IP Library Granted Patent US 8,653,144
Granted Patent B2
US 8,653,144 · App. 13/651,330 · Granted Feb 18, 2014

Treatment of pervasive developmental disorders with redox-active therapeutics

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Quick Facts
Patent No.
US 8,653,144
App. No.
13/651,330
Granted
Feb 18, 2014
Kind
B2
Abstract

Methods of treating or suppressing pervasive developmental disorders (PDDs) including; autistic disorder, Asperger's syndrome, childhood disintegrative disorder (CDD), Rett's disorder, and PDD-not otherwise specified (PDD-NOS) or attention deficit/hyperactivity disorder (ADHD) comprising administering to a subject in need thereof a therapeutically effective amount of one or more compounds as disclosed herein.

Claims (35)

1. A method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD) or attention deficit/hyperactivity disorder (ADHD) in a patient in need of such treatment, comprising administering to the patient a therapeutically or physiologically effective amount of a compound of Formula V,

wherein:

R 1 , R 2 , and R 3 are independently selected from the group consisting of H, (C 1 -C 6 )alkyl, (C 1 -C 6 )haloalkyl, (C 1 -C 6 )alkoxy, halogen and CN;

or a stereoisomer, a mixture of stereoisomers, a solvate or a hydrate thereof.

2. The method according to claim 1 , wherein the compound of Formula V has the formula:

or a solvate or a hydrate thereof.

3. The method according to claim 2 , wherein the compound is

4. The method according to claim 1 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is autistic spectrum disorder (ASD).

5. The method according to claim 2 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is autistic spectrum disorder (ASD).

6. The method according to claim 3 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is autistic spectrum disorder (ASD).

7. The method according to claim 1 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing attention deficit/hyperactivity disorder (ADHD).

8. The method according to claim 2 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing attention deficit/hyperactivity disorder (ADHD).

9. The method according to claim 3 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing attention deficit/hyperactivity disorder (ADHD).

10. The method of claim 4 , wherein the autistic spectrum disorder is autistic disorder.

11. The method of claim 5 , wherein the autistic spectrum disorder is autistic disorder.

12. The method of claim 6 , wherein the autistic spectrum disorder is autistic disorder.

13. The method of claim 1 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is Rett's disorder.

14. The method of claim 2 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is Rett's disorder.

15. The method of claim 3 , wherein the method is a method of reducing the symptoms associated with, or for treating or suppressing a pervasive developmental disorder (PDD), wherein the PDD is Rett's disorder.

16. The method according to claim 1 , wherein R 1 , R 2 , and R 3 are independently selected from (C 1 -C 4 ) alkyl.

17. The method according to claim 1 , wherein R 1 , R 2 , and R 3 are methyl.

18. The method according to claim 1 , wherein at least one of R 1 , R 2 , and R 3 is not methyl.

19. The method according to claim 1 , wherein R 1 and R 2 are independently selected from (C 1 -C 4 ) alkoxy, and R 3 is (C 1 -C 4 ) alkyl.

20. The method according to claim 1 , wherein R 1 and R 2 are methoxy, and R 3 is methyl.

21. The method according to claim 1 , wherein the compound is administered as a composition comprising at least one physiologically acceptable carrier, adjuvant, excipient, buffer, or diluent.

22. The method according to claim 2 , wherein the compound is administered as a composition comprising at least one physiologically acceptable carrier, adjuvant, excipient, buffer, or diluent.

23. The method according to claim 3 , wherein the compound is administered as a composition comprising at least one physiologically acceptable carrier, adjuvant, excipient, buffer, or diluent.

24. The method according to claim 1 , wherein the method comprises administering to the patient a food, medical food, functional food, food supplement, or dietary supplement comprising a composition comprising the compound and at least one physiologically or nutritionally acceptable carrier, adjuvant, excipient, buffer, or diluent.

25. The method according to claim 1 , wherein the method is a method for treating a pervasive developmental disorder (PDD) or attention deficit/hyperactivity disorder (ADHD).

26. The method according to claim 2 , wherein the method is a method for treating a pervasive developmental disorder (PDD) or attention deficit/hyperactivity disorder (ADHD).

27. The method according to claim 3 , wherein the method is a method for treating a pervasive developmental disorder (PDD) or attention deficit/hyperactivity disorder (ADHD).

28. The method of claim 4 , wherein the method is a method of treating autistic spectrum disorder (ASD).

29. The method of claim 6 , wherein the method is a method of treating autistic spectrum disorder (ASD).

30. The method of claim 13 , wherein the method is a method of treating Rett's disorder.

31. The method of claim 15 , wherein the method is a method of treating Rett's disorder.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 15, 2019
From: BIOELECTRON TECHNOLOGY CORPORATION
To: PTC THERAPEUTICS, INC.
Reel/Frame 051041/0478 →
CHANGE OF NAME Recorded Feb 8, 2017
From: EDISON PHARMACEUTICALS, INC.
To: BIOELECTRON TECHNOLOGY CORPORATION
Reel/Frame 041660/0644 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 17, 2012
From: MILLER, GUY M.; KHEIFETS, VIKTORIA
To: EDISON PHARMACEUTICALS, INC.
Reel/Frame 029147/0017 →