IP Library Granted Patent US 8,623,894
Granted Patent B2
US 8,623,894 · App. 13/714,911 · Granted Jan 7, 2014

Solid forms of N-[2,4-Bis(1,1-dimethyethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquioline-3-carboxamide

Inventors: John DeMattei (Berthoud, CO); Yushi Feng (Zionsville, IN); Cristian L. Harrison (Beverly, MA); Adam R. Looker (Cambridge, MA); Praveen Mudunuri (Waltham, MA); Stefanie Roeper (Medford, MA); Yuegang Zhang (Wayland, MA)
Assignee: Vertex Pharmaceuticals Incorporated
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Quick Facts
Patent No.
US 8,623,894
App. No.
13/714,911
Granted
Jan 7, 2014
Kind
B2
Abstract

Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide are described herein, including crystalline forms thereof.

Claims (3)

1. A method for treating a CFTR mediated disease in a mammal comprising administering a solid form of a compound selected from Compound 1.2-methylbutyric acid, Compound 1.propylene glycol, Compound 1.PEG 400.KOAc, Compound 1.lactic acid, Compound 1.isobutyric acid, Compound 1.propionic acid, Compound 1.2-propanol, Compound 1.besylate, and Compound 1.besylate.H 2 O, wherein said disease is selected from cystic fibrosis, hereditary emphysema, COPD, and dry-eye disease, and Compound 1 is N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide.

2. The method according to claim 1 , wherein said disease is cystic fibrosis.

3. The method according to claim 1 , further comprising administering an additional therapeutic agent.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded Oct 14, 2016
From: MACQUARIE US TRADING LLC
To: VERTEX PHARMACEUTICALS INCORPORATED; VERTEX PHARMACEUTICALS (SAN DIEGO) LLC
Reel/Frame 040357/0001 →
ASSIGNEE CHANGE OF ADDRESS Recorded Feb 17, 2016
From: VERTEX PHARMACEUTICALS INCORPORATED
To: VERTEX PHARMACEUTICALS INCORPORATED
Reel/Frame 037841/0274 →
SECURITY INTEREST Recorded Jul 10, 2014
From: VERTEX PHARMACEUTICALS INCORPORATED; VERTEX PHARMACEUTICALS (SAN DIEGO) LLC
To: MACQUARIE US TRADING LLC
Reel/Frame 033292/0311 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2013
From: DEMATTEI, JOHN; FENG, YUSHI; HARRISON, CRISTIAN; LOOKER, ADAM; MUDUNURI, PRAVEEN; ROEPER, STEFANIE; ZHANG, YUEGANG
To: VERTEX PHARMACEUTICALS INCORPORATED
Reel/Frame 030345/0600 →
Continuity (4)
Continuation 13413327 · Mar 6, 2012
Continuation 12283702 · Sep 15, 2008
Provisional Application 60972605 · Sep 14, 2007
Related Publication 20130109717A1 · May 2, 2013