IP Library Granted Patent US 9,675,565
Granted Patent B2
US 9,675,565 · App. 13/957,861 · Granted Jun 13, 2017

D3 dopamine receptor agonists to treat dyskinesia in parkinson's disease

Inventors: Sandhya Kortagere (Newtown, PA); Eldo V. Kuzhikandahil (Chester, NJ)
Assignees: Drexel University; Rutgers, The State University of New Jersey
A61K31/137A61K31/198A61K31/4045A61K31/4184A61K31/428A61K31/473A61K31/48A61K31/506A61K31/519A61K31/5513A61K45/06C07C211/29C07C215/08C07C215/54C07C217/62C07D209/14C07D235/16C07D471/04
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Quick Facts
Patent No.
US 9,675,565
App. No.
13/957,861
Granted
Jun 13, 2017
Kind
B2
Abstract

The present invention provides a method of inhibiting, suppressing or preventing levodopa-induced dyskinesia in a patient suffering from Parkinson's Disease, comprising the step of administering to the patient a pharmaceutical composition comprising at least one compound of the invention. The present invention further provides a method of inhibiting, suppressing or preventing Parkinson's Disease in a patient, comprising the step of administering to the patient a pharmaceutical composition comprising at least one compound of the invention.

Claims (21)

1. A pharmaceutical composition comprising at least one compound selected from the group consisting of:

2-amino-4-(2-chlorophenyl)butan-1-ol;

2-(3-aminohexyl)phenol;

4-(2-chlorophenyl)-butan-2-amine;

4-(2-chlorophenyl)-2-methylamino-butane;

4-(2-fluorophenyl)butan-2-amine;

4-(2-bromophenyl)butan-2-amine;

4-(2-iodophenyl)butan-2-amine;

4-(2-methoxyphenyl)butan-2-amine;

3-(3,4-diethoxyphenyl)propan-1-amine;

4-(4-chlorophenyl)butan-2-amine;

4-(4-methoxyphenyl)butan-2-amine;

any mixtures thereof; and any pharmaceutically acceptable salts thereof.

2. A compound selected from the group consisting of:

2-amino-4-(2-chlorophenyl)butan-1-ol;

2-(3-aminohexyl)phenol;

4-(2-iodophenyl)butan-2-amine;

4-(2-methoxyphenyl)butan-2-amine;

4-(4-chlorophenyl)butan-2-amine;

any mixtures thereof; and any pharmaceutically acceptable salts thereof.

3. A pharmaceutical composition comprising 4-(2-chlorophenyl)-butan-2-amine, or a pharmaceutically acceptable salt thereof.

Assignments (1)
MERGER Recorded Jan 14, 2015
From: PHILADELPHIA HEALTH & EDUCATION CORPORATION
To: DREXEL UNIVERSITY
Reel/Frame 034764/0236 →
Continuity (3)
Division 13764623
Provisional Application 61372733 · Aug 11, 2010
Related Publication 20140228380A1 · Aug 14, 2014