IP Library › Granted Patent US 9,144,573
Granted Patent B2
US 9,144,573 · App. 13/555,408 · Granted Sep 29, 2015

Prostaglandin transporter inhibitors

View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,144,573
App. No.
13/555,408
Granted
Sep 29, 2015
Kind
B2
Abstract

The present invention generally relates to prostaglandin transport. More specifically, the invention is directed to compounds that inhibit prostaglandin transport and subsequent COX-2 induction, and methods relating thereto.

Claims (11)

1. A compound having the structure:

wherein R1 is:

and wherein R2 is:

or a pharmaceutically acceptable salt, ester or tautomer thereof.

2. The compound of claim 1 having the structure:

or a pharmaceutically acceptable salt thereof.

3. The compound of claim 1 having the structure:

or a pharmaceutically acceptable salt thereof.

4. The compound of claim 2 which is:

5. The compound of claim 3 which is:

6. A composition comprising the compound of claim 1 in a pharmaceutically acceptable excipient.

Assignments (3)
MERGER AND CHANGE OF NAME Recorded Feb 26, 2019
From: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.; ALBERT EINSTEIN COLLEGE OF MEDICINE
To: ALBERT EINSTEIN COLLEGE OF MEDICINE
Reel/Frame 048438/0275 →
CHANGE OF NAME Recorded Oct 19, 2015
From: COM AFFILIATION, INC.
To: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.
Reel/Frame 036888/0682 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 15, 2015
From: ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY
To: COM AFFILIATION, INC.
Reel/Frame 036873/0672 →