIRMS THE MERGER AND CHANGE OF NAME. Recorded May 17, 2016
From: PHARMACYCLICS, INC.; OXFORD AMHERST LLC
To: PHARMACYCLICS LLC
Reel/Frame 038722/0043 →
MERGER Recorded Jul 10, 2015
From: OXFORD AMHERST CORPORATION
To: PHARMACYCLICS, INC.
Reel/Frame 036058/0429 →
MERGER AND CHANGE OF NAME Recorded Jul 10, 2015
From: PHARMACYCLICS, INC.; OXFORD AMHERST LLC
To: PHARMACYCLICS LLC
Reel/Frame 036058/0755 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 3, 2012
From: BUGGY, JOSEPH J.; ELIAS, LAURENCE; FYFE, GWEN; HEDRICK, ERIK; LOURY, DAVID J.; MODY, TARAK D.
To: PHARMACYCLICS, INC.
Reel/Frame 027471/0541 →