IP Library Granted Patent US 8,586,586
Granted Patent B2
US 8,586,586 · App. 13/791,059 · Granted Nov 19, 2013

Methods and compositions for treating or preventing erythema

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Quick Facts
Patent No.
US 8,586,586
App. No.
13/791,059
Granted
Nov 19, 2013
Kind
B2
Abstract

Methods and products for treating or preventing erythema or a symptom associated with erythema in a subject are described. The methods involve topically applying to an affected skin area a topical aqueous gel composition comprising about 0.01% to about 10% by weight of at least one α-adrenergic receptor agonist and a pharmaceutically acceptable carrier.

Claims (14)

1. A method of treating erythema or a symptom associated therewith in a subject, the method comprising topically administering to a skin area of the subject a topical composition comprising about 0.01% to about 10% by weight of at least one alpha adrenergic receptor agonist and a pharmaceutically acceptable carrier, wherein the skin area is, or is prone to be, affected by the erythema or the symptom associated therewith.

2. The method of claim 1 , wherein the topical composition is selected from the group consisting of an aqueous solution topical formulation, cream topical formulation, and ointment formulation.

3. The method of claim 1 , wherein the erythema is erythema of rosacea.

4. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is an agonist selective for an alpha 1-adrenergic receptor.

5. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is an agonist selective for an alpha 2-adrenergic receptor.

6. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is a non-selective alpha-adrenergic receptor agonist.

7. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is brimonidine.

8. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is oxymetazoline.

9. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is naphazoline.

10. The method of claim 1 , wherein the at least one alpha-adrenergic receptor agonist is selected from the group consisting of tetrahydrozoline, xylometazoline, phenylephrine, methoxamine, mephentermine, metaraminol, midodrine, epinephrine and norepinephrine.

11. The method of claim 1 , further comprising administering to the subject at least one additional treatment and medication for erythema or the symptom associated therewith.

12. The method of claim 1 , wherein the topical composition is administered to the skin area once daily.

13. The method of claim 1 , wherein the topical composition comprises about 0.1% to 3% by weight of the at least one alpha adrenergic receptor agonist.

14. The method of claim 1 , wherein the topical composition comprises about 0.05%-1% by weight of the at least one alpha adrenergic receptor agonist.

Assignments (4)
MERGER AND CHANGE OF NAME Recorded Mar 10, 2022
From: NESTLÉ SKIN HEALTH SA; GALDERMA HOLDINGS SA
To: GALDERMA HOLDING SA
Reel/Frame 060044/0523 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 22, 2021
From: GALDERMA LABORATORIES, INC.; GALDERMA LABORATORIES, L.P.
To: NESTLÉ SKIN HEALTH SA
Reel/Frame 058461/0396 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 7, 2014
From: GALDERMA LABORATORIES INC.
To: GALDERMA LABORATORIES, L.P.
Reel/Frame 033483/0127 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 11, 2013
From: GRAEBER, MICHAEL; LOESCHE, CHRISTIAN; FREIDENREICH, PHILIP; DEJOVIN, JACK A.; DEJOVIN, ISABELLE JEAN; LIU, YIN-SANG; LEONI, MATTHEW JAMES
To: GALDERMA LABORATORIES INC.
Reel/Frame 030198/0701 →