IP Library Granted Patent US 9,114,136
Granted Patent B2
US 9,114,136 · App. 13/725,627 · Granted Aug 25, 2015

Treatment of progressive neurodegenerative disease with ibudilast

Inventors: Michael E. Kalafer (San Diego, CA); Kenneth W. Locke (Carlsbad, CA); Kazuko Matsuda (Beverly Hills, CA); Richard E. Gammans (Edmond, OK)
Assignee: MEDICINOVA, INC.
A61K31/437
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Quick Facts
Patent No.
US 9,114,136
App. No.
13/725,627
Granted
Aug 25, 2015
Kind
B2
Abstract

Compositions and methods for treating progressive neurodegenerative diseases, and their associated symptoms by administration of ibudilast (3-isobutyryl-2-isopropylpyrazolo[1,5-a]pyridine).

Claims (11)

1. A method of reducing brain volume loss in a patient diagnosed with a progressive form of multiple sclerosis, comprising administering to the patient in need thereof a therapeutically effective amount of ibudilast or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 which further comprises observing changes in the patient's cerebral MR or CT images to track changes in the patient's brain volume.

3. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least six months.

4. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least one year.

5. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least two years.

6. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered at least once daily.

7. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered orally.

8. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in an amount of 30 mg to 240 mg daily.

9. The method of claim 1 in which the progressive form of multiple sclerosis has progressed beyond relapse remitting multiple sclerosis.

10. The method of claim 9 in which the patient has been diagnosed with secondary progressive multiple sclerosis.

11. The method of claim 9 in which the patient has been diagnosed with primary progressive multiple sclerosis.

Continuity (5)
Continuation 13402702 · Feb 22, 2012
Continuation 12169042 · Jul 8, 2008
Provisional Application 60929745 · Jul 11, 2007
Provisional Application 61042181 · Apr 3, 2008
Related Publication 20130217718A1 · Aug 22, 2013