IP Library Granted Patent US 9,139,579
Granted Patent B2
US 9,139,579 · App. 13/544,321 · Granted Sep 22, 2015

Heteroaryl carboxamides

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Quick Facts
Patent No.
US 9,139,579
App. No.
13/544,321
Granted
Sep 22, 2015
Kind
B2
Abstract

The invention relates to novel heteroaryl carboxamides, a process for their preparation, and pharmaceutical compositions containing them. These materials are useful for the treatment and/or prophylaxis of diseases and for improving perception, concentration, learning and/or memory.

Claims (7)

1. A compound of the formula (I):

in which

R 1 is 1-azabicyclo[2.2.2]oct-3-yl,

the ring A is pyridazino,

and

R 2 and R 3 are identical or different and are radicals selected from the group of hydrogen, halogen, formyl, carbamoyl, cyano, trifluoromethyl, trifluoromethoxy, nitro, (C 1 -C 6 )-alkyl , (C 1 -C 6 )-alkoxy, (C 1 -C 6 )-alkylthio, (C 3 -C 8 )-cycloalkyl, 4- to 8-membered heterocyclyl, phenyl or 5- to 6-membered heteroaryl, where phenyl and heteroaryl are optionally substituted by halogen, (C 1 -C 4 )-alkyl, (C 1 -C 4 )-alkoxy, amino, mono- or di-(C 1 -C 4 )-alkylamino, (C 1 -C 4 )-alkanoylamino or (C 1 -C 4 ) -alkanesulfonylamino;

or a salt thereof.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 12, 2019
From: HENDRIX, MARTIN; BÖSS, FRANK-GERHARD; ERB, CHRISTINA; KRÜGER, JOACHIM; LUITHLE, JOACHIM; METHFESSEL, CHRISTOPH; SCHREIBER, RUDY; WIESE, WELF-BURKHARD
To: BAYER HEALTHCARE AG
Reel/Frame 049743/0070 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 12, 2019
From: BAYER PHARMA AKTIENGESELLSCHAFT
To: BAYER INTELLECTUAL PROPERTY GMBH
Reel/Frame 049743/0098 →
MERGER Recorded Jul 12, 2019
From: BAYER HEALTHCARE AG
To: BAYER SCHERING PHARMA AKTIENGESELLSCHAFT
Reel/Frame 049743/0577 →
CHANGE OF NAME Recorded Jul 12, 2019
From: BAYER SCHERING PHARMA AKTIENGESELLSCHAFT
To: BAYER PHARMA AKTIENGESELLSCHAFT
Reel/Frame 049743/0713 →