IP Library Granted Patent US 8,686,019
Granted Patent B2
US 8,686,019 · App. 13/559,253 · Granted Apr 1, 2014

Use of amisulpride as an anti-emetic

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Quick Facts
Patent No.
US 8,686,019
App. No.
13/559,253
Granted
Apr 1, 2014
Kind
B2
Abstract

Amisulpride is used in the therapy of nausea, vomiting or retches. The therapy may utilize a novel injectable formulation, in unit dosage form, comprising less than 50 mg amisulpride.

Claims (24)

1. A method for the prevention and/or treatment of nausea and/or vomiting that is induced by chemotherapy or radiation wherein said method comprises administering, to a subject in need of such prevention and/or treatment, amisulpride at a dose of 1-40 mg in combination with another anti-emetic drug, wherein the subject is also administered an emetogenic chemotherapeutic agent or the subject receives radiation therapy.

2. The method according to claim 1 , wherein the subject is further administered another emetogenic agent.

3. The method according to claim 2 , wherein the subject has cancer.

4. The method according to claim 1 , wherein the chemotherapeutic emetogenic agent is cisplatin.

5. The method according to claim 2 , wherein said another emetogenic agent is an opiate.

6. The method according to claim 2 , wherein said another emetogenic agent is morphine.

7. The method according to claim 1 , wherein the amisulpride is administered by intravenous injection.

8. The method according to claim 1 , wherein the amisulpride is administered by intramuscular injection.

9. The method according to claim 1 , wherein the amisulpride is administered by subcutaneous injection.

10. The method according to claim 1 , wherein the amisulpride is administered by rectal administration.

11. The method according to claim 1 , wherein the amisulpride is administered by intranasal administration.

12. The method according to claim 1 , wherein the amisulpride is administered by buccal administration.

13. The method according to claim 1 , wherein the amisulpride is administered by oral, transdermal, sublingual or inhaled administration.

14. The method according to claim 1 , wherein the subject is a human.

15. The method according to claim 1 , wherein the amisulpride is in the form of an acceptable pharmaceutical salt.

16. The method according to claim 1 , wherein the another anti-emetic drug is a 5HT3 antagonist.

17. The method according to claim 16 , wherein the 5HT3 antagonist is ondansetron.

18. The method according to claim 1 , wherein the subject receives radiation therapy.

19. The method according to claim 2 , wherein amisulpride is administered simultaneously or sequentially with the emetogenic chemotherapeutic agent.

20. The method according to claim 2 , wherein amisulpride is administered before or after the administration of the emetogenic chemotherapeutic agent.

21. The method according claim 1 , wherein the amisulpride is administered at a dose of 2.5 mg to 20 mg.

22. The method according to claim 1 , wherein the amisulpride is administered at a dose of 5 to 35 mg.

23. The method according claim 1 , wherein the amisulpride is administered once or twice a day.

24. A method for the prevention and/or treatment of nausea and/or vomiting wherein said method comprises administering, to a subject in need of such prevention and/or treatment, amisulpride at a dose of 1-40 mg in combination with another anti-emetic drug, wherein the subject is also administered an emetogenic agent that is an opiate.

Assignments (7)
SECURITY INTEREST Recorded Apr 27, 2026
From: LXO IRELAND DESIGNATED ACTIVITY COMPANY
To: KROLL TRUSTEE SERVICES LIMITED, AS SECURITY AGENT
Reel/Frame 074483/0163 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 4, 2026
From: ACACIA PHARMA LIMITED; ACACIA PHARMA, INC.; EAGLE PHARMACEUTICALS, INC.
To: LXO IRELAND DESIGNATED ACTIVITY COMPANY; LXO US, INC.
Reel/Frame 073967/0303 →
RELEASE OF SECURITY INTEREST Recorded Apr 1, 2025
From: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
To: ACACIA PHARMA LIMITED
Reel/Frame 070698/0351 →
SECURITY INTEREST Recorded Apr 28, 2023
From: ACACIA PHARMA LIMITED
To: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 063476/0631 →
RELEASE OF SECURITY INTEREST Recorded Jul 5, 2018
From: SILICON VALLEY BANK
To: ACACIA PHARMA LIMITED
Reel/Frame 046273/0930 →
SECURITY AGREEMENT Recorded Feb 24, 2016
From: ACACIA PHARMA LIMITED
To: SILICON VALLEY BANK
Reel/Frame 037899/0594 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 15, 2012
From: GILBERT, JULIAN CLIVE; GRISTWOOD, ROBERT WILLIAM; COOPER, NICOLA; FOX, GABRIEL
To: ACACIA PHARMA LIMITED
Reel/Frame 029128/0552 →