IP Library Granted Patent US 8,629,100
Granted Patent B2
US 8,629,100 · App. 13/950,202 · Granted Jan 14, 2014

Method of inhibiting clostridium difficile by administration of oritavancin

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Quick Facts
Patent No.
US 8,629,100
App. No.
13/950,202
Granted
Jan 14, 2014
Kind
B2
Abstract

Glycopeptide antibiotics, such as oritavancin, demonstrate significant activity against both a vegetative form of C. difficile and C. difficile spores. Methods for the treatment, prophylaxis and prevention of C. difficile infection and disease in animals, including humans, are described.

Claims (11)

1. A method of treating a C. difficile infection in a subject, comprising administering a therapeutically effective amount of a glycopeptide antibiotic to a subject having a C. difficile infection, thereby treating a C. difficile infection in a subject, wherein the glycopeptide antibiotic is oritavancin, or a pharmaceutically acceptable salt, hydrate, or solvate thereof, or a mixture thereof, and wherein the C. difficile infection comprises C. difficile spores or a mixture of C. difficile spores and C. difficile in vegetative form.

2. A method of treating a C. difficile infection in a subject, comprising administering a therapeutically effective amount of a glycopeptide antibiotic to a subject having a C. difficile infection, wherein said treatment inhibits C. difficile sporulation, thereby treating a C. difficile infection in a subject, wherein the glycopeptide antibiotic is oritavancin, or a pharmaceutically acceptable salt, hydrate, or solvate thereof, or a mixture thereof, and wherein the C. difficile infection comprises C. difficile spores or a mixture of C. difficile spores and C. difficile in vegetative form.

3. The method of claim 1 , wherein said treatment inhibits outgrowth of a C. difficile spore, inhibits growth of a vegetative form of C. difficile , or inhibits C. difficile sporulation.

4. The method of claim 1 , wherein the glycopeptide antibiotic is in the form of a pharmaceutical composition comprising the glycopeptide antibiotic and a pharmaceutically acceptable carrier or diluent.

5. The method of claim 1 , wherein said administering is via intravenous administration or oral administration.

6. The method of claim 1 , wherein the therapeutically effective amount of the glycopeptide antibiotic is between about 5 and 30 mg/kg body weight.

7. The method of claim 1 , wherein said administering is BID for four days.

8. The method of claim 2 , wherein the glycopeptide antibiotic is in the form of a pharmaceutical composition comprising the glycopeptide antibiotic and a pharmaceutically acceptable carrier or diluent.

9. The method of claim 2 , wherein said administering is via intravenous administration or oral administration.

10. The method of claim 2 , wherein the therapeutically effective amount of the glycopeptide antibiotic is between about 5 and 30 mg/kg body weight.

11. The method of claim 2 , wherein said administering is BID for four days.

Assignments (8)
TERMINATION AND RELEASE OF INTELLECTUAL PROPERTY SECURITY AGREEMENT (PATENTS) AT REEL 054836 AND FRAME 0765 AND REEL 061314 AND 0459 Recorded Aug 29, 2025
From: SILICON VALLEY BANK, A DIVISION OF FIRST-CITIZENS BANK & TRUST COMPANY
To: MELINTA THERAPEUTICS, LLC
Reel/Frame 072772/0097 →
AMENDED AND RESTATED INTELLECTUAL PROPERTY SECURITY AGREEMENT Recorded Aug 25, 2022
From: MELINTA THERAPEUTICS, LLC
To: SILICON VALLEY BANK
Reel/Frame 061314/0459 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2019
From: WILCOX, MARK HARVEY; BAINES, SIMON
To: UNIVERSITY OF LEEDS
Reel/Frame 048400/0254 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2019
From: LEHOUX, DARIO; PARR, THOMAS REEVES, JR
To: TARGANTA THERAPEUTICS CORP.
Reel/Frame 048400/0331 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2019
From: UNIVERSITY OF LEEDS
To: THE MEDICINES COMPANY
Reel/Frame 048400/0438 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2019
From: TARGANTA THERAPEUTICS CORP.
To: THE MEDICINES COMPANY
Reel/Frame 048400/0485 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2019
From: THE MEDICINES COMPANY
To: MELINTA THERAPEUTICS, INC.
Reel/Frame 048407/0911 →
SECURITY INTEREST Recorded Jan 8, 2018
From: MELINTA THERAPEUTICS, INC.; REMPEX PHARMACEUTICALS, INC.; CEMPRA PHARMACEUTICALS, INC.; CEM-102 PHARMACEUTICALS, INC.
To: CORTLAND CAPITAL MARKET SERVICES LLC, AS AGENT
Reel/Frame 045019/0552 →