IP Library Granted Patent US 9,995,755
Granted Patent B2
US 9,995,755 · App. 14/021,947 · Granted Jun 12, 2018

Diagnosis and treatments relating to TH2 inhibition

Inventors: Joseph R. Arron (San Mateo, CA); Richard W. Erickson (Castro Valley, CA); Michelle Freemer (Mill Valley, CA); Meredith Hazen (Belmont, CA); Guiquan Jia (Foster City, CA); John G. Matthews (San Francisco, CA); Wendy Putnam (Belmont, CA); Heleen Scheerens (Menlo Park, CA); Yanan Zheng (Redwood City, CA)
Assignee: GENENTECH, INC.
G01N33/6884A61K31/522A61K31/573A61K39/3955A61K39/39566A61K45/06C07K16/18C07K16/28G01N33/6887G01N33/6893G01N2333/475G01N2800/122G01N2800/52
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Quick Facts
Patent No.
US 9,995,755
App. No.
14/021,947
Granted
Jun 12, 2018
Kind
B2
Abstract

Methods of diagnosing and treating disorders related to TH2 inhibition, including but not limited to asthma, are provided. Also provided are methods of selecting or identifying patients for treatment with certain therapeutic agents that are TH2 pathway inhibitors.

Claims (29)

1. A method of identifying an asthma patient or a respiratory disorder patient who is likely to suffer from severe exacerbations comprising determining whether the patient is Eosinophilic Inflammation Positive (EIP) using an Eosinophilic Inflammation Diagnostic Assay (EIDA), wherein the EIP status indicates that the patient is likely to suffer from an increase in severe exacerbations, and wherein the EIDA comprises the steps of:

a) determining the amount of Total Periostin in a sample obtained from an asthma patient or a respiratory disorder patient using (i) an antibody, which binds to periostin, comprising the sequences SEQ ID NO: 1 and SEQ ID NO: 2, or (ii) an antibody, which binds to periostin, comprising the sequences of SEQ ID NO: 3 and SEQ ID NO: 4, or (iii) both antibodies;

b) comparing the amount of Total Periostin determined in step a) to a reference amount; and

c) stratifying said patient into the category of likely to suffer from an increase in severe exacerbations or not likely to suffer from an increase in severe exacerbations based on the comparison obtained in step b).

2. A method of identifying an asthma patient or a respiratory disorder patient who is likely to suffer from severe exacerbations comprising determining whether the patient is Eosinophilic Inflammation Positive (EIP) using an Eosinophilic Inflammation Diagnostic Assay (EIDA), wherein the EIP status indicates that the patient is likely to suffer from an increase in severe exacerbations, and wherein the EIDA comprises the steps of:

a) determining the amount of Total Periostin in a sample obtained from an asthma patient or a respiratory disorder patient using an antibody, which binds to periostin, comprising the hypervariable region (“HVR”) sequences of SEQ ID NO: 1 and SEQ ID NO: 2;

b) comparing the amount of Total Periostin determined in step a) to a reference amount; and

c) stratifying said patient into the category of likely to suffer from an increase in severe exacerbations or not likely to suffer from an increase in severe exacerbations based on the comparison obtained in step b).

3. A method of identifying an asthma patient or a respiratory disorder patient who is likely to suffer from severe exacerbations comprising determining whether the patient is Eosinophilic Inflammation Positive (EIP) using an Eosinophilic Inflammation Diagnostic Assay (EIDA), wherein the EIP status indicates that the patient is likely to suffer from an increase in severe exacerbations, and wherein the EIDA comprises the steps of:

a) determining the amount of Total Periostin in a sample obtained from an asthma patient or a respiratory disorder patient using an antibody, which binds to periostin, comprising the hypervariable region (“HVR”) sequences of SEQ ID NO: 3 and SEQ ID NO: 4;

b) comparing the amount of Total Periostin determined in step a) to a reference amount; and

c) stratifying said patient into the category of likely to suffer from an increase in severe exacerbations or not likely to suffer from an increase in severe exacerbations based on the comparison obtained in step b).

4. A method of identifying an asthma patient or a respiratory disorder patient who is likely to suffer from severe exacerbations comprising determining whether the patient is Eosinophilic Inflammation Positive (EIP) using an Eosinophilic Inflammation Diagnostic Assay (EIDA), wherein the EIP status indicates that the patient is likely to suffer from an increase in severe exacerbations, and wherein the EIDA comprises the steps of:

a) determining the amount of Total Periostin in a sample obtained from an asthma patient or a respiratory disorder patient using (i) an antibody, which binds to periostin, comprising the hypervariable region (“HVR”) sequences of SEQ ID NO: 1 and SEQ ID NO: 2 and (ii) an antibody, which binds to periostin, comprising the hypervariable region (“HVR”) sequences of SEQ ID NO: 3 and SEQ ID NO: 4;

b) comparing the amount of Total Periostin determined in step a) to a reference amount; and

c) stratifying said patient into the category of likely to suffer from an increase in severe exacerbations or not likely to suffer from an increase in severe exacerbations based on the comparison obtained in step b).

5. The method according to any one of claims 1 - 4 , wherein the Total Periostin is serum periostin, which periostin is measured using an immunoassay.

6. The method according to claim 5 , wherein the immunoassay is a sandwich immunoassay.

7. The method according to claim 6 , wherein the sandwich immunoassay is an E4 Assay.

8. The method according to any one of claims 1 - 4 , wherein the reference amount for EIP is 23 ng/ml or greater when using an E4 Assay in step (a).

9. The method according to any one of claims 1 - 4 , wherein the reference amount for Eosinophilic Inflammation Negative (EIN) is 21 ng/ml or lower when using an E4 Assay in step (a).

10. The method according to any one of claims 1 - 4 , wherein the patient is suffering from moderate to severe asthma.

11. The method according to any one of claims 1 - 4 , wherein the asthma or respiratory disorder is uncontrolled on a first controller, wherein said first controller is a corticosteroid.

12. The method according to claim 11 , wherein the corticosteroid is an inhaled corticosteroid.

13. The method according to claim 12 , wherein the inhaled corticosteroid is beclomethasone dipropionate, budesonide, budesonide and formoterol, flunisolide, fluticasone propionate, fluticasone, or triamcinolone acetonide.

14. The method according to any one of claims 1 - 4 , wherein the patient is also being treated with a second controller.

15. The method according to claim 14 , wherein the second controller is a long acting bronchial dilator (LABD).

16. The method according to claim 15 , wherein the LABD is a long-acting beta-2 agonist (LABA), leukotriene receptor antagonist (LTRA), long-acting muscarinic antagonist (LAMA), theophylline, or oral corticosteroids (OCS).

17. The method according to claim 15 , wherein the LABD is budesonide and formoterol, fluticasone propionate, arformoterol, formoterol or salmeterol.

Continuity (7)
Division 13328830 · Dec 16, 2011
Provisional Application 61557295 · Nov 8, 2011
Provisional Application 61574485 · Aug 2, 2011
Provisional Application 61484650 · May 10, 2011
Provisional Application 61465425 · Mar 18, 2011
Provisional Application 61459760 · Dec 16, 2010
Related Publication 20140044702A1 · Feb 13, 2014