IP Library Patent Application 13482720
Patent Application
App. No. 13/482,720

METHODS OF TREATING HYPERTRIGLYCERIDEMIA

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Quick Facts
Patent No.
US None
App. No.
13/482,720
Abstract

In various embodiments, the present invention provides methods of treating and/or preventing cardiovascular-related disease and, in particular, a method of blood lipid therapy comprising administering to a subject in need thereof a pharmaceutical composition comprising eicosapentaenoic acid or a derivative thereof

Claims (18)

1 . A method of reducing triglycerides in a subject in need thereof comprising: administering to the subject having a fasting baseline triglyceride level of 500 mg/dl to about 1500 mg/dl about 2 g to per day of a pharmaceutical composition comprising at least about 90%, by weight, ethyl eicosapentaenoate for a period of 12 weeks to effect a reduction in triglycerides compared to a second subject having a fasting baseline triglyceride level of 500 mg/dl to about 1500 mg/dl who has not received the pharmaceutical composition.

2 . The method of claim 1 , wherein the pharmaceutical composition is administered to the subject 1 to 4 times per day.

3 . The method of claim 2 wherein, the pharmaceutical composition is present in one or more capsules.

4 . The method of claim 1 , wherein the subject and the second subject have one or more of: a baseline fasting non-HDL-C of about 200 mg/dl to about 300 mg/dl, a baseline fasting total cholesterol of about 250 mg/dl to about 300 mg/dl, a baseline fasting VLDL-C of about 140 mg/dl to about 200 mg/dl, and/or a baseline fasting HDL-C of about 10 mg/dl to about 80 mg/dl.

5 . The method of claim 4 , comprising administering to the subject about 2 g of the pharmaceutical composition daily for the period of 12 weeks to effect a reduction in fasting non-HDL-C and a reduction in fasting VLDL-C compared to the second subject.

6 . The method of claim 4 , comprising administering to the subject about 2 g of the pharmaceutical composition daily for the period of 12 weeks to effect a reduction in fasting triglycerides of at least about 15% compared to the second subject.

7 . A method of reducing triglycerides in a subject with very high triglycerides and in need thereof comprising, administering to the subject having a fasting baseline triglyceride level of 500 mg/dl to about 1500 mg/dl who does not receive concurrent lipid altering therapy about 2 g per day of a pharmaceutical composition comprising at least about 90%, by weight, ethyl eicosapentaenoate for a period of 12 weeks to effect a reduction in fasting triglycerides of at least about 15% without increasing LDL-C compared to a second subject having a fasting baseline triglyceride level of 500 mg/dl to about 1500 mg/dl who does not receive concurrent lipid altering therapy or the pharmaceutical composition.

8 . The method of claim 8 , wherein the pharmaceutical composition is administered to the subject 1 to 4 times per day.

9 . The method of claim 9 , wherein the pharmaceutical composition is present in one or more capsules.

10 . The method of claim 8 , wherein the subject and the second subject have one or more of: a baseline fasting non-HDL-C of about 200 mg/dl to about 300 mg/dl, a baseline fasting total cholesterol of about 250 mg/dl to about 300 mg/dl, a baseline fasting VLDL-C of about 140 mg/dl to about 200 mg/dl, and/or a baseline fasting HDL-C of about 10 mg/dl to about 80 mg/dl.

11 . The method of claim 10 , comprising administering to the subject about 2 g of the pharmaceutical composition daily for the period of 12 weeks to effect a reduction in fasting non-HDL-C and a reduction in fasting VLDL-C compared to the second subject.

12 . The method of claim 11 , comprising administering to the subject about 2 g of the pharmaceutical composition daily for the period of 12 weeks to effect a reduction in fasting triglycerides of at least about 15% compared to the second subject.

13 . The method of claim 1 , wherein the subject and the second subject consume a Western diet.

14 . The method of claim 1 , wherein the subject and the second subject do not receive a concurrent lipid altering therapy.

15 . The method of claim 14 , wherein the concurrent lipid altering therapy comprises a statin.

16 . The method of claim 7 , wherein the concurrent lipid altering therapy comprises a statin.

17 . The method of claim 16 , wherein the subject and the second subject consume a Western diet.

18 . The method of claim 17 , wherein the pharmaceutical composition comprises not more than about 0.6% by weight of any individual fatty acid other than ethyl-EPA.

Assignments (5)
RELEASE OF SECURITY INTEREST Recorded Nov 19, 2020
From: CPPIB CREDIT EUROPE S.À R.L.
To: AMARIN PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 054484/0552 →
SECURITY INTEREST Recorded Dec 21, 2017
From: AMARIN PHARMACEUTICALS IRELAND LIMITED
To: CPPIB CREDIT EUROPE S.À R.L.
Reel/Frame 044938/0257 →
PATENT SECURITY ASSIGNMENT AND ASSUMPTION AGREEMENT Recorded Dec 20, 2017
From: BIOPHARMA SECURED DEBT FUND II HOLDINGS CAYMAN LP
To: CPPIB CREDIT EUROPE S.À R.L.
Reel/Frame 044956/0395 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 5, 2013
From: MANKU, MEHAR; OSTERLOH, IAN; WICKER, PIERRE; BRAECKMAN, RENE; SONI, PARESH
To: AMARIN PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 030960/0014 →
SECURITY AGREEMENT Recorded Dec 19, 2012
From: AMARIN PHARMACEUTICALS IRELAND LIMITED
To: BIOPHARMA SECURED DEBT FUND II HOLDINGS CAYMAN LP
Reel/Frame 029499/0087 →